JP7605579B2 - フッ素置換シクロプロピルアミン系化合物並びにその製造方法、薬物組成物及び使用 - Google Patents

フッ素置換シクロプロピルアミン系化合物並びにその製造方法、薬物組成物及び使用 Download PDF

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JP7605579B2
JP7605579B2 JP2018548895A JP2018548895A JP7605579B2 JP 7605579 B2 JP7605579 B2 JP 7605579B2 JP 2018548895 A JP2018548895 A JP 2018548895A JP 2018548895 A JP2018548895 A JP 2018548895A JP 7605579 B2 JP7605579 B2 JP 7605579B2
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JP2019515878A (ja
JP2019515878A5 (https=
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ホン リュウ
ジア リ
ジアン ワン
ミンボ ス
シュニ ワン
ユボ ヂョウ
ウェイ ヂュ
ウェイ シュ
チュンプ リ
フアリャン ジアン
カイシャン チェン
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シャンハイ インスティチュート オブ マテリア メディカ，チャイニーズ アカデミー オブ サイエンシーズ
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • A61K31/5375—1,4-Oxazines, e.g. morpholine
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    • C07D211/40—Oxygen atoms
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
JP2018548895A 2016-03-16 2017-03-16 フッ素置換シクロプロピルアミン系化合物並びにその製造方法、薬物組成物及び使用 Active JP7605579B2 (ja)

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CN201610149958.6 2016-03-16
CN201610149958.6A CN107200706A (zh) 2016-03-16 2016-03-16 一类氟取代的环丙胺类化合物及其制备方法、药物组合物和用途
PCT/CN2017/076967 WO2017157322A1 (zh) 2016-03-16 2017-03-16 一类氟取代的环丙胺类化合物及其制备方法、药物组合物和用途

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JP2019515878A5 JP2019515878A5 (https=) 2022-03-09
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JP7605579B2 true JP7605579B2 (ja) 2024-12-24

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KR102479789B1 (ko) 2016-05-09 2022-12-22 주빌런트 에피코어 엘엘씨 이중 lsd1/hdac 억제제로서 사이클로프로필-아마이드 화합물
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