JP6063482B2 - トリアゾロ［４，５−ｄ］ピリミジン誘導体 - Google Patents
トリアゾロ［４，５−ｄ］ピリミジン誘導体 Download PDFInfo
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- JP6063482B2 JP6063482B2 JP2014553622A JP2014553622A JP6063482B2 JP 6063482 B2 JP6063482 B2 JP 6063482B2 JP 2014553622 A JP2014553622 A JP 2014553622A JP 2014553622 A JP2014553622 A JP 2014553622A JP 6063482 B2 JP6063482 B2 JP 6063482B2
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- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
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| EP12000558 | 2012-01-28 | ||
| PCT/EP2012/005358 WO2013110309A1 (en) | 2012-01-28 | 2012-12-21 | Triazolo[4,5-d]pyrimidine derivatives |
Publications (3)
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| JP2015505541A JP2015505541A (ja) | 2015-02-23 |
| JP2015505541A5 JP2015505541A5 (enExample) | 2016-12-15 |
| JP6063482B2 true JP6063482B2 (ja) | 2017-01-18 |
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| EP (1) | EP2807161B1 (enExample) |
| JP (1) | JP6063482B2 (enExample) |
| KR (1) | KR20140117636A (enExample) |
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| AR (1) | AR089810A1 (enExample) |
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Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
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| EP2994471B1 (en) * | 2013-05-06 | 2017-05-17 | Merck Patent GmbH | Macrocycles as kinase inhibitors |
| US20160222014A1 (en) * | 2013-09-10 | 2016-08-04 | Asana Biosciences, Llc | Compounds for regulating fak and/or src pathways |
| CN106220644B (zh) * | 2015-04-24 | 2020-07-31 | 广州再极医药科技有限公司 | 稠环嘧啶氨基衍生物﹑其制备方法、中间体、药物组合物及应用 |
| PL3498693T3 (pl) * | 2016-08-10 | 2025-03-24 | Takeda Pharmaceutical Company Limited | Związek heterocykliczny |
| WO2018119440A1 (en) | 2016-12-22 | 2018-06-28 | Calithera Biosciences, Inc. | Compositions and methods for inhibiting arginase activity |
| KR102328423B1 (ko) * | 2018-09-11 | 2021-11-18 | 재단법인 대구경북첨단의료산업진흥재단 | 신규 트리아졸로-피리미딘 유도체, 이의 제조방법 및 이를 유효성분으로 함유하는 단백질 키나아제 관련 질환의 예방 또는 치료용 약학적 조성물 |
| US20220040183A1 (en) * | 2018-10-01 | 2022-02-10 | INSERM (Institut National de la Santé et de la Recherche Médicale) | Use of inhibitors of stress granule formation for targeting the regulation of immune responses |
| WO2021222147A1 (en) * | 2020-04-27 | 2021-11-04 | Hibercell, Inc. | Heterocyclic gcn2 modulators |
| GB202008749D0 (en) | 2020-06-09 | 2020-07-22 | Ip2Ipo Innovations Ltd | Novel compounds |
| KR20250122240A (ko) | 2024-02-06 | 2025-08-13 | 한미약품 주식회사 | 신규한 함질소 헤테로고리 유도체 및 이의 용도 |
| WO2025179188A1 (en) * | 2024-02-22 | 2025-08-28 | Juno Therapeutics, Inc. | Pyrazole-based inhibitors of dna-dependent protein kinase and compositions and applications in gene editing |
| CN120504636B (zh) * | 2025-07-22 | 2025-10-31 | 江西中医药大学 | 一种磺胺噻唑-甲氧苄啶药物晶盐及其制备方法和应用 |
Family Cites Families (17)
| Publication number | Priority date | Publication date | Assignee | Title |
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| GB9624482D0 (en) | 1995-12-18 | 1997-01-15 | Zeneca Phaema S A | Chemical compounds |
