DK2461686T3 - N1-SUBSTITUTED 5-FLUORO-2-OXOPYRIMIDINON-1 (2H) CARBOXAMIDE DERIVATIVES - Google Patents

N1-SUBSTITUTED 5-FLUORO-2-OXOPYRIMIDINON-1 (2H) CARBOXAMIDE DERIVATIVES Download PDF

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Publication number
DK2461686T3
DK2461686T3 DK10807175.4T DK10807175T DK2461686T3 DK 2461686 T3 DK2461686 T3 DK 2461686T3 DK 10807175 T DK10807175 T DK 10807175T DK 2461686 T3 DK2461686 T3 DK 2461686T3
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DK
Denmark
Prior art keywords
optionally substituted
benzyl
alkyl
phenyl
ring system
Prior art date
Application number
DK10807175.4T
Other languages
Danish (da)
English (en)
Inventor
Timothy Boebel
Kristy Bryan
Beth Lorsbach
Timothy Martin
W Owen
Mark Pobanz
Scott Thornburgh
Jeffery Webster
Chenglin Yao
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535294&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK2461686(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Application granted granted Critical
Publication of DK2461686T3 publication Critical patent/DK2461686T3/en

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Classifications

    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A01N47/38Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the group >N—CO—N< where at least one nitrogen atom is part of a heterocyclic ring; Thio analogues thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK10807175.4T 2009-08-07 2010-08-05 N1-SUBSTITUTED 5-FLUORO-2-OXOPYRIMIDINON-1 (2H) CARBOXAMIDE DERIVATIVES DK2461686T3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23224509P 2009-08-07 2009-08-07
PCT/US2010/044588 WO2011017545A1 (en) 2009-08-07 2010-08-05 N1-substituted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives

Publications (1)

Publication Number Publication Date
DK2461686T3 true DK2461686T3 (en) 2016-01-18

Family

ID=43535294

Family Applications (1)

Application Number Title Priority Date Filing Date
DK10807175.4T DK2461686T3 (en) 2009-08-07 2010-08-05 N1-SUBSTITUTED 5-FLUORO-2-OXOPYRIMIDINON-1 (2H) CARBOXAMIDE DERIVATIVES

Country Status (26)

Country Link
US (2) US8552020B2 (OSRAM)
EP (1) EP2461686B1 (OSRAM)
JP (1) JP5735510B2 (OSRAM)
KR (1) KR101792284B1 (OSRAM)
CN (1) CN102497781B (OSRAM)
BR (1) BR112012002757B1 (OSRAM)
CA (1) CA2769656C (OSRAM)
CL (1) CL2012000312A1 (OSRAM)
CO (1) CO6491115A2 (OSRAM)
CR (1) CR20120032A (OSRAM)
DK (1) DK2461686T3 (OSRAM)
EA (1) EA020910B1 (OSRAM)
EC (1) ECSP12011652A (OSRAM)
ES (1) ES2552097T3 (OSRAM)
HU (1) HUE027390T2 (OSRAM)
IL (1) IL217950A (OSRAM)
IN (1) IN2012DN00369A (OSRAM)
MX (1) MX2012001617A (OSRAM)
NI (1) NI201200021A (OSRAM)
NZ (1) NZ597483A (OSRAM)
PE (1) PE20120692A1 (OSRAM)
PL (1) PL2461686T3 (OSRAM)
PT (1) PT2461686E (OSRAM)
UA (1) UA107671C2 (OSRAM)
WO (1) WO2011017545A1 (OSRAM)
ZA (1) ZA201200813B (OSRAM)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
UA107671C2 (en) * 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
UA106764C2 (uk) * 2009-08-07 2014-10-10 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні n1-сульфоніл-5-фторпіримідинону
CN102548411B (zh) 2009-08-07 2014-07-02 陶氏益农公司 杀虫组合物
US9271497B2 (en) * 2012-12-28 2016-03-01 Dow Agrosciences Llc 1-(substituted-benzoyl)-5-fluoro-4-imino-3-methyl-3,4-dihydropyrimidin-2(1H)-one derivatives
US9321734B2 (en) * 2012-12-28 2016-04-26 Dow Agrosciences Llc N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2H)-carboxamide derivatives
CA2893778A1 (en) * 2012-12-28 2014-07-03 Dow Agrosciences Llc N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2h)-carboxylate derivatives
PL2953463T3 (pl) 2012-12-31 2022-01-03 Adama Makhteshim Ltd. Pochodne 3-alkilo-5-fluoro-4-podstawione-imino-3,4-dihydropirymidyn-2(1h)-onu jako środki grzybobójcze
EA030030B1 (ru) 2013-12-31 2018-06-29 Адама Мактешим Лтд. Синергетические фунгицидные смеси и синергетические фунгицидные композиции для борьбы с грибами
EA036389B1 (ru) 2013-12-31 2020-11-03 Адама Мактешим Лтд. 5-фтор-4-имино-3-(алкил/замещенный алкил)-1-(арилсульфонил)-3,4-дигидропиримидин-2(1h)-он и способы их получения
CN118515619A (zh) 2017-07-17 2024-08-20 阿达玛克西姆股份有限公司 5-氟-4-亚氨基-3-甲基-1-甲苯磺酰基-3,4-二氢嘧啶-2-酮的多晶型物
AU2019374510A1 (en) 2018-11-05 2021-06-17 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof

