JP5735510B2 - Ｎ１−置換−５−フルオロ−２−オキソピリミジノン−１（２ｈ）−カルボキサミド誘導体 - Google Patents

Ｎ１−置換−５−フルオロ−２−オキソピリミジノン−１（２ｈ）−カルボキサミド誘導体 Download PDF

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Publication number
JP5735510B2
JP5735510B2 JP2012523955A JP2012523955A JP5735510B2 JP 5735510 B2 JP5735510 B2 JP 5735510B2 JP 2012523955 A JP2012523955 A JP 2012523955A JP 2012523955 A JP2012523955 A JP 2012523955A JP 5735510 B2 JP5735510 B2 JP 5735510B2
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optionally substituted
benzyl
alkyl
phenyl
ring system
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JP2012523955A
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Japanese (ja)
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JP2013501727A (ja
Inventor
ボーベル，ティモティー
ブライアン，クリスティー
ロースバーチ，ベス
マーティン，ティモティー
オーウェン，ダブリュ．
ポバンズ，マーク
トーンバーグ，スコット
ウェブスター，ジェフリー
ヤオ，チェンリン
Original Assignee
ダウ アグロサイエンシィズ エルエルシー
ダウ アグロサイエンシィズ エルエルシー
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Application filed by ダウ アグロサイエンシィズ エルエルシー, ダウ アグロサイエンシィズ エルエルシー filed Critical ダウ アグロサイエンシィズ エルエルシー
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    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A01N47/38—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the group >N—CO—N< where at least one nitrogen atom is part of a heterocyclic ring; Thio analogues thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
JP2012523955A 2009-08-07 2010-08-05 Ｎ１−置換−５−フルオロ−２−オキソピリミジノン−１（２ｈ）−カルボキサミド誘導体 Active JP5735510B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US23224509P 2009-08-07 2009-08-07
US61/232,245 2009-08-07
PCT/US2010/044588 WO2011017545A1 (en) 2009-08-07 2010-08-05 N1-substituted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives

Publications (2)

Publication Number Publication Date
JP2013501727A JP2013501727A (ja) 2013-01-17
JP5735510B2 true JP5735510B2 (ja) 2015-06-17

Family

ID=43535294

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2012523955A Active JP5735510B2 (ja) 2009-08-07 2010-08-05 Ｎ１−置換−５−フルオロ−２−オキソピリミジノン−１（２ｈ）−カルボキサミド誘導体

Country Status (26)

Country Link
US (2) US8552020B2 (OSRAM)
EP (1) EP2461686B1 (OSRAM)
JP (1) JP5735510B2 (OSRAM)
KR (1) KR101792284B1 (OSRAM)
CN (1) CN102497781B (OSRAM)
BR (1) BR112012002757B1 (OSRAM)
CA (1) CA2769656C (OSRAM)
CL (1) CL2012000312A1 (OSRAM)
CO (1) CO6491115A2 (OSRAM)
CR (1) CR20120032A (OSRAM)
DK (1) DK2461686T3 (OSRAM)
EA (1) EA020910B1 (OSRAM)
EC (1) ECSP12011652A (OSRAM)
ES (1) ES2552097T3 (OSRAM)
HU (1) HUE027390T2 (OSRAM)
IL (1) IL217950A (OSRAM)
IN (1) IN2012DN00369A (OSRAM)
MX (1) MX2012001617A (OSRAM)
NI (1) NI201200021A (OSRAM)
NZ (1) NZ597483A (OSRAM)
PE (1) PE20120692A1 (OSRAM)
PL (1) PL2461686T3 (OSRAM)
PT (1) PT2461686E (OSRAM)
UA (1) UA107671C2 (OSRAM)
WO (1) WO2011017545A1 (OSRAM)
ZA (1) ZA201200813B (OSRAM)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PE20120691A1 (es) * 2009-08-07 2012-06-08 Dow Agrosciences Llc Derivados de n1-sulfonil-5-fluoropirimidinona
DK2461688T3 (en) 2009-08-07 2016-06-20 Dow Agrosciences Llc pesticide Compositions
UA107671C2 (en) * 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
CN104994859B (zh) * 2012-12-28 2018-10-26 阿达玛马克西姆股份有限公司 1-(取代的苯甲酰基)-5-氟-4-亚氨基-3-甲基-3,4-二氢嘧啶-2(1h)-酮衍生物
CN104884062B (zh) * 2012-12-28 2018-11-06 阿达玛马克西姆股份有限公司 N-(取代的)-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1(2h)-甲酰胺衍生物
CN104902757B (zh) 2012-12-28 2019-01-08 阿达玛马克西姆股份有限公司 N-(取代的)-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1(2h)-羧酸酯衍生物
JP2016503816A (ja) 2012-12-31 2016-02-08 ダウ アグロサイエンシィズ エルエルシー 殺真菌剤としての３−アルキル−５−フルオロ−４置換イミノ−３，４−ジヒドロピリミジン−２（１ｈ）−オン誘導体
CR20160345A (es) 2013-12-31 2017-02-21 Adama Makhteshim Ltd Mezclas fungicidas sinérgicas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2(1h)-ona e inhibidor(es) de la biosíntesis de esteroles para el control fúngico
JP6585057B2 (ja) 2013-12-31 2019-10-02 アダマ・マクテシム・リミテッド ５−フルオロ−４−イミノ−３−（アルキル／置換アルキル）−１−（アリールスルホニル）−３，４−ジヒドロピリミジン−２（１ｈ）−オンおよびそれらの調製方法
AU2018320492C1 (en) 2017-07-17 2023-07-13 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
WO2020095181A1 (en) 2018-11-05 2020-05-14 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof
UY38890A (es) 2019-09-23 2021-04-30 Adama Makhteshim Ltd Procedimiento para preparar 5-(fluoro-4-imino-3-metil)-1-tosil-3,4-dihidropirimidin-(1h)-ona y derivados del compuesto
WO2021115926A1 (en) * 2019-12-10 2021-06-17 Syngenta Crop Protection Ag Methods of controlling or preventing infestation of peanut plants by phytopathogenic microorganisms

