JP6118392B2 - 非麻薬性鎮痛作用を有する合成ペプチド - Google Patents

非麻薬性鎮痛作用を有する合成ペプチド Download PDF

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Publication number
JP6118392B2
JP6118392B2 JP2015501616A JP2015501616A JP6118392B2 JP 6118392 B2 JP6118392 B2 JP 6118392B2 JP 2015501616 A JP2015501616 A JP 2015501616A JP 2015501616 A JP2015501616 A JP 2015501616A JP 6118392 B2 JP6118392 B2 JP 6118392B2
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peptide
amino acids
amino acid
ala
substitution
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JP2015501616A
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Japanese (ja)
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JP2015512385A (ja
Inventor
ペトロヴィチ ヴラーソフ,ゲンナジー
ペトロヴィチ ヴラーソフ,ゲンナジー
ミハイロヴィチ コチン,アルカディー
ミハイロヴィチ コチン,アルカディー
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コチン,オレク アルカーディエヴィチ
コチン,オレク アルカーディエヴィチ
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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/06Linear peptides containing only normal peptide links having 5 to 11 amino acids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00Anaesthetics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A61P29/02Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID] without antiinflammatory effect
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Rheumatology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Anesthesiology (AREA)
  • Engineering & Computer Science (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
JP2015501616A 2012-03-22 2012-12-07 非麻薬性鎮痛作用を有する合成ペプチド Active JP6118392B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
RU2012110908/10A RU2508295C2 (ru) 2012-03-22 2012-03-22 Синтетические пептиды с ненаркотическим типом анальгетического действия
RU2012110908 2012-03-22
PCT/RU2012/001036 WO2013141750A1 (ru) 2012-03-22 2012-12-07 Синтетические пептиды с ненаркотическим типом анальгетического действия

Publications (2)

Publication Number Publication Date
JP2015512385A JP2015512385A (ja) 2015-04-27
JP6118392B2 true JP6118392B2 (ja) 2017-04-19

Family

ID=49223070

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2015501616A Active JP6118392B2 (ja) 2012-03-22 2012-12-07 非麻薬性鎮痛作用を有する合成ペプチド

Country Status (8)

Country Link
US (1) US9260482B2 (OSRAM)
EP (1) EP2848629B1 (OSRAM)
JP (1) JP6118392B2 (OSRAM)
CA (1) CA2867994C (OSRAM)
ES (1) ES2651265T3 (OSRAM)
IN (1) IN2014MN02080A (OSRAM)
RU (1) RU2508295C2 (OSRAM)
WO (1) WO2013141750A1 (OSRAM)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2932529C (en) * 2013-12-19 2022-03-22 Eisai R&D Management Co., Ltd. Therapeutic and/or preventive agent comprising 1-indansulfamide derivative for pain
DE102016125645A1 (de) 2016-12-23 2018-06-28 Forschungszentrum Jülich GmbH D-enantiomere Peptide zur Therapie von chronischem und neuropathischem Schmerz
RU2651491C1 (ru) 2017-04-07 2018-04-19 Общество с ограниченной ответственностью "Биофармокс" Специфические пептидные ингибиторы клатрина
US20210228677A1 (en) * 2020-01-28 2021-07-29 Pharmbiotech OY Pharmaceutical composition and a method for its manufacture

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1229658B (it) 1989-04-21 1991-09-06 Eniricerche Spa Analoghi della timopentina retro-inversi ad uno o piu' legami, il metodo per la loro sintesi ed il loro impiego per la preparazione di composizioni farmaceutiche.
US5175146A (en) * 1989-12-05 1992-12-29 Vical, Inc. Synthetic calcitonin peptides

Also Published As

Publication number Publication date
CA2867994C (en) 2017-05-16
IN2014MN02080A (OSRAM) 2015-08-21
US9260482B2 (en) 2016-02-16
RU2012110908A (ru) 2013-09-27
US20150073123A1 (en) 2015-03-12
WO2013141750A1 (ru) 2013-09-26
EP2848629A1 (en) 2015-03-18
ES2651265T3 (es) 2018-01-25
EP2848629B1 (en) 2017-09-06
CA2867994A1 (en) 2013-09-26
RU2508295C2 (ru) 2014-02-27
JP2015512385A (ja) 2015-04-27
EP2848629A4 (en) 2016-03-02

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