JP6025871B2 - ペプチドホルモンのカルシトニンｃｇｒｐファミリーのペプチドアンタゴニスト及びその使用 - Google Patents

ペプチドホルモンのカルシトニンｃｇｒｐファミリーのペプチドアンタゴニスト及びその使用 Download PDF

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JP6025871B2
JP6025871B2 JP2014554880A JP2014554880A JP6025871B2 JP 6025871 B2 JP6025871 B2 JP 6025871B2 JP 2014554880 A JP2014554880 A JP 2014554880A JP 2014554880 A JP2014554880 A JP 2014554880A JP 6025871 B2 JP6025871 B2 JP 6025871B2
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JP2015513318A5 (cg-RX-API-DMAC7.html
JP2015513318A (ja
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クリストファー ジェイ． ソアレス
クリストファー ジェイ． ソアレス
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22—Hormones
    • A61K38/225—Calcitonin gene related peptide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22—Hormones
    • A61K38/23—Calcitonins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/18—Drugs for disorders of the endocrine system of the parathyroid hormones
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/18—Drugs for disorders of the endocrine system of the parathyroid hormones
    • A61P5/22—Drugs for disorders of the endocrine system of the parathyroid hormones for decreasing, blocking or antagonising the activity of calcitonin
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/57527—Calcitonin gene related peptide
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/585—Calcitonins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

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  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Endocrinology (AREA)
  • Genetics & Genomics (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Zoology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Molecular Biology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biophysics (AREA)
  • Toxicology (AREA)
  • Biochemistry (AREA)
  • Immunology (AREA)
  • Epidemiology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Diabetes (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Pain & Pain Management (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
JP2014554880A 2012-01-26 2013-01-25 ペプチドホルモンのカルシトニンｃｇｒｐファミリーのペプチドアンタゴニスト及びその使用 Active JP6025871B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261591236P 2012-01-26 2012-01-26
US61/591,236 2012-01-26
PCT/US2013/023260 WO2013112912A1 (en) 2012-01-26 2013-01-25 Peptide antagonists of the calcitonin cgrp family of peptide hormones and their use

Related Child Applications (1)

Application Number Title Priority Date Filing Date
JP2016199234A Division JP6411425B2 (ja) 2012-01-26 2016-10-07 ペプチドホルモンのカルシトニンｃｇｒｐファミリーのペプチドアンタゴニスト及びその使用

Publications (3)

Publication Number Publication Date
JP2015513318A JP2015513318A (ja) 2015-05-07
JP2015513318A5 JP2015513318A5 (cg-RX-API-DMAC7.html) 2016-03-10
JP6025871B2 true JP6025871B2 (ja) 2016-11-16

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Family Applications (3)

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JP2014554880A Active JP6025871B2 (ja) 2012-01-26 2013-01-25 ペプチドホルモンのカルシトニンｃｇｒｐファミリーのペプチドアンタゴニスト及びその使用
JP2016199234A Active JP6411425B2 (ja) 2012-01-26 2016-10-07 ペプチドホルモンのカルシトニンｃｇｒｐファミリーのペプチドアンタゴニスト及びその使用
JP2018177504A Pending JP2019006821A (ja) 2012-01-26 2018-09-21 ペプチドホルモンのカルシトニンｃｇｒｐファミリーのペプチドアンタゴニスト及びその使用

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JP2016199234A Active JP6411425B2 (ja) 2012-01-26 2016-10-07 ペプチドホルモンのカルシトニンｃｇｒｐファミリーのペプチドアンタゴニスト及びその使用
JP2018177504A Pending JP2019006821A (ja) 2012-01-26 2018-09-21 ペプチドホルモンのカルシトニンｃｇｒｐファミリーのペプチドアンタゴニスト及びその使用

Country Status (14)

Country Link
US (3) US9193776B2 (cg-RX-API-DMAC7.html)
EP (2) EP3272769B1 (cg-RX-API-DMAC7.html)
JP (3) JP6025871B2 (cg-RX-API-DMAC7.html)
KR (2) KR102052983B1 (cg-RX-API-DMAC7.html)
CN (2) CN108997490A (cg-RX-API-DMAC7.html)
AU (2) AU2013211929B2 (cg-RX-API-DMAC7.html)
CA (1) CA2861392C (cg-RX-API-DMAC7.html)
DK (1) DK2807187T3 (cg-RX-API-DMAC7.html)
ES (2) ES2819825T3 (cg-RX-API-DMAC7.html)
IL (2) IL233655A (cg-RX-API-DMAC7.html)
MX (1) MX347229B (cg-RX-API-DMAC7.html)
NO (1) NO2864579T3 (cg-RX-API-DMAC7.html)
RU (2) RU2624016C2 (cg-RX-API-DMAC7.html)
WO (1) WO2013112912A1 (cg-RX-API-DMAC7.html)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2017036308A (ja) * 2012-01-26 2017-02-16 クリストファー ジェイ． ソアレス ペプチドホルモンのカルシトニンｃｇｒｐファミリーのペプチドアンタゴニスト及びその使用

