JP7150213B2 - アゾール誘導体、アゾール誘導体の製造方法、ならびに農園芸用薬剤 - Google Patents

アゾール誘導体、アゾール誘導体の製造方法、ならびに農園芸用薬剤 Download PDF

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JP7150213B2
JP7150213B2 JP2022504475A JP2022504475A JP7150213B2 JP 7150213 B2 JP7150213 B2 JP 7150213B2 JP 2022504475 A JP2022504475 A JP 2022504475A JP 2022504475 A JP2022504475 A JP 2022504475A JP 7150213 B2 JP7150213 B2 JP 7150213B2
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azole derivative
compound
group
added
methyl
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JPWO2021177442A1 (https=
JPWO2021177442A5 (https=
Inventor
大河 正野
勉 百足
朋之 高下
泰司 三宅
淳也 平田
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Kureha Corp
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Kureha Corp
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    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01PBIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P3/00Fungicides
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/501,3-Diazoles; Hydrogenated 1,3-diazoles
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/64Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
    • A01N43/647Triazoles; Hydrogenated triazoles
    • A01N43/6531,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/02Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having no bond to a nitrogen atom
    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01PBIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
    • A01P1/00Disinfectants; Antimicrobial compounds or mixtures thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D233/00Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/56Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
    • C07D233/60Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms with hydrocarbon radicals, substituted by oxygen or sulfur atoms, attached to ring nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D249/00Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/081,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02ATECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

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  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Engineering & Computer Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Wood Science & Technology (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Dentistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Microbiology (AREA)
  • Mycology (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
JP2022504475A 2020-03-06 2021-03-05 アゾール誘導体、アゾール誘導体の製造方法、ならびに農園芸用薬剤 Active JP7150213B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
JP2020039353 2020-03-06
JP2020039353 2020-03-06
PCT/JP2021/008690 WO2021177442A1 (ja) 2020-03-06 2021-03-05 アゾール誘導体、アゾール誘導体の製造方法、ならびに農園芸用薬剤および工業用材料保護剤

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JPWO2021177442A1 JPWO2021177442A1 (https=) 2021-09-10
JPWO2021177442A5 JPWO2021177442A5 (https=) 2022-08-17
JP7150213B2 true JP7150213B2 (ja) 2022-10-07

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Country Status (19)

Country Link
US (1) US20230192630A1 (https=)
EP (1) EP4116292A1 (https=)
JP (1) JP7150213B2 (https=)
KR (1) KR102497895B1 (https=)
CN (1) CN115052863B (https=)
AR (1) AR121486A1 (https=)
AU (1) AU2021230953B2 (https=)
BR (1) BR112022017644B1 (https=)
CA (1) CA3170548A1 (https=)
CL (1) CL2022002418A1 (https=)
CO (1) CO2022013071A2 (https=)
CR (1) CR20220440A (https=)
EC (1) ECSP22077395A (https=)
IL (1) IL295773B2 (https=)
MX (1) MX2022010857A (https=)
NZ (1) NZ792521A (https=)
PH (1) PH12022552096A1 (https=)
UA (1) UA127256C2 (https=)
WO (1) WO2021177442A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2023033180A1 (ja) * 2021-09-06 2023-03-09 株式会社クレハ アゾール誘導体のr-エナンチオマー、農園芸用薬剤および工業用材料保護剤
CN114262250A (zh) * 2021-12-24 2022-04-01 乐威医药(江苏)股份有限公司 芳香环苄基邻位双烷基的合成方法
CN119504731A (zh) * 2024-11-14 2025-02-25 广东省科学院测试分析研究所(中国广州分析测试中心) 一类含1,3,4-噁二唑酰腙结构的柚皮素衍生物及其制备方法

Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2012501294A (ja) 2008-08-26 2012-01-19 株式会社クレハ 5−ベンジル−4−アゾリルメチル−4−スピロ[2.4]ヘプタノール誘導体、その製造方法、農園芸用薬剤および工業用材料保護剤
WO2012169516A1 (ja) 2011-06-07 2012-12-13 株式会社クレハ アゾール誘導体、その製造方法、中間体化合物、ならびに農園芸用薬剤および工業用材料保護剤
JP2014520832A (ja) 2011-07-13 2014-08-25 ビーエーエスエフ ソシエタス・ヨーロピア 殺菌性置換2−[2−ハロゲンアルキル−4−(フェノキシ)−フェニル]−1−[1,2,4]トリアゾール−1−イル−エタノール化合物
WO2019093522A1 (ja) 2017-11-13 2019-05-16 株式会社クレハ アゾール誘導体、中間体化合物、及びアゾール誘導体の製造方法、ならびに農園芸用薬剤及び工業用材料保護剤

Family Cites Families (7)

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US4413003A (en) * 1977-07-29 1983-11-01 Rohm And Haas Company β-Hydroxyarylethylimidazoles
DE3608144A1 (de) * 1986-03-12 1987-09-24 Hoechst Ag Aryl-azolylmethyl-benzocycloalken-derivate, verfahren zu ihrer herstellung und ihre verwendung
GB8705174D0 (en) * 1987-03-05 1987-04-08 Ici Plc Heterocyclic compounds
JP4161331B2 (ja) * 1997-09-02 2008-10-08 株式会社クレハ アゾリルメチルビシクロヘキサノール誘導体、その製造方法及び、農薬並びに、医薬としての利用
US20030166476A1 (en) 2002-01-31 2003-09-04 Winemiller Mark D. Lubricating oil compositions with improved friction properties
UA108867C2 (uk) * 2009-12-08 2015-06-25 Похідні азолу, спосіб їх одержання (варіанти), проміжні продукти, засіб для сільського господарства і садівництва
KR101464420B1 (ko) * 2009-12-08 2014-11-21 가부시끼가이샤 구레하 아졸 유도체 및 그의 제조 방법, 상기 유도체의 중간체 화합물 및 그의 제조 방법, 및 상기 유도체를 함유하는 농원예용 약제 및 공업용 재료 보호제

Patent Citations (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2012501294A (ja) 2008-08-26 2012-01-19 株式会社クレハ 5−ベンジル−4−アゾリルメチル−4−スピロ[2.4]ヘプタノール誘導体、その製造方法、農園芸用薬剤および工業用材料保護剤
WO2012169516A1 (ja) 2011-06-07 2012-12-13 株式会社クレハ アゾール誘導体、その製造方法、中間体化合物、ならびに農園芸用薬剤および工業用材料保護剤
JP2014520832A (ja) 2011-07-13 2014-08-25 ビーエーエスエフ ソシエタス・ヨーロピア 殺菌性置換2−[2−ハロゲンアルキル−4−(フェノキシ)−フェニル]−1−[1,2,4]トリアゾール−1−イル−エタノール化合物
WO2019093522A1 (ja) 2017-11-13 2019-05-16 株式会社クレハ アゾール誘導体、中間体化合物、及びアゾール誘導体の製造方法、ならびに農園芸用薬剤及び工業用材料保護剤

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Publication number Publication date
WO2021177442A1 (ja) 2021-09-10
CA3170548A1 (en) 2021-09-10
CN115052863A (zh) 2022-09-13
BR112022017644A2 (pt) 2022-10-18
AU2021230953B2 (en) 2022-10-06
CR20220440A (es) 2022-12-06
MX2022010857A (es) 2023-03-14
EP4116292A1 (en) 2023-01-11
PH12022552096A1 (en) 2023-11-29
JPWO2021177442A1 (https=) 2021-09-10
AU2021230953A1 (en) 2022-09-22
IL295773B2 (en) 2023-04-01
IL295773A (en) 2022-10-01
US20230192630A1 (en) 2023-06-22
KR20220129652A (ko) 2022-09-23
NZ792521A (en) 2023-01-27
ECSP22077395A (es) 2022-11-30
BR112022017644B1 (pt) 2023-05-02
IL295773B (en) 2022-12-01
CN115052863B (zh) 2023-04-28
CL2022002418A1 (es) 2023-04-14
CO2022013071A2 (es) 2022-09-20
KR102497895B1 (ko) 2023-02-08
AR121486A1 (es) 2022-06-08
UA127256C2 (uk) 2023-06-21

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