PL2461686T3 - Pochodne N1-podstawionych 5-fluoro-2-oksopirymidynono-1(2H)-karboksyamidów - Google Patents
Pochodne N1-podstawionych 5-fluoro-2-oksopirymidynono-1(2H)-karboksyamidówInfo
- Publication number
- PL2461686T3 PL2461686T3 PL10807175T PL10807175T PL2461686T3 PL 2461686 T3 PL2461686 T3 PL 2461686T3 PL 10807175 T PL10807175 T PL 10807175T PL 10807175 T PL10807175 T PL 10807175T PL 2461686 T3 PL2461686 T3 PL 2461686T3
- Authority
- PL
- Poland
- Prior art keywords
- oxopyrimidinone
- fluoro
- substituted
- carboxamide derivatives
- carboxamide
- Prior art date
Links
- 229940053202 antiepileptics carboxamide derivative Drugs 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
- A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
- A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
- A01N47/38—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the group >N—CO—N< where at least one nitrogen atom is part of a heterocyclic ring; Thio analogues thereof
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US23224509P | 2009-08-07 | 2009-08-07 | |
| PCT/US2010/044588 WO2011017545A1 (en) | 2009-08-07 | 2010-08-05 | N1-substituted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives |
| EP10807175.4A EP2461686B1 (en) | 2009-08-07 | 2010-08-05 | N1-substituted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PL2461686T3 true PL2461686T3 (pl) | 2016-04-29 |
Family
ID=43535294
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PL10807175T PL2461686T3 (pl) | 2009-08-07 | 2010-08-05 | Pochodne N1-podstawionych 5-fluoro-2-oksopirymidynono-1(2H)-karboksyamidów |
Country Status (26)
| Country | Link |
|---|---|
| US (2) | US8552020B2 (OSRAM) |
| EP (1) | EP2461686B1 (OSRAM) |
| JP (1) | JP5735510B2 (OSRAM) |
| KR (1) | KR101792284B1 (OSRAM) |
| CN (1) | CN102497781B (OSRAM) |
| BR (1) | BR112012002757B1 (OSRAM) |
| CA (1) | CA2769656C (OSRAM) |
| CL (1) | CL2012000312A1 (OSRAM) |
| CO (1) | CO6491115A2 (OSRAM) |
| CR (1) | CR20120032A (OSRAM) |
| DK (1) | DK2461686T3 (OSRAM) |
| EA (1) | EA020910B1 (OSRAM) |
| EC (1) | ECSP12011652A (OSRAM) |
| ES (1) | ES2552097T3 (OSRAM) |
| HU (1) | HUE027390T2 (OSRAM) |
| IL (1) | IL217950A (OSRAM) |
| IN (1) | IN2012DN00369A (OSRAM) |
| MX (1) | MX2012001617A (OSRAM) |
| NI (1) | NI201200021A (OSRAM) |
| NZ (1) | NZ597483A (OSRAM) |
| PE (1) | PE20120692A1 (OSRAM) |
| PL (1) | PL2461686T3 (OSRAM) |
| PT (1) | PT2461686E (OSRAM) |
| UA (1) | UA107671C2 (OSRAM) |
| WO (1) | WO2011017545A1 (OSRAM) |
| ZA (1) | ZA201200813B (OSRAM) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NZ597644A (en) * | 2009-08-07 | 2014-05-30 | Dow Agrosciences Llc | N1-sulfonyl-5-fluoropyrimidinone derivatives |
| PL2461688T3 (pl) | 2009-08-07 | 2017-08-31 | Dow Agrosciences Llc | Kompozycje szkodnikobójcze |
| UA107671C2 (en) * | 2009-08-07 | 2015-02-10 | Dow Agrosciences Llc | N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives |
