CO2026004110A2 - Método para producir selectivamente un compuesto axialmente quiral sencillo - Google Patents

Método para producir selectivamente un compuesto axialmente quiral sencillo

Info

Publication number
CO2026004110A2
CO2026004110A2 CONC2026/0004110A CO2026004110A CO2026004110A2 CO 2026004110 A2 CO2026004110 A2 CO 2026004110A2 CO 2026004110 A CO2026004110 A CO 2026004110A CO 2026004110 A2 CO2026004110 A2 CO 2026004110A2
Authority
CO
Colombia
Prior art keywords
formula
compound
salt
chiral compound
selectively producing
Prior art date
Application number
CONC2026/0004110A
Other languages
English (en)
Spanish (es)
Inventor
Kenichi Kawaguchi
Sunao Imada
Tomohiro Yoshinari
Eiji Kawaminami
Hiroki Ishioka
Junpei Ohtaka
Yuki Hirose
Original Assignee
Astellas Pharma Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Astellas Pharma Inc filed Critical Astellas Pharma Inc
Publication of CO2026004110A2 publication Critical patent/CO2026004110A2/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D405/00Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D451/00Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CONC2026/0004110A 2023-09-08 2026-03-30 Método para producir selectivamente un compuesto axialmente quiral sencillo CO2026004110A2 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
PCT/JP2023/032816 WO2025052649A1 (ja) 2023-09-08 2023-09-08 単一の軸不斉化合物の選択的製造法
PCT/JP2024/031959 WO2025053242A1 (ja) 2023-09-08 2024-09-06 単一の軸不斉化合物の選択的製造法

Publications (1)

Publication Number Publication Date
CO2026004110A2 true CO2026004110A2 (es) 2026-04-16

Family

ID=94923286

Family Applications (1)

Application Number Title Priority Date Filing Date
CONC2026/0004110A CO2026004110A2 (es) 2023-09-08 2026-03-30 Método para producir selectivamente un compuesto axialmente quiral sencillo

Country Status (7)

Country Link
JP (1) JP7700399B1 (https=)
CN (1) CN121843933A (https=)
AU (1) AU2024337896A1 (https=)
CO (1) CO2026004110A2 (https=)
MX (1) MX2026002723A (https=)
TW (1) TW202527939A (https=)
WO (2) WO2025052649A1 (https=)

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JOP20190186A1 (ar) * 2017-02-02 2019-08-01 Astellas Pharma Inc مركب كينازولين
WO2022173032A1 (ja) * 2021-02-15 2022-08-18 アステラス製薬株式会社 G12d変異krasタンパクの分解を誘導するためのキナゾリン化合物
EP4293025B1 (en) * 2021-02-15 2025-10-29 Astellas Pharma Inc. 4-aminoquinazoline compound
TW202346270A (zh) * 2022-03-11 2023-12-01 日商安斯泰來製藥股份有限公司 用於誘發g12d突變kras蛋白分解之雜環化合物
US20250145631A1 (en) * 2022-07-21 2025-05-08 Astellas Pharma Inc. Heterocyclic compound acting on g12d mutant kras protein
TW202412789A (zh) * 2022-08-05 2024-04-01 日商安斯泰來製藥股份有限公司 用於誘導突變kras蛋白分解之雜環化合物
EP4570794A1 (en) * 2022-08-09 2025-06-18 Astellas Pharma, Inc. Heterocyclic compound for inhibiting and/or inducing degradation of kras protein
EP4570795A1 (en) * 2022-08-09 2025-06-18 Astellas Pharma, Inc. Heterocyclic compound for inducing degradation of g12v mutant kras protein

Also Published As

Publication number Publication date
MX2026002723A (es) 2026-04-01
TW202527939A (zh) 2025-07-16
JP7700399B1 (ja) 2025-06-30
WO2025052649A1 (ja) 2025-03-13
WO2025053242A1 (ja) 2025-03-13
AU2024337896A1 (en) 2026-03-19
JPWO2025053242A1 (https=) 2025-03-13
CN121843933A (zh) 2026-04-10

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