JP6589246B2 - イミダゾ［４，５‐ｃ］ピリジン由来のｓｓａｏ阻害剤 - Google Patents
イミダゾ［４，５‐ｃ］ピリジン由来のｓｓａｏ阻害剤 Download PDFInfo
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- JP6589246B2 JP6589246B2 JP2017515186A JP2017515186A JP6589246B2 JP 6589246 B2 JP6589246 B2 JP 6589246B2 JP 2017515186 A JP2017515186 A JP 2017515186A JP 2017515186 A JP2017515186 A JP 2017515186A JP 6589246 B2 JP6589246 B2 JP 6589246B2
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| PCT/GB2015/052691 WO2016042332A1 (en) | 2014-09-17 | 2015-09-17 | Imidazo[4,5-c]pyridine derived ssao inhibitors |
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| WO2018148856A1 (en) * | 2017-02-14 | 2018-08-23 | Eli Lilly And Company | Diazaspirodecanyl-pyrimidine compounds useful as ssao inhibitors |
| AU2021332217A1 (en) | 2020-08-25 | 2023-05-11 | Eli Lilly And Company | Polymorphs of an ssao inhibitor |
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| US6982286B2 (en) | 2001-07-12 | 2006-01-03 | Biotie Therapies Corp. | Carbocyclic hydrazino inhibitors of copper-containing amine oxidases |
| US20050096360A1 (en) | 2003-08-08 | 2005-05-05 | Salter-Cid Luisa M. | Inhibitors of semicarbazide-sensitive amine oxidase (SSAO) and VAP-1 mediated adhesion useful for treatment of diseases |
| AU2004270187A1 (en) | 2003-09-04 | 2005-03-17 | Aventis Pharmaceuticals Inc. | Substituted indoles as inhibitors of poly (ADP-ribose) polymerase (PARP) |
| EP2004166A2 (en) | 2006-03-31 | 2008-12-24 | La Jolla Pharmaceutical Company | Inhibitors of semicarbazide-sensitive amine oxidase (ssao) and vap-1 mediated adhesion useful for treatment and prevention of diseases |
| US7947723B2 (en) | 2008-02-01 | 2011-05-24 | Spelman College | Synthesis and anti-proliferative effect of benzimidazole derivatives |
| JP5613671B2 (ja) * | 2008-09-16 | 2014-10-29 | プロキシマジェン エルティーディーＰｒｏｘｉｍａｇｅｎ Ｌｔｄ． | 新規化合物ｉｉ |
| BRPI0918602B8 (pt) * | 2008-09-16 | 2021-05-25 | Benevolentai Cambridge Ltd | inibidores da atividade de ssao, seu uso, e formulação farmacêutica |
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| GB201416446D0 (en) | 2014-09-17 | 2014-10-29 | Proximagen Ltd | New enzyme inhibitor compounds |
| JP2019502672A (ja) * | 2015-12-07 | 2019-01-31 | ベネボレンタイ ケンブリッジ リミティド | 疼痛の治療のためのｖａｐ−１阻害剤 |
| GB201709136D0 (en) * | 2017-06-08 | 2017-07-26 | Proximagen Ltd | New therapeutic uses of enzyme inhibitors |
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| WO2016042332A1 (en) | 2016-03-24 |
| HUE045827T2 (hu) | 2020-01-28 |
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| GB201416444D0 (en) | 2014-10-29 |
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| PL3194389T3 (pl) | 2019-11-29 |
| US20170275281A1 (en) | 2017-09-28 |
| IL251166A0 (en) | 2017-04-30 |
| CA2961424A1 (en) | 2016-03-24 |
| IL251166B (en) | 2020-06-30 |
| AU2015316611A1 (en) | 2017-04-06 |
| US11530208B2 (en) | 2022-12-20 |
| CN107074853A (zh) | 2017-08-18 |
| ES2744548T3 (es) | 2020-02-25 |
| CN107074853B (zh) | 2019-07-23 |
| AU2015316611B2 (en) | 2019-05-30 |
| EP3194389B1 (en) | 2019-08-07 |
| PT3194389T (pt) | 2019-09-19 |
| EP3194389A1 (en) | 2017-07-26 |
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