Families Citing this family (10)

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WO2015017455A1 (en) * 2013-07-30 2015-02-05 Soares Christopher J Cgrp agonist peptides
JO3669B1 (ar) 2015-01-06 2020-08-27 Ferring Bv بيبتيدات مضَادَّة لببتيد المرتبط بجين الكالسيتونين
CN109311959A (zh) * 2016-01-04 2019-02-05 艾得佩索拉公司 肽类似物
US11390654B2 (en) * 2016-09-02 2022-07-19 Christopher Joseph Soares Use of CGRP receptor antagonists in neuroprotection and neurological disorders
CA2967616A1 (en) * 2016-09-19 2018-03-19 The Governors Of The University Of Alberta Brain penetrant amylin receptor based peptides for alzheimer's disease
EP3707157A4 (en) * 2017-11-06 2021-08-18 Auckland Uniservices Limited PEPTIDIC CONJUGATES AS ANAGONISTS OF THE CGRP RECEIVER, THEIR PREPARATION METHODS AND THEIR USES
JP7214102B2 (ja) * 2019-01-18 2023-01-30 株式会社大一商会 遊技機
JP7214104B2 (ja) * 2019-01-18 2023-01-30 株式会社大一商会 遊技機
JP7214100B2 (ja) * 2019-01-18 2023-01-30 株式会社大一商会 遊技機
CN116456981A (zh) * 2020-11-19 2023-07-18 辉瑞爱尔兰制药公司 用于改善的grp抑制剂递送的组合物

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Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2017036308A (ja) * 2012-01-26 2017-02-16 クリストファー ジェイ． ソアレス ペプチドホルモンのカルシトニンｃｇｒｐファミリーのペプチドアンタゴニスト及びその使用

Also Published As

Publication number Publication date
RU2742826C2 (ru) 2021-02-11
AU2013211929B2 (en) 2016-05-26
MX347229B (es) 2017-04-19
JP2019006821A (ja) 2019-01-17
KR20170071613A (ko) 2017-06-23
RU2624016C2 (ru) 2017-06-30
ES2641325T3 (es) 2017-11-08
DK2807187T3 (en) 2017-09-11
AU2016205801A1 (en) 2016-08-04
US9193776B2 (en) 2015-11-24
KR101855242B1 (ko) 2018-05-09
CN108997490A (zh) 2018-12-14
EP2807187A1 (en) 2014-12-03
KR102052983B1 (ko) 2019-12-06
EP3272769A1 (en) 2018-01-24
JP2017036308A (ja) 2017-02-16
IL233655A0 (en) 2014-08-31
WO2013112912A1 (en) 2013-08-01
MX2014008960A (es) 2015-01-16
CN104271596A (zh) 2015-01-07
HK1201068A1 (en) 2015-08-21
IL252555B (en) 2020-06-30
RU2014131605A (ru) 2016-03-20
IL233655A (en) 2017-06-29
RU2017119773A3 (cg-RX-API-DMAC7.html) 2020-11-18
ES2819825T3 (es) 2021-04-19
BR112014018284A2 (pt) 2017-07-04
RU2017119773A (ru) 2018-12-06
US20170204155A1 (en) 2017-07-20
CN104271596B (zh) 2018-09-18
IL252555A0 (en) 2017-07-31
EP3272769B1 (en) 2020-06-17
US20140329752A1 (en) 2014-11-06
HK1249915A1 (en) 2018-11-16
JP6411425B2 (ja) 2018-10-24
AU2013211929A1 (en) 2014-09-11
US10370425B2 (en) 2019-08-06
KR20140132342A (ko) 2014-11-17
US20160145315A1 (en) 2016-05-26
CA2861392A1 (en) 2013-08-01
NO2864579T3 (cg-RX-API-DMAC7.html) 2018-01-20
JP2015513318A (ja) 2015-05-07
EP2807187B1 (en) 2017-07-26
CA2861392C (en) 2021-08-17

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