JP7150213B2 - アゾール誘導体、アゾール誘導体の製造方法、ならびに農園芸用薬剤 - Google Patents
アゾール誘導体、アゾール誘導体の製造方法、ならびに農園芸用薬剤 Download PDFInfo
- Publication number
- JP7150213B2 JP7150213B2 JP2022504475A JP2022504475A JP7150213B2 JP 7150213 B2 JP7150213 B2 JP 7150213B2 JP 2022504475 A JP2022504475 A JP 2022504475A JP 2022504475 A JP2022504475 A JP 2022504475A JP 7150213 B2 JP7150213 B2 JP 7150213B2
- Authority
- JP
- Japan
- Prior art keywords
- azole derivative
- compound
- group
- added
- methyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Active
Links
Classifications
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
- A01P3/00—Fungicides
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/50—1,3-Diazoles; Hydrogenated 1,3-diazoles
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/64—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with three nitrogen atoms as the only ring hetero atoms
- A01N43/647—Triazoles; Hydrogenated triazoles
- A01N43/653—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
- A01N47/02—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having no bond to a nitrogen atom
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01P—BIOCIDAL, PEST REPELLANT, PEST ATTRACTANT OR PLANT GROWTH REGULATORY ACTIVITY OF CHEMICAL COMPOUNDS OR PREPARATIONS
- A01P1/00—Disinfectants; Antimicrobial compounds or mixtures thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
- C07D233/60—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms with hydrocarbon radicals, substituted by oxygen or sulfur atoms, attached to ring nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change
Landscapes
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Environmental Sciences (AREA)
- Zoology (AREA)
- Engineering & Computer Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Wood Science & Technology (AREA)
- Agronomy & Crop Science (AREA)
- General Health & Medical Sciences (AREA)
- Dentistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Microbiology (AREA)
- Mycology (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2020039353 | 2020-03-06 | ||
| JP2020039353 | 2020-03-06 | ||
| PCT/JP2021/008690 WO2021177442A1 (ja) | 2020-03-06 | 2021-03-05 | アゾール誘導体、アゾール誘導体の製造方法、ならびに農園芸用薬剤および工業用材料保護剤 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JPWO2021177442A1 JPWO2021177442A1 (https=) | 2021-09-10 |
| JPWO2021177442A5 JPWO2021177442A5 (https=) | 2022-08-17 |
| JP7150213B2 true JP7150213B2 (ja) | 2022-10-07 |
Family
ID=77614085
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2022504475A Active JP7150213B2 (ja) | 2020-03-06 | 2021-03-05 | アゾール誘導体、アゾール誘導体の製造方法、ならびに農園芸用薬剤 |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US20230192630A1 (https=) |
| EP (1) | EP4116292A1 (https=) |
| JP (1) | JP7150213B2 (https=) |
| KR (1) | KR102497895B1 (https=) |
| CN (1) | CN115052863B (https=) |
| AR (1) | AR121486A1 (https=) |
| AU (1) | AU2021230953B2 (https=) |
| BR (1) | BR112022017644B1 (https=) |
| CA (1) | CA3170548A1 (https=) |
| CL (1) | CL2022002418A1 (https=) |
| CO (1) | CO2022013071A2 (https=) |
| CR (1) | CR20220440A (https=) |
| EC (1) | ECSP22077395A (https=) |
| IL (1) | IL295773B2 (https=) |
| MX (1) | MX2022010857A (https=) |
| NZ (1) | NZ792521A (https=) |
| PH (1) | PH12022552096A1 (https=) |
| UA (1) | UA127256C2 (https=) |
| WO (1) | WO2021177442A1 (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2023033180A1 (ja) * | 2021-09-06 | 2023-03-09 | 株式会社クレハ | アゾール誘導体のr-エナンチオマー、農園芸用薬剤および工業用材料保護剤 |
| CN114262250A (zh) * | 2021-12-24 | 2022-04-01 | 乐威医药(江苏)股份有限公司 | 芳香环苄基邻位双烷基的合成方法 |