Family Cites Families (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3309359A (en) * 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) * 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (OSRAM) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
EP0139613A1 (de) 1983-08-29 1985-05-02 Ciba-Geigy Ag N-(2-Nitrophenyl)-4-aminopyrimidin-Derivate, deren Herstellung und Verwendung
JPS60123486A (ja) 1983-12-09 1985-07-02 Asahi Glass Co Ltd フルオロブラストサイジンsおよびその製法
US4845081A (en) * 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
ATE109776T1 (de) 1988-03-09 1994-08-15 Ciba Geigy Ag Mittel zum schutz von pflanzen gegen krankheiten.
DE3821711A1 (de) * 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3109012B2 (ja) 1992-06-18 2000-11-13 クミアイ化学工業株式会社 チアゾロ[5,4−d]ピリミジン誘導体及び農園芸用殺菌剤
JP3217191B2 (ja) * 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
DE69618959T2 (de) * 1995-07-05 2002-08-29 E.I. Du Pont De Nemours And Co., Wilmington Pyrimidone und ihre verwendug als fungizide
ATE216999T1 (de) 1996-03-11 2002-05-15 Syngenta Participations Ag Pyrimidin-4-on derivate als pestizidesmittel
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
US7914799B2 (en) * 2001-08-27 2011-03-29 Immunitor USA, Inc. Anti-fungal composition
JPWO2005095419A1 (ja) * 2004-04-01 2008-02-21 武田薬品工業株式会社 チアゾロピリミジン誘導体
EP2044086A2 (en) * 2006-06-30 2009-04-08 Janssen Pharmaceutica N.V. Thiazolopyrimidine modulators of trpv1
EP2562165A1 (en) 2008-01-22 2013-02-27 Dow AgroSciences LLC 5-fluoro pyrimidine derivatives as fungicides
US20100029482A1 (en) * 2008-08-01 2010-02-04 Benko Zoltan L Use of 5-fluorocytosine as a fungicide
ME02254B (me) * 2009-01-23 2015-12-31 Euro Celtique Sa Derivati hidroksamske kiseline
UA107671C2 (en) * 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
UA106764C2 (uk) * 2009-08-07 2014-10-10 ДАУ АГРОСАЙЄНСІЗ ЕлЕлСі Похідні n1-сульфоніл-5-фторпіримідинону

Also Published As

Publication number Publication date
NZ597483A (en) 2014-02-28
WO2011017545A1 (en) 2011-02-10
ECSP12011652A (es) 2012-03-30
EP2461686A4 (en) 2013-02-13
PT2461686E (pt) 2015-11-18
CA2769656A1 (en) 2011-02-10
US20140011824A1 (en) 2014-01-09
BR112012002757A2 (pt) 2019-12-17
BR112012002757B1 (pt) 2020-10-06
PE20120692A1 (es) 2012-06-08
MX2012001617A (es) 2012-04-11
CL2012000312A1 (es) 2012-10-05
CN102497781B (zh) 2014-12-10
JP2013501727A (ja) 2013-01-17
CR20120032A (es) 2012-03-22
KR20120052281A (ko) 2012-05-23
IL217950A0 (en) 2012-03-29
NI201200021A (es) 2012-05-22
PL2461686T3 (pl) 2016-04-29
US9000002B2 (en) 2015-04-07
HUE027390T2 (en) 2016-10-28
EA020910B1 (ru) 2015-02-27
CA2769656C (en) 2018-05-15
IN2012DN00369A (OSRAM) 2015-08-21
KR101792284B1 (ko) 2017-10-31
CO6491115A2 (es) 2012-07-31
HK1171915A1 (en) 2013-04-12
ES2552097T3 (es) 2015-11-25
UA107671C2 (en) 2015-02-10
EP2461686A1 (en) 2012-06-13
ZA201200813B (en) 2013-05-29
IL217950A (en) 2015-04-30
EA201270256A1 (ru) 2012-07-30
JP5735510B2 (ja) 2015-06-17
EP2461686B1 (en) 2015-10-07
US20110034492A1 (en) 2011-02-10
AU2010279409A1 (en) 2012-02-02
US8552020B2 (en) 2013-10-08
CN102497781A (zh) 2012-06-13

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