JP6095075B2 - キナーゼ阻害剤としてのプリノン化合物 - Google Patents
キナーゼ阻害剤としてのプリノン化合物 Download PDFInfo
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- JP6095075B2 JP6095075B2 JP2014555678A JP2014555678A JP6095075B2 JP 6095075 B2 JP6095075 B2 JP 6095075B2 JP 2014555678 A JP2014555678 A JP 2014555678A JP 2014555678 A JP2014555678 A JP 2014555678A JP 6095075 B2 JP6095075 B2 JP 6095075B2
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- substituted
- unsubstituted
- alkyl
- cycloalkyl
- compound
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Classifications
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Landscapes
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| US201261637765P | 2012-04-24 | 2012-04-24 | |
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| US13/460,524 US8501724B1 (en) | 2012-01-31 | 2012-04-30 | Purinone compounds as kinase inhibitors |
| PCT/US2013/023918 WO2013116382A1 (en) | 2012-01-31 | 2013-01-30 | Purinone compounds as kinase inhibitors |
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| JP2018228582A Pending JP2019059758A (ja) | 2012-01-31 | 2018-12-05 | キナーゼ阻害剤としてのプリノン化合物 |
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| JP (3) | JP6095075B2 (enExample) |
| KR (2) | KR20180030730A (enExample) |
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| CA (2) | CA2863140C (enExample) |
| HK (1) | HK1203489A1 (enExample) |
| IL (1) | IL261282A (enExample) |
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| PH (1) | PH12014501815A1 (enExample) |
| RU (2) | RU2018118216A (enExample) |
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Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2017114880A (ja) * | 2012-01-31 | 2017-06-29 | ファーマサイクリックス エルエルシー | キナーゼ阻害剤としてのプリノン化合物 |
| JP2019069977A (ja) * | 2013-07-02 | 2019-05-09 | ファーマサイクリックス エルエルシー | キナーゼ阻害剤としてのプリノン化合物 |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| EP2529621B1 (en) | 2006-09-22 | 2016-10-05 | Pharmacyclics LLC | Inhibitors of bruton's tyrosine kinase |
| US8809273B2 (en) | 2007-03-28 | 2014-08-19 | Pharmacyclics, Inc. | Inhibitors of Bruton's tyrosine kinase |
| CN102159214A (zh) | 2008-07-16 | 2011-08-17 | 药品循环公司 | 用于实体肿瘤的治疗的布鲁顿酪氨酸激酶的抑制剂 |
| MX380504B (es) | 2010-06-03 | 2025-03-12 | Pharmacyclics Llc | El uso de inhibidores de la tirosina quinasa de bruton (btk). |
| AU2012255860C1 (en) | 2011-05-17 | 2015-12-10 | Principia Biopharma Inc. | Tyrosine kinase inhibitors |
| WO2012158795A1 (en) | 2011-05-17 | 2012-11-22 | Principia Biopharma Inc. | Pyrazolopyrimidine derivatives as tyrosine kinase inhibitors |
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Cited By (3)
| Publication number | Priority date | Publication date | Assignee | Title |
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| JP2017114880A (ja) * | 2012-01-31 | 2017-06-29 | ファーマサイクリックス エルエルシー | キナーゼ阻害剤としてのプリノン化合物 |
| JP2019059758A (ja) * | 2012-01-31 | 2019-04-18 | ファーマサイクリックス エルエルシー | キナーゼ阻害剤としてのプリノン化合物 |
| JP2019069977A (ja) * | 2013-07-02 | 2019-05-09 | ファーマサイクリックス エルエルシー | キナーゼ阻害剤としてのプリノン化合物 |
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