| CN119504731A (zh) * | 2024-11-14 | 2025-02-25 | 广东省科学院测试分析研究所(中国广州分析测试中心) | 一类含1,3,4-噁二唑酰腙结构的柚皮素衍生物及其制备方法 |
Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2012501294A (ja) | 2008-08-26 | 2012-01-19 | 株式会社クレハ | 5−ベンジル−4−アゾリルメチル−4−スピロ[2.4]ヘプタノール誘導体、その製造方法、農園芸用薬剤および工業用材料保護剤 |
| WO2012169516A1 (ja) | 2011-06-07 | 2012-12-13 | 株式会社クレハ | アゾール誘導体、その製造方法、中間体化合物、ならびに農園芸用薬剤および工業用材料保護剤 |
| JP2014520832A (ja) | 2011-07-13 | 2014-08-25 | ビーエーエスエフ ソシエタス・ヨーロピア | 殺菌性置換2−[2−ハロゲンアルキル−4−(フェノキシ)−フェニル]−1−[1,2,4]トリアゾール−1−イル−エタノール化合物 |
| WO2019093522A1 (ja) | 2017-11-13 | 2019-05-16 | 株式会社クレハ | アゾール誘導体、中間体化合物、及びアゾール誘導体の製造方法、ならびに農園芸用薬剤及び工業用材料保護剤 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4413003A (en) * | 1977-07-29 | 1983-11-01 | Rohm And Haas Company | β-Hydroxyarylethylimidazoles |
| DE3608144A1 (de) * | 1986-03-12 | 1987-09-24 | Hoechst Ag | Aryl-azolylmethyl-benzocycloalken-derivate, verfahren zu ihrer herstellung und ihre verwendung |
| GB8705174D0 (en) * | 1987-03-05 | 1987-04-08 | Ici Plc | Heterocyclic compounds |
| JP4161331B2 (ja) * | 1997-09-02 | 2008-10-08 | 株式会社クレハ | アゾリルメチルビシクロヘキサノール誘導体、その製造方法及び、農薬並びに、医薬としての利用 |
| US20030166476A1 (en) | 2002-01-31 | 2003-09-04 | Winemiller Mark D. | Lubricating oil compositions with improved friction properties |
| UA108867C2 (uk) * | 2009-12-08 | 2015-06-25 | Похідні азолу, спосіб їх одержання (варіанти), проміжні продукти, засіб для сільського господарства і садівництва | |
| KR101464420B1 (ko) * | 2009-12-08 | 2014-11-21 | 가부시끼가이샤 구레하 | 아졸 유도체 및 그의 제조 방법, 상기 유도체의 중간체 화합물 및 그의 제조 방법, 및 상기 유도체를 함유하는 농원예용 약제 및 공업용 재료 보호제 |
-
2021
- 2021-03-01 AR ARP210100533A patent/AR121486A1/es not_active Application Discontinuation
- 2021-03-05 PH PH1/2022/552096A patent/PH12022552096A1/en unknown
- 2021-03-05 MX MX2022010857A patent/MX2022010857A/es unknown
- 2021-03-05 BR BR112022017644-9A patent/BR112022017644B1/pt not_active IP Right Cessation
- 2021-03-05 IL IL295773A patent/IL295773B2/en unknown
- 2021-03-05 CN CN202180012657.8A patent/CN115052863B/zh not_active Expired - Fee Related
- 2021-03-05 CA CA3170548A patent/CA3170548A1/en active Pending
- 2021-03-05 NZ NZ792521A patent/NZ792521A/en not_active IP Right Cessation
- 2021-03-05 JP JP2022504475A patent/JP7150213B2/ja active Active
- 2021-03-05 US US17/905,446 patent/US20230192630A1/en not_active Abandoned
- 2021-03-05 AU AU2021230953A patent/AU2021230953B2/en not_active Ceased
- 2021-03-05 UA UAA202203641A patent/UA127256C2/uk unknown
- 2021-03-05 EP EP21765257.7A patent/EP4116292A1/en not_active Withdrawn
- 2021-03-05 WO PCT/JP2021/008690 patent/WO2021177442A1/ja not_active Ceased
- 2021-03-05 CR CR20220440A patent/CR20220440A/es unknown
- 2021-03-05 KR KR1020227030308A patent/KR102497895B1/ko active Active
-
2022
- 2022-09-05 CL CL2022002418A patent/CL2022002418A1/es unknown
- 2022-09-14 CO CONC2022/0013071A patent/CO2022013071A2/es unknown
- 2022-10-03 EC ECSENADI202277395A patent/ECSP22077395A/es unknown
Patent Citations (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2012501294A (ja) | 2008-08-26 | 2012-01-19 | 株式会社クレハ | 5−ベンジル−4−アゾリルメチル−4−スピロ[2.4]ヘプタノール誘導体、その製造方法、農園芸用薬剤および工業用材料保護剤 |
| WO2012169516A1 (ja) | 2011-06-07 | 2012-12-13 | 株式会社クレハ | アゾール誘導体、その製造方法、中間体化合物、ならびに農園芸用薬剤および工業用材料保護剤 |
| JP2014520832A (ja) | 2011-07-13 | 2014-08-25 | ビーエーエスエフ ソシエタス・ヨーロピア | 殺菌性置換2−[2−ハロゲンアルキル−4−(フェノキシ)−フェニル]−1−[1,2,4]トリアゾール−1−イル−エタノール化合物 |
| WO2019093522A1 (ja) | 2017-11-13 | 2019-05-16 | 株式会社クレハ | アゾール誘導体、中間体化合物、及びアゾール誘導体の製造方法、ならびに農園芸用薬剤及び工業用材料保護剤 |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2021177442A1 (ja) | 2021-09-10 |
| CA3170548A1 (en) | 2021-09-10 |