| CA2242425C (en) | 1996-02-13 | 2006-07-18 | Zeneca Limited | Quinazoline derivatives as vegf inhibitors |
| NZ331191A (en) | 1996-03-05 | 2000-03-27 | Zeneca Ltd | 4-anilinoquinazoline derivatives and pharmaceutical compositions thereof |
| GB9718972D0 (en) | 1996-09-25 | 1997-11-12 | Zeneca Ltd | Chemical compounds |
| GB9714249D0 (en) | 1997-07-08 | 1997-09-10 | Angiogene Pharm Ltd | Vascular damaging agents |
| GB9900334D0 (en) | 1999-01-07 | 1999-02-24 | Angiogene Pharm Ltd | Tricylic vascular damaging agents |
| GB9900752D0 (en) | 1999-01-15 | 1999-03-03 | Angiogene Pharm Ltd | Benzimidazole vascular damaging agents |
| BR0111230A (pt) | 2000-05-31 | 2003-06-10 | Astrazeneca Ab | Composto, e, uso e processo para a preparação do mesmo |
| KR20030014425A (ko) | 2000-07-07 | 2003-02-17 | 앤지오젠 파마슈티칼스 리미티드 | 혈관 손상제인 콜치놀 유도체 |
| EE200300015A (et) | 2000-07-07 | 2004-10-15 | Angiogene Pharmaceuticals Limited | Kolhinooli derivaadid kui angiogeneesi inhibiitorid |
| NZ545058A (en) | 2003-07-16 | 2008-05-30 | Janssen Pharmaceutica Nv | Triazolopyrimidine derivatives as glycogen synthase kinase 3 inhibitors |
| JP5704785B2 (ja) | 2004-07-19 | 2015-04-22 | ザ・ジョンズ・ホプキンス・ユニバーシティ | 免疫抑制のためのｆｌｔ３阻害剤 |
| DE102004051827A1 (de) | 2004-10-25 | 2006-05-04 | Hörmann KG Antriebstechnik | Armbandsender |
| BRPI0517272A (pt) * | 2004-10-29 | 2008-10-07 | Tibotec Pharm Ltd | derivados de pirimidina bicìclicos de inibição de hiv |
| WO2006075023A2 (en) | 2005-01-14 | 2006-07-20 | Janssen Pharmaceutica N.V. | Triazolopyrimidine derivatives as glycogen synthase kinase 3 inhibitors |
| WO2006091737A1 (en) | 2005-02-24 | 2006-08-31 | Kemia, Inc. | Modulators of gsk-3 activity |
| EA022120B1 (ru) * | 2009-10-20 | 2015-11-30 | Целльзом Лимитид | Аналоги гетероциклил пиразолопиримидина в качестве ингибиторов jak |
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- 2012-12-21 SG SG11201404234YA patent/SG11201404234YA/en unknown
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- 2012-12-21 MX MX2014008864A patent/MX2014008864A/es unknown
- 2012-12-21 BR BR112014016884A patent/BR112014016884A2/pt not_active IP Right Cessation
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- 2014-08-27 ZA ZA2014/06323A patent/ZA201406323B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| KR20140117636A (ko) | 2014-10-07 |
| MX2014008864A (es) | 2014-12-15 |
| IL233808B (en) | 2018-03-29 |
| US9409914B2 (en) | 2016-08-09 |
| AU2012367141B2 (en) | 2016-12-22 |
| JP2015505541A (ja) | 2015-02-23 |
| ZA201406323B (en) | 2016-08-31 |
| CA2862694A1 (en) | 2013-08-01 |
| AR089810A1 (es) | 2014-09-17 |
| EP2807161A1 (en) | 2014-12-03 |
| BR112014016884A2 (pt) | 2017-06-27 |
| ES2655264T3 (es) | 2018-02-19 |
| CN104066734B (zh) | 2017-03-29 |
| EP2807161B1 (en) | 2017-10-04 |
| WO2013110309A1 (en) | 2013-08-01 |
| CN104066734A (zh) | 2014-09-24 |
| AU2012367141A1 (en) | 2014-09-11 |
| US20140378431A1 (en) | 2014-12-25 |
| CA2862694C (en) | 2020-07-28 |
| SG11201404234YA (en) | 2014-08-28 |
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