JP5837890B2 - 神経膠芽腫および星状細胞腫の治療におけるフェノテロールおよびフェノテロール類似体の使用 - Google Patents

神経膠芽腫および星状細胞腫の治療におけるフェノテロールおよびフェノテロール類似体の使用 Download PDF

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JP5837890B2
JP5837890B2 JP2012557260A JP2012557260A JP5837890B2 JP 5837890 B2 JP5837890 B2 JP 5837890B2 JP 2012557260 A JP2012557260 A JP 2012557260A JP 2012557260 A JP2012557260 A JP 2012557260A JP 5837890 B2 JP5837890 B2 JP 5837890B2
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fenoterol
tumor
naphthylfenoterol
pharmaceutical composition
methoxy
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JP2013522230A5 (enExample
JP2013522230A (ja
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アービング ダブリュ． ワイネル
アービング ダブリュ． ワイネル
ミシェル ベルニエ
ミシェル ベルニエ
ローレンス ロバート トール
ローレンス ロバート トール
リュシータ アレナス ヒメネス
リュシータ アレナス ヒメネス
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SRI International Inc
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Emergency Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
JP2012557260A 2010-03-10 2011-03-10 神経膠芽腫および星状細胞腫の治療におけるフェノテロールおよびフェノテロール類似体の使用 Active JP5837890B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US31264210P 2010-03-10 2010-03-10
US61/312,642 2010-03-10
PCT/US2011/027988 WO2011112867A1 (en) 2010-03-10 2011-03-10 The use of fenoterol and fenoterol analogues in the treatment of glioblastomas and astrocytomas

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JP2013522230A JP2013522230A (ja) 2013-06-13
JP2013522230A5 JP2013522230A5 (enExample) 2014-04-17
JP5837890B2 true JP5837890B2 (ja) 2015-12-24

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US (4) US9492405B2 (enExample)
EP (1) EP2544676B1 (enExample)
JP (1) JP5837890B2 (enExample)
AU (2) AU2011224241B2 (enExample)
BR (1) BR112012022552A8 (enExample)
CA (1) CA2791702C (enExample)
WO (1) WO2011112867A1 (enExample)

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EP3125877A4 (en) * 2014-04-03 2017-11-22 Mitchell Woods Pharmaceuticals, Inc. Methods of treating melanoma
KR101585619B1 (ko) * 2014-11-20 2016-01-15 주식회사 아모텍 감전보호소자 및 이를 구비한 휴대용 전자장치
WO2016144371A1 (en) * 2015-03-06 2016-09-15 Mitchell Woods Pharmaceuticals, Inc. Methods of treating cancer
US20180271808A1 (en) * 2015-10-01 2018-09-27 Mitchell Woods Pharmaceuticals, Inc. Methods of reducing chemoresistance and treating cancer
US20190337889A1 (en) * 2015-10-18 2019-11-07 Onco Therapies Llc Compositions and methods of regulating cancer related disorders and diseases
EP3490581A4 (en) * 2016-07-26 2020-10-14 Flagship Pioneering Innovations V, Inc. NEUROMODULATORY COMPOSITIONS AND ASSOCIATED CANCER TREATMENT METHODS
GB201714734D0 (en) 2017-09-13 2017-10-25 Atrogi Ab New compounds and uses
GB201714745D0 (en) 2017-09-13 2017-10-25 Atrogi Ab New compounds and uses
GB201714740D0 (en) 2017-09-13 2017-10-25 Atrogi Ab New compounds and uses
GB201714736D0 (en) 2017-09-13 2017-10-25 Atrogi Ab New compounds and uses
CN109942462B (zh) * 2019-03-06 2022-01-14 宏冠生物药业有限公司 一种盐酸班布特罗的合成工艺
GB201903832D0 (en) 2019-03-20 2019-05-01 Atrogi Ab New compounds and methods
CN114456078B (zh) * 2022-01-19 2022-09-16 汉瑞药业(荆门)有限公司 一种(r)-n-苄基-1-(4-甲氧基苯基)丙-2-胺的制备方法

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CH564509A5 (enExample) 1969-12-12 1975-07-31 Boehringer Sohn Ingelheim
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Publication number Publication date
WO2011112867A1 (en) 2011-09-15
WO2011112867A8 (en) 2012-09-27
AU2014210656A1 (en) 2014-08-28
AU2014210656B2 (en) 2016-03-17
US20130005799A1 (en) 2013-01-03
US10130594B2 (en) 2018-11-20
AU2011224241B2 (en) 2014-05-08
BR112012022552A8 (pt) 2017-12-05
US10925840B2 (en) 2021-02-23
AU2011224241A1 (en) 2012-09-20
US10617654B2 (en) 2020-04-14
US9492405B2 (en) 2016-11-15
US20190008802A1 (en) 2019-01-10
CA2791702C (en) 2018-05-29
BR112012022552A2 (pt) 2016-08-30
JP2013522230A (ja) 2013-06-13
CA2791702A1 (en) 2011-09-15
EP2544676A1 (en) 2013-01-16
US20200197332A1 (en) 2020-06-25
US20170007556A1 (en) 2017-01-12
EP2544676B1 (en) 2018-09-19

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