Family Cites Families (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3309359A (en) 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (OSRAM) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
GR80171B (en) 1983-08-29 1985-01-02 Ciba Geigy Ag N-(2-nitrophenyl)-4-aminopyrimidine derivatives process for the preparation thereof and use
JPS60123486A (ja) * 1983-12-09 1985-07-02 Asahi Glass Co Ltd フルオロブラストサイジンｓおよびその製法
US4845081A (en) 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
ATE109776T1 (de) 1988-03-09 1994-08-15 Ciba Geigy Ag Mittel zum schutz von pflanzen gegen krankheiten.
DE3821711A1 (de) 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3109012B2 (ja) 1992-06-18 2000-11-13 クミアイ化学工業株式会社 チアゾロ［５，４−ｄ］ピリミジン誘導体及び農園芸用殺菌剤
JP3217191B2 (ja) 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
WO1997002262A1 (en) 1995-07-05 1997-01-23 E.I. Du Pont De Nemours And Company Fungicidal pyrimidinones
PL328777A1 (en) 1996-03-11 1999-02-15 Novartis Ag Pesticides
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
WO2003018051A1 (en) 2001-08-27 2003-03-06 Vic Jira Anti-fungal composition
JPWO2005095419A1 (ja) 2004-04-01 2008-02-21 武田薬品工業株式会社 チアゾロピリミジン誘導体
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EP2252594B1 (en) 2008-01-22 2015-08-19 Dow AgroSciences LLC 4-amino-5-fluoro-pyrimidine derivatives as fungicides
EP2317851B1 (en) * 2008-08-01 2014-01-15 Dow AgroSciences LLC Use of 5-fluorocytosine as a fungicide
USRE46144E1 (en) * 2009-01-23 2016-09-13 Purdue Pharmaceutical Products L.P. Hydroxamic acid derivatives
PE20120691A1 (es) 2009-08-07 2012-06-08 Dow Agrosciences Llc Derivados de n1-sulfonil-5-fluoropirimidinona
UA107671C2 (en) * 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives

Also Published As

Publication number Publication date
EP2461686A1 (en) 2012-06-13
IL217950A0 (en) 2012-03-29
US9000002B2 (en) 2015-04-07
IL217950A (en) 2015-04-30
ES2552097T3 (es) 2015-11-25
ECSP12011652A (es) 2012-03-30
EA201270256A1 (ru) 2012-07-30
CN102497781B (zh) 2014-12-10
DK2461686T3 (en) 2016-01-18
MX2012001617A (es) 2012-04-11
CA2769656A1 (en) 2011-02-10
CO6491115A2 (es) 2012-07-31
NI201200021A (es) 2012-05-22
US20110034492A1 (en) 2011-02-10
KR101792284B1 (ko) 2017-10-31
JP2013501727A (ja) 2013-01-17
EP2461686B1 (en) 2015-10-07
UA107671C2 (en) 2015-02-10
BR112012002757A2 (pt) 2019-12-17
EP2461686A4 (en) 2013-02-13
NZ597483A (en) 2014-02-28
CA2769656C (en) 2018-05-15
WO2011017545A1 (en) 2011-02-10
PT2461686E (pt) 2015-11-18
US20140011824A1 (en) 2014-01-09
PL2461686T3 (pl) 2016-04-29
HUE027390T2 (en) 2016-10-28
US8552020B2 (en) 2013-10-08
PE20120692A1 (es) 2012-06-08
EA020910B1 (ru) 2015-02-27
CL2012000312A1 (es) 2012-10-05
IN2012DN00369A (OSRAM) 2015-08-21
CN102497781A (zh) 2012-06-13
AU2010279409A1 (en) 2012-02-02
BR112012002757B1 (pt) 2020-10-06
ZA201200813B (en) 2013-05-29
HK1171915A1 (en) 2013-04-12
CR20120032A (es) 2012-03-22
KR20120052281A (ko) 2012-05-23

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