| US9321734B2 (en) | 2012-12-28 | 2016-04-26 | Dow Agrosciences Llc | N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2H)-carboxamide derivatives |
| HK1214518A1 (zh) * | 2012-12-28 | 2016-07-29 | Adama Makhteshim Ltd. | 1-(经取代之苯甲醯基)-5-氟-4-亚胺基-3-甲基-3,4-二氢嘧啶-2(1h)-酮衍生物 |
| CN104902757B (zh) | 2012-12-28 | 2019-01-08 | 阿达玛马克西姆股份有限公司 | N-(取代的)-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1(2h)-羧酸酯衍生物 |
| CN105007737A (zh) | 2012-12-31 | 2015-10-28 | 美国陶氏益农公司 | 作为杀真菌剂的3-烷基-5-氟-4-取代的-亚氨基-3,4-二氢嘧啶-2(1h)-酮衍生物 |
| PE20161174A1 (es) | 2013-12-31 | 2016-10-26 | Adama Makhteshim Ltd | 5-fluor-4-imino-3-(alquil/alquilo sustituido)-1-(arilsulfonil)-3,4-dihidropirimidin-2(1h)-ona y los procesos para su preparacion |
| CN106061262A (zh) | 2013-12-31 | 2016-10-26 | 阿达玛马克西姆股份有限公司 | 用防治谷类中真菌的协同杀真菌混合物 |
| WO2019038583A1 (en) | 2017-07-17 | 2019-02-28 | Adama Makhteshim Ltd. | 5-FLUORO-4-IMINO-3-METHYL-1-TOSYL-3,4-DIHYDROPYRIMIDIN-2-ONE POLYMORPHS |
| MX2021005283A (es) | 2018-11-05 | 2021-06-18 | Adama Makhteshim Ltd | Mezclas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1- tosil-3,4-dihidropirimidin-2-ona, y metodos de uso de los mismos. |
| US12466796B2 (en) | 2019-09-23 | 2025-11-11 | Adama Makhteshim Ltd. | Process for preparing 5-(fluoro-4-imino-3-methyl)-1-tosyl-3,4 dihydropyrimidine-(1H)-one and derivatives of the compound |
Family Cites Families (24)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3309359A (en) * | 1965-10-22 | 1967-03-14 | Hoffmann La Roche | N-mono-acyl-5-fluorocytosine derivatives and process |
| US3368938A (en) | 1966-01-13 | 1968-02-13 | Hoffmann La Roche | Controlling fungi with 5-fluorocytosine |
| US3868373A (en) | 1970-01-27 | 1975-02-25 | Hoffmann La Roche | 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines |
| CH579057A5 (OSRAM) | 1973-09-07 | 1976-08-31 | Hoffmann La Roche | |
| FR2530636A1 (fr) | 1982-07-23 | 1984-01-27 | Rhone Poulenc Agrochimie | Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides |
| EP0139613A1 (de) | 1983-08-29 | 1985-05-02 | Ciba-Geigy Ag | N-(2-Nitrophenyl)-4-aminopyrimidin-Derivate, deren Herstellung und Verwendung |
| JPS60123486A (ja) | 1983-12-09 | 1985-07-02 | Asahi Glass Co Ltd | フルオロブラストサイジンsおよびその製法 |
| US4845081A (en) | 1984-10-18 | 1989-07-04 | University Of Florida | Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes |
| ES2057172T3 (es) | 1988-03-09 | 1994-10-16 | Ciba Geigy Ag | Agente para la proteccion de plantas contra enfermedades. |
| DE3821711A1 (de) | 1988-06-28 | 1990-02-08 | Bayer Ag | Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel |
| JP3109012B2 (ja) | 1992-06-18 | 2000-11-13 | クミアイ化学工業株式会社 | チアゾロ[5,4−d]ピリミジン誘導体及び農園芸用殺菌剤 |
| JP3217191B2 (ja) | 1992-07-16 | 2001-10-09 | ビーエーエスエフ アクチェンゲゼルシャフト | ヘテロ芳香族化合物およびこれを含有する植物保護剤 |
| WO1997002262A1 (en) * | 1995-07-05 | 1997-01-23 | E.I. Du Pont De Nemours And Company | Fungicidal pyrimidinones |
| DE69712331T2 (de) | 1996-03-11 | 2002-11-28 | Syngenta Participations Ag, Basel | Pyrimidin-4-on derivate als pestizidesmittel |