| CN115052863A (zh) | 2022-09-13 |
| BR112022017644A2 (pt) | 2022-10-18 |
| AU2021230953B2 (en) | 2022-10-06 |
| CR20220440A (es) | 2022-12-06 |
| MX2022010857A (es) | 2023-03-14 |
| EP4116292A1 (en) | 2023-01-11 |
| PH12022552096A1 (en) | 2023-11-29 |
| JPWO2021177442A1 (https=) | 2021-09-10 |
| AU2021230953A1 (en) | 2022-09-22 |
| IL295773B2 (en) | 2023-04-01 |
| IL295773A (en) | 2022-10-01 |
| US20230192630A1 (en) | 2023-06-22 |
| KR20220129652A (ko) | 2022-09-23 |
| NZ792521A (en) | 2023-01-27 |
| ECSP22077395A (es) | 2022-11-30 |
| BR112022017644B1 (pt) | 2023-05-02 |
| IL295773B (en) | 2022-12-01 |
| CN115052863B (zh) | 2023-04-28 |
| CL2022002418A1 (es) | 2023-04-14 |
| CO2022013071A2 (es) | 2022-09-20 |
| KR102497895B1 (ko) | 2023-02-08 |
| AR121486A1 (es) | 2022-06-08 |
| UA127256C2 (uk) | 2023-06-21 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| KR102148124B1 (ko) | 아졸 유도체, 중간체 화합물 및 아졸 유도체의 제조 방법, 및 농원예용 약제 및 공업용 재료 보호제 | |
| JP6942284B2 (ja) | 農園芸用殺菌剤、植物病害防除方法及び植物病害防除用製品 | |
| WO2021230382A1 (ja) | トリアゾール誘導体の(-)-エナンチオマー、農園芸用薬剤および工業用材料保護剤 | |
| JP7150213B2 (ja) | アゾール誘導体、アゾール誘導体の製造方法、ならびに農園芸用薬剤 | |
| JP2019031463A (ja) | アゾール誘導体、およびその農園芸用薬剤としての利用 | |
| WO2010074021A1 (ja) | 置換1-(1-クロロシクロプロピル)-2-(1h-1,2,4-トリアゾール-1-イル)-2-プロペン-1-オール誘導体、その製造方法、これを含有する農園芸用薬剤及び工業用材料保護剤 | |
| JP2020186178A (ja) | 農園芸用薬剤、植物病害防除方法、及び植物病害防除用製品 | |
| JP2025519412A (ja) | 4-[(6-クロロ-3-ピリジルメチル)(2,2-ジフルオロエチル)アミノ]フラン-2(5h)-オンの結晶形態aを含む農薬製剤 | |
| JP2023138105A (ja) | 農園芸用殺菌剤、植物病害防除方法及び植物病害防除用製品 | |
| JP2021014437A (ja) | アゾール誘導体、ならびに農園芸用薬剤および工業用材料保護剤 | |
| JP2021080280A (ja) | 農園芸用病害防除剤及び植物病害の防除方法 | |
| WO2023033180A1 (ja) | アゾール誘導体のr-エナンチオマー、農園芸用薬剤および工業用材料保護剤 | |
| JP2020180055A (ja) | アゾール誘導体、ならびに農園芸用薬剤および工業用材料保護剤 | |
| WO2025089146A1 (ja) | ピラゾール誘導体、またはその許容可能な塩もしくはそのn-オキシド、ならびに農園芸用薬剤および工業用材料保護剤 | |
| NZ762344B2 (en) | Azole derivative, intermediate compound, method for producing azole derivative, agricultural or horticultural chemical agent, and protective agent for industrial material | |
| BR112020002160B1 (pt) | Derivado de azol, composto intermediário, método para produção de derivado de azol, agente químico agrícola ou hortícola e agente protetor para material industrial, método para controlar uma doença em uma planta, semente revestida e uso do composto | |
| JP2016033127A (ja) | 農園芸用薬剤 |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| A521 | Request for written amendment filed |
Free format text: JAPANESE INTERMEDIATE CODE: A523 Effective date: 20220524 |
|
| A621 | Written request for application examination |
Free format text: JAPANESE INTERMEDIATE CODE: A621 Effective date: 20220524 |
|
| A871 | Explanation of circumstances concerning accelerated examination |
Free format text: JAPANESE INTERMEDIATE CODE: A871 Effective date: 20220524 |
|
| A131 | Notification of reasons for refusal |
Free format text: JAPANESE INTERMEDIATE CODE: A131 Effective date: 20220705 |
|
| A521 | Request for written amendment filed |
Free format text: JAPANESE INTERMEDIATE CODE: A523 Effective date: 20220818 |
|
| TRDD | Decision of grant or rejection written | ||
| A01 | Written decision to grant a patent or to grant a registration (utility model) |
Free format text: JAPANESE INTERMEDIATE CODE: A01 Effective date: 20220906 |
|
| A61 | First payment of annual fees (during grant procedure) |
Free format text: JAPANESE INTERMEDIATE CODE: A61 Effective date: 20220927 |
|
| R150 | Certificate of patent or registration of utility model |
Ref document number: 7150213 Country of ref document: JP Free format text: JAPANESE INTERMEDIATE CODE: R150 |