JP6425734B2 - Ｎ−ベンジル−２−（２−ニトロ−１ｈ−イミダゾール−１−イル）アセトアミドを得るための製造工程 - Google Patents

Ｎ−ベンジル−２−（２−ニトロ−１ｈ−イミダゾール−１−イル）アセトアミドを得るための製造工程 Download PDF

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JP6425734B2
JP6425734B2 JP2016554169A JP2016554169A JP6425734B2 JP 6425734 B2 JP6425734 B2 JP 6425734B2 JP 2016554169 A JP2016554169 A JP 2016554169A JP 2016554169 A JP2016554169 A JP 2016554169A JP 6425734 B2 JP6425734 B2 JP 6425734B2
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benzyl
nitro
acetamide
imidazol
obtaining
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Japanese (ja)
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JP2016539185A (ja
JP2016539185A5 (enExample
Inventor
ベガ，エルリンダ ハンダル
ベガ，エルリンダ ハンダル
リバス，カルメン エレナ アリアス
リバス，カルメン エレナ アリアス
デ メルロス，アナ カリナ クチジャ
デ メルロス，アナ カリナ クチジャ
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ミニステリオ・デ・エデュカシオン
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/91—Nitro radicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis

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  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)
JP2016554169A 2013-11-19 2014-11-19 Ｎ−ベンジル−２−（２−ニトロ−１ｈ−イミダゾール−１−イル）アセトアミドを得るための製造工程 Active JP6425734B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
SV2013004584A SV2013004584A (es) 2013-11-19 2013-11-19 Procedimiento de manufactura para obtención de de n-bencil-2-(2-nitro-1h-imidazol-1-il)acetamida
SV2013004584 2013-11-19
PCT/SV2014/000001 WO2015076760A1 (es) 2013-11-19 2014-11-19 Procedimiento de manufactura para obtención de n-bencil-2-(2-nitro-1h-imidazol-1-il)acetamida

Publications (3)

Publication Number Publication Date
JP2016539185A JP2016539185A (ja) 2016-12-15
JP2016539185A5 JP2016539185A5 (enExample) 2018-04-26
JP6425734B2 true JP6425734B2 (ja) 2018-11-21

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JP2016554169A Active JP6425734B2 (ja) 2013-11-19 2014-11-19 Ｎ−ベンジル−２−（２−ニトロ−１ｈ−イミダゾール−１−イル）アセトアミドを得るための製造工程

Country Status (5)

Country Link
US (1) US9765036B2 (enExample)
JP (1) JP6425734B2 (enExample)
BR (1) BR112016011160B1 (enExample)
SV (1) SV2013004584A (enExample)
WO (1) WO2015076760A1 (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2017205622A1 (en) * 2016-05-25 2017-11-30 Savant Neglected Diseases, Llc Method of making benznidazole
WO2019240671A1 (es) * 2018-06-11 2019-12-19 Ministerio De Educación, Ciencia Y Tecnología Método de manufactura para la producción de benznidazol y su escalado industrial

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3505349A (en) * 1966-04-18 1970-04-07 Hoffmann La Roche 2-nitro-imidazolyl-1-acetamides
WO2001087848A2 (en) * 2000-05-17 2001-11-22 Manufacturas Humberto Bukele E Hijos, S.A. De C.V. Synthesis procedure for biphenylimidazolyl-(1)-phenylmethane and related compounds

Also Published As

Publication number Publication date
JP2016539185A (ja) 2016-12-15
US20160289197A1 (en) 2016-10-06
WO2015076760A1 (es) 2015-05-28
SV2013004584A (es) 2015-09-07
BR112016011160A2 (enExample) 2017-08-08
BR112016011160B1 (pt) 2022-07-05
US9765036B2 (en) 2017-09-19

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