| HRP970239B1 (en) | 1997-05-09 | 2004-04-30 | Inst Ru Er Bouekovic | Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity |
| GT199900185A (es) | 1998-11-06 | 2001-04-18 | Novedosa pirimidin-4-enamina como fungicida. | |
| US7914799B2 (en) | 2001-08-27 | 2011-03-29 | Immunitor USA, Inc. | Anti-fungal composition |
| JPWO2005095419A1 (ja) | 2004-04-01 | 2008-02-21 | 武田薬品工業株式会社 | チアゾロピリミジン誘導体 |
| WO2008005303A2 (en) | 2006-06-30 | 2008-01-10 | Janssen Pharmaceutica N.V. | Thiazolopyrimidine modulators of trpv1 |
| PT2252594E (pt) | 2008-01-22 | 2015-11-30 | Dow Agrosciences Llc | Derivados de 5-fluoro-pirimidina como fungicidas |
| CN102215691B (zh) * | 2008-08-01 | 2015-02-04 | 陶氏益农公司 | 5-氟胞嘧啶作为杀真菌剂的用途 |
| JP5576402B2 (ja) * | 2009-01-23 | 2014-08-20 | ユーロ−セルティーク エス.エイ. | ヒドロキサム酸誘導体 |
| NZ597644A (en) | 2009-08-07 | 2014-05-30 | Dow Agrosciences Llc | N1-sulfonyl-5-fluoropyrimidinone derivatives |
| UA107671C2 (en) * | 2009-08-07 | 2015-02-10 | Dow Agrosciences Llc | N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives |
-
2010
- 2010-05-08 UA UAA201202732A patent/UA107671C2/ru unknown
- 2010-08-05 DK DK10807175.4T patent/DK2461686T3/en active
- 2010-08-05 WO PCT/US2010/044588 patent/WO2011017545A1/en not_active Ceased
- 2010-08-05 CA CA2769656A patent/CA2769656C/en not_active Expired - Fee Related
- 2010-08-05 PE PE2012000171A patent/PE20120692A1/es not_active Application Discontinuation
- 2010-08-05 NZ NZ597483A patent/NZ597483A/en unknown
- 2010-08-05 IN IN369DEN2012 patent/IN2012DN00369A/en unknown
- 2010-08-05 PL PL10807175T patent/PL2461686T3/pl unknown
- 2010-08-05 HU HUE10807175A patent/HUE027390T2/en unknown
- 2010-08-05 ES ES10807175.4T patent/ES2552097T3/es active Active
- 2010-08-05 KR KR1020127003168A patent/KR101792284B1/ko not_active Expired - Fee Related
- 2010-08-05 BR BR112012002757-3A patent/BR112012002757B1/pt active IP Right Grant
- 2010-08-05 EP EP10807175.4A patent/EP2461686B1/en active Active
- 2010-08-05 MX MX2012001617A patent/MX2012001617A/es active IP Right Grant
- 2010-08-05 EA EA201270256A patent/EA020910B1/ru not_active IP Right Cessation
- 2010-08-05 PT PT108071754T patent/PT2461686E/pt unknown
- 2010-08-05 CN CN201080034900.8A patent/CN102497781B/zh active Active
- 2010-08-05 JP JP2012523955A patent/JP5735510B2/ja active Active
- 2010-08-05 US US12/851,331 patent/US8552020B2/en active Active
-
2012
- 2012-01-18 CR CR20120032A patent/CR20120032A/es unknown
- 2012-02-02 ZA ZA2012/00813A patent/ZA201200813B/en unknown
- 2012-02-03 NI NI201200021A patent/NI201200021A/es unknown
- 2012-02-05 IL IL217950A patent/IL217950A/en active IP Right Grant
- 2012-02-06 CO CO12019947A patent/CO6491115A2/es active IP Right Grant
- 2012-02-06 CL CL2012000312A patent/CL2012000312A1/es unknown
- 2012-02-07 EC ECSP12011652 patent/ECSP12011652A/es unknown
-
2013
- 2013-09-12 US US14/024,795 patent/US9000002B2/en active Active
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