JP7205529B2 - オキサゾリジノン化合物の製造方法 - Google Patents

オキサゾリジノン化合物の製造方法 Download PDF

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Publication number
JP7205529B2
JP7205529B2 JP2020501763A JP2020501763A JP7205529B2 JP 7205529 B2 JP7205529 B2 JP 7205529B2 JP 2020501763 A JP2020501763 A JP 2020501763A JP 2020501763 A JP2020501763 A JP 2020501763A JP 7205529 B2 JP7205529 B2 JP 7205529B2
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compound
mol
mixture
acetonitrile
hours
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Japanese (ja)
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JPWO2019163731A1 (ja
Inventor
敏彦 秋山
優花 大倉
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Sumitomo Chemical Co Ltd
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Sumitomo Chemical Co Ltd
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2020501763A 2018-02-26 2019-02-19 オキサゾリジノン化合物の製造方法 Active JP7205529B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2018031603 2018-02-26
JP2018031603 2018-02-26
PCT/JP2019/005969 WO2019163731A1 (ja) 2018-02-26 2019-02-19 オキサゾリジノン化合物の製造方法

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JPWO2019163731A1 JPWO2019163731A1 (ja) 2021-02-04
JP7205529B2 true JP7205529B2 (ja) 2023-01-17

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JP2020501763A Active JP7205529B2 (ja) 2018-02-26 2019-02-19 オキサゾリジノン化合物の製造方法

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JP (1) JP7205529B2 (zh)
CN (1) CN111699184B (zh)
IL (1) IL275443B (zh)
TW (1) TW201936603A (zh)
WO (1) WO2019163731A1 (zh)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP7339754B2 (ja) * 2019-03-27 2023-09-06 ダイト株式会社 中間体の製造方法
CN111039937B (zh) * 2019-12-16 2021-08-31 浙江海翔药业股份有限公司 一种利伐沙班中间体的制备方法

Citations (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2005524660A (ja) 2002-02-25 2005-08-18 ファルマシア・アンド・アップジョン・カンパニー・エルエルシー Ｎ−アリール−２−オキサゾリジノン−５−カルボキサミドおよびその誘導体ならびに抗細菌剤としてのそれらの使用
JP2007517816A (ja) 2004-01-15 2007-07-05 バイエル・ヘルスケア・アクチェンゲゼルシャフト 製造方法
JP2010530385A (ja) 2007-06-20 2010-09-09 バイエル・シェーリング・ファルマ・アクチェンゲゼルシャフト 置換オキサゾリジノン類およびそれらの使用
CN104031036A (zh) 2014-05-16 2014-09-10 南通常佑药业科技有限公司 一种利伐沙班的制备方法
WO2014155259A2 (en) 2013-03-25 2014-10-02 Glenmark Pharmaceuticals Limited; Glenmark Generics Limited Process for the preparation of rivaroxaban
US20150038704A1 (en) 2012-02-24 2015-02-05 China National Medicines Guorui Pharmaceutical Co. Method for preparing rivaroxaban intermediate

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2016199027A1 (en) * 2015-06-08 2016-12-15 Mehta Api Pvt. Ltd. An improved process for preparation of rivaroxaban

Patent Citations (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2005524660A (ja) 2002-02-25 2005-08-18 ファルマシア・アンド・アップジョン・カンパニー・エルエルシー Ｎ−アリール−２−オキサゾリジノン−５−カルボキサミドおよびその誘導体ならびに抗細菌剤としてのそれらの使用
JP2007517816A (ja) 2004-01-15 2007-07-05 バイエル・ヘルスケア・アクチェンゲゼルシャフト 製造方法
JP2010530385A (ja) 2007-06-20 2010-09-09 バイエル・シェーリング・ファルマ・アクチェンゲゼルシャフト 置換オキサゾリジノン類およびそれらの使用
US20150038704A1 (en) 2012-02-24 2015-02-05 China National Medicines Guorui Pharmaceutical Co. Method for preparing rivaroxaban intermediate
WO2014155259A2 (en) 2013-03-25 2014-10-02 Glenmark Pharmaceuticals Limited; Glenmark Generics Limited Process for the preparation of rivaroxaban
CN104031036A (zh) 2014-05-16 2014-09-10 南通常佑药业科技有限公司 一种利伐沙班的制备方法

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
FATTAH, Tanzeela A. et al.，A review on the synthetic approaches of rivaroxaban: An anticoagulant drug，Tetrahedron: Asymmetry，2017年，Vol.28, No.4，pp.485-504，DOI: 10.1016/j.tetasy.2017.02.010

Also Published As

Publication number Publication date
WO2019163731A1 (ja) 2019-08-29
TW201936603A (zh) 2019-09-16
CN111699184A (zh) 2020-09-22
IL275443B (en) 2022-07-01
CN111699184B (zh) 2023-05-23
IL275443A (en) 2020-08-31
JPWO2019163731A1 (ja) 2021-02-04

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