JP6820254B2 - 治療用化合物およびその使用 - Google Patents

治療用化合物およびその使用 Download PDF

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JP6820254B2
JP6820254B2 JP2017518804A JP2017518804A JP6820254B2 JP 6820254 B2 JP6820254 B2 JP 6820254B2 JP 2017518804 A JP2017518804 A JP 2017518804A JP 2017518804 A JP2017518804 A JP 2017518804A JP 6820254 B2 JP6820254 B2 JP 6820254B2
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membered
alkyl
group
cancer
mmol
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Japanese (ja)
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JP2017530176A (ja
JP2017530176A5 (enExample
Inventor
エフ． アントニー ロメロ，
エフ． アントニー ロメロ，
スティーブン アール． マグヌソン，
スティーブン アール． マグヌソン，
リチャード パスター，
リチャード パスター，
ビッキー シャオ−ウェイ ツイ，
ビッキー シャオ−ウェイ ツイ，
ジェレミー マレー，
ジェレミー マレー，
テリー クローフォード，
テリー クローフォード，
ダニエル ジェイ． バーディック，
ダニエル ジェイ． バーディック，
ブライアン ケー． アルブレヒト，
ブライアン ケー． アルブレヒト，
アレクサンドル コート，
アレクサンドル コート，
アレクサンダー エム． テイラー，
アレクサンダー エム． テイラー，
クリストファー ジー． ナスヴェスチャック，
クリストファー ジー． ナスヴェスチャック，
イブ レブラン，
イブ レブラン，
マイケル チャールズ ヒューイット，
マイケル チャールズ ヒューイット，
ヲン ワー ライ，
ヲン ワー ライ，
ケビン チェン，
ケビン チェン，
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Constellation Pharmaceuticals Inc
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Constellation Pharmaceuticals Inc
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JP2017518804A 2014-10-10 2015-10-10 治療用化合物およびその使用 Expired - Fee Related JP6820254B2 (ja)

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CN2014088315 2014-10-10
CNPCT/CN2014/088315 2014-10-10
PCT/CN2015/091614 WO2016055028A1 (en) 2014-10-10 2015-10-10 Therapeutic compounds and uses thereof

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JP2017530176A JP2017530176A (ja) 2017-10-12
JP2017530176A5 JP2017530176A5 (enExample) 2018-11-22
JP6820254B2 true JP6820254B2 (ja) 2021-01-27

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JP6639497B2 (ja) * 2014-11-10 2020-02-05 ジェネンテック， インコーポレイテッド ブロモドメインインヒビターおよびその使用
AU2017213628B2 (en) 2016-02-05 2021-07-29 Denali Therapeutics Inc. Inhibitors of receptor-interacting protein kinase 1
WO2017205536A2 (en) * 2016-05-24 2017-11-30 Genentech, Inc. Therapeutic compounds and uses thereof
CN109715790A (zh) 2016-07-25 2019-05-03 埃皮兹姆公司 Crebbp相关的癌症疗法
WO2018107060A1 (en) 2016-12-09 2018-06-14 Denali Therapeutics Inc. Compounds, compositions and methods
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CN107643405B (zh) * 2017-09-19 2020-07-17 上海市肺科医院 一种基于自身抗体检测的肺癌诊断试剂盒及其应用
WO2019070742A1 (en) * 2017-10-03 2019-04-11 Sidecar Therapeutics, Inc. APOPTOSIS SIGNAL REGULATION KINASE 1 (ASK 1) INHIBITORS COMPOUNDS
CA3095367A1 (en) 2018-03-29 2019-10-03 Board Of Regents, The University Of Texas System Imidazopiperazine inhibitors of transcription activating proteins
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