JP6533798B2 - ジヒドロイソオキサゾール誘導体の製造方法 - Google Patents

ジヒドロイソオキサゾール誘導体の製造方法 Download PDF

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Publication number
JP6533798B2
JP6533798B2 JP2016569396A JP2016569396A JP6533798B2 JP 6533798 B2 JP6533798 B2 JP 6533798B2 JP 2016569396 A JP2016569396 A JP 2016569396A JP 2016569396 A JP2016569396 A JP 2016569396A JP 6533798 B2 JP6533798 B2 JP 6533798B2
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Japan
Prior art keywords
formula
chlorine
acid
mixture
compound
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JP2016569396A
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English (en)
Japanese (ja)
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JP2017517513A (ja
JP2017517513A5 (OSRAM
Inventor
オムバーガー，ギュンター
フォード，マルク・ジェイムズ
ヒューゲル，アンドレアス
知己 土屋
知己 土屋
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Bayer CropScience AG
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Bayer CropScience AG
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Publication of JP2017517513A5 publication Critical patent/JP2017517513A5/ja
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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
    • C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
    • C07D261/04—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/72—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms
    • A01N43/80—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with nitrogen atoms and oxygen or sulfur atoms as ring hetero atoms five-membered rings with one nitrogen atom and either one oxygen atom or one sulfur atom in positions 1,2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Plant Pathology (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2016569396A 2014-05-28 2015-05-27 ジヒドロイソオキサゾール誘導体の製造方法 Active JP6533798B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP14170155 2014-05-28
EP14170155.7 2014-05-28
PCT/EP2015/061623 WO2015181189A1 (en) 2014-05-28 2015-05-27 Process for preparing dihydroisoxazole derivatives

Publications (3)

Publication Number Publication Date
JP2017517513A JP2017517513A (ja) 2017-06-29
JP2017517513A5 JP2017517513A5 (OSRAM) 2018-07-05
JP6533798B2 true JP6533798B2 (ja) 2019-06-19

Family

ID=50828731

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2016569396A Active JP6533798B2 (ja) 2014-05-28 2015-05-27 ジヒドロイソオキサゾール誘導体の製造方法

Country Status (12)

Country Link
US (1) US9796690B2 (OSRAM)
EP (1) EP3148976B1 (OSRAM)
JP (1) JP6533798B2 (OSRAM)
KR (1) KR102337028B1 (OSRAM)
CN (1) CN106414417B (OSRAM)
BR (1) BR112016027824B1 (OSRAM)
DK (1) DK3148976T3 (OSRAM)
ES (1) ES2730048T3 (OSRAM)
IL (1) IL248568B (OSRAM)
MX (1) MX382631B (OSRAM)
TW (1) TWI665192B (OSRAM)
WO (1) WO2015181189A1 (OSRAM)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN107406374B (zh) * 2015-03-05 2020-07-14 拜耳作物科学股份公司 制备3-氯-2-乙烯基苯基磺酸酯的方法
DK3548463T3 (da) * 2016-12-05 2020-11-30 Bayer Cropscience Ag Fremgangsmåde til fremstilling af 3-substituerede 2-vinylphenylsulfonater
WO2020251006A1 (ja) * 2019-06-14 2020-12-17 クミアイ化学工業株式会社 ジヒドロイソキサゾールの製造方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
OA09122A (en) 1988-07-08 1991-10-31 Schering Agrochemicals Ltd Triazole insecticides.
DE4331448A1 (de) 1993-09-16 1995-03-23 Hoechst Schering Agrevo Gmbh Substituierte Isoxazoline, Verfahren zu deren Herstellung, diese enthaltende Mittel und deren Verwendung als Safener
EP1878730A1 (en) 2006-07-12 2008-01-16 Bayer Schering Pharma Aktiengesellschaft Substituted isoxazolines, pharmaceutical compositions containing the same, methods of preparing the same, and uses of the same
WO2008013622A2 (en) * 2006-07-27 2008-01-31 E. I. Du Pont De Nemours And Company Fungicidal azocyclic amides
KR20100105890A (ko) * 2008-01-25 2010-09-30 이 아이 듀폰 디 네모아 앤드 캄파니 살균제 아미드
CN101970432B (zh) * 2008-01-25 2014-05-28 杜邦公司 杀真菌杂环化合物
US20110223257A1 (en) 2008-11-17 2011-09-15 Enzon Pharmaceuticals, Inc. Releasable fusogenic lipids for nucleic acids delivery systems
PL2521450T3 (pl) * 2010-01-07 2015-07-31 Du Pont Grzybobójcze związki heterocykliczne
EP2921481A1 (de) * 2011-12-27 2015-09-23 Bayer Intellectual Property GmbH 4-piperidine carboxylic acid derivatives
WO2013127808A1 (en) * 2012-03-02 2013-09-06 Syngenta Participations Ag Microbiocidal pyrazole derivatives

Also Published As

Publication number Publication date
DK3148976T3 (da) 2019-05-27
TW201625567A (zh) 2016-07-16
CN106414417B (zh) 2019-04-16
IL248568B (en) 2019-03-31
IL248568A0 (en) 2016-12-29
EP3148976B1 (en) 2019-03-13
US9796690B2 (en) 2017-10-24
CN106414417A (zh) 2017-02-15
EP3148976A1 (en) 2017-04-05
JP2017517513A (ja) 2017-06-29
MX2016015623A (es) 2017-02-27
BR112016027824B1 (pt) 2021-03-23
TWI665192B (zh) 2019-07-11
ES2730048T3 (es) 2019-11-07
KR20170012331A (ko) 2017-02-02
WO2015181189A1 (en) 2015-12-03
KR102337028B1 (ko) 2021-12-07
MX382631B (es) 2025-03-13
US20170247345A1 (en) 2017-08-31

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