CN107108512B - 治疗性化合物及其用途 - Google Patents

治疗性化合物及其用途 Download PDF

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CN107108512B
CN107108512B CN201580066923.XA CN201580066923A CN107108512B CN 107108512 B CN107108512 B CN 107108512B CN 201580066923 A CN201580066923 A CN 201580066923A CN 107108512 B CN107108512 B CN 107108512B
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compound
membered
methyl
cancer
alkyl
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CN107108512A (zh
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F·A·罗梅罗
S·R·马格努森
R·帕斯托
V·H-W·崔
J·默里
T·克劳福德
D·J·伯迪克
B·K·阿尔布雷克特
A·科特
A·M·泰勒
C·G·纳斯维斯查克
Y·勒布朗
M·C·休伊特
K·W·莱
K·陈
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Genentech Inc
Constellation Pharmaceuticals Inc
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Genentech Inc
Constellation Pharmaceuticals Inc
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CN201580066923.XA 2014-10-10 2015-10-10 治疗性化合物及其用途 Active CN107108512B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN2014088315 2014-10-10
CNPCT/CN2014/088315 2014-10-10
PCT/CN2015/091614 WO2016055028A1 (en) 2014-10-10 2015-10-10 Therapeutic compounds and uses thereof

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CN107108512A CN107108512A (zh) 2017-08-29
CN107108512B true CN107108512B (zh) 2021-05-04

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EP (1) EP3204360B1 (enExample)
JP (1) JP6820254B2 (enExample)
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JP7160688B2 (ja) * 2016-05-24 2022-10-25 ジェネンテック， インコーポレイテッド Ｃｂｐ／ｅｐ３００の複素環式インヒビターおよびがんの処置におけるそれらの使用
CN109715790A (zh) 2016-07-25 2019-05-03 埃皮兹姆公司 Crebbp相关的癌症疗法
HUE058802T2 (hu) 2016-12-09 2022-09-28 Denali Therapeutics Inc RIPK1 inhibitorokként alkalmas vegyületek
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CN107643405B (zh) * 2017-09-19 2020-07-17 上海市肺科医院 一种基于自身抗体检测的肺癌诊断试剂盒及其应用
WO2019070742A1 (en) * 2017-10-03 2019-04-11 Sidecar Therapeutics, Inc. APOPTOSIS SIGNAL REGULATION KINASE 1 (ASK 1) INHIBITORS COMPOUNDS
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