PT2461686E - Derivados de 5-fluoro-2-oxopirimidinona-1(2h)-carboxamida substituídos em n1 - Google Patents

Derivados de 5-fluoro-2-oxopirimidinona-1(2h)-carboxamida substituídos em n1 Download PDF

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Publication number
PT2461686E
PT2461686E PT108071754T PT10807175T PT2461686E PT 2461686 E PT2461686 E PT 2461686E PT 108071754 T PT108071754 T PT 108071754T PT 10807175 T PT10807175 T PT 10807175T PT 2461686 E PT2461686 E PT 2461686E
Authority
PT
Portugal
Prior art keywords
oxopyrimidinone
fluoro
substituted
carboxamide derivatives
carboxamide
Prior art date
Application number
PT108071754T
Other languages
English (en)
Portuguese (pt)
Inventor
Chenglin Yao
Timothy Boebel
Kristy Bryan
Beth Lorsbach
Timothy Martin
W Owen
Mark Pobanz
Scott Thornburgh
Jeffery Webster
Original Assignee
Dow Agrosciences Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535294&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=PT2461686(E) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dow Agrosciences Llc filed Critical Dow Agrosciences Llc
Publication of PT2461686E publication Critical patent/PT2461686E/pt

Links

Classifications

    • AHUMAN NECESSITIES
    • A01AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01NPRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A01N47/38Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the group >N—CO—N< where at least one nitrogen atom is part of a heterocyclic ring; Thio analogues thereof
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D239/00Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D409/00Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/12Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Dentistry (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
PT108071754T 2009-08-07 2010-08-05 Derivados de 5-fluoro-2-oxopirimidinona-1(2h)-carboxamida substituídos em n1 PT2461686E (pt)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US23224509P 2009-08-07 2009-08-07

Publications (1)

Publication Number Publication Date
PT2461686E true PT2461686E (pt) 2015-11-18

Family

ID=43535294

Family Applications (1)

Application Number Title Priority Date Filing Date
PT108071754T PT2461686E (pt) 2009-08-07 2010-08-05 Derivados de 5-fluoro-2-oxopirimidinona-1(2h)-carboxamida substituídos em n1

Country Status (26)

Country Link
US (2) US8552020B2 (OSRAM)
EP (1) EP2461686B1 (OSRAM)
JP (1) JP5735510B2 (OSRAM)
KR (1) KR101792284B1 (OSRAM)
CN (1) CN102497781B (OSRAM)
BR (1) BR112012002757B1 (OSRAM)
CA (1) CA2769656C (OSRAM)
CL (1) CL2012000312A1 (OSRAM)
CO (1) CO6491115A2 (OSRAM)
CR (1) CR20120032A (OSRAM)
DK (1) DK2461686T3 (OSRAM)
EA (1) EA020910B1 (OSRAM)
EC (1) ECSP12011652A (OSRAM)
ES (1) ES2552097T3 (OSRAM)
HU (1) HUE027390T2 (OSRAM)
IL (1) IL217950A (OSRAM)
IN (1) IN2012DN00369A (OSRAM)
MX (1) MX2012001617A (OSRAM)
NI (1) NI201200021A (OSRAM)
NZ (1) NZ597483A (OSRAM)
PE (1) PE20120692A1 (OSRAM)
PL (1) PL2461686T3 (OSRAM)
PT (1) PT2461686E (OSRAM)
UA (1) UA107671C2 (OSRAM)
WO (1) WO2011017545A1 (OSRAM)
ZA (1) ZA201200813B (OSRAM)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ES2471371T3 (es) * 2009-08-07 2014-06-26 Dow Agrosciences Llc Derivados de N1-sulfonil-5-fluoropirimidinona
JP5771207B2 (ja) 2009-08-07 2015-08-26 ダウ アグロサイエンシィズ エルエルシー 有害生物防除組成物
UA107671C2 (en) * 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives
WO2014105844A1 (en) * 2012-12-28 2014-07-03 Dow Agrosciences Llc N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2h)-carboxylate derivatives
CN104884062B (zh) * 2012-12-28 2018-11-06 阿达玛马克西姆股份有限公司 N-(取代的)-5-氟-4-亚氨基-3-甲基-2-氧代-3,4-二氢嘧啶-1(2h)-甲酰胺衍生物
MX2015008443A (es) * 2012-12-28 2015-09-23 Dow Agrosciences Llc Derivados de 1-(benzoilo-sustituido) -5-fluoro-4-imino-3-metil-3, 4-dihidropirimidin-2 (1h)-ona.
NZ749557A (en) 2012-12-31 2020-01-31 Adama Makhteshim Ltd 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides
CN106028816A (zh) 2013-12-31 2016-10-12 阿达玛马克西姆股份有限公司 用防治谷类中真菌的协同杀真菌混合物
NZ722439A (en) 2013-12-31 2018-01-26 Adama Makhteshim Ltd 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1- (arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
AU2018320492C1 (en) 2017-07-17 2023-07-13 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
EP3876717A1 (en) 2018-11-05 2021-09-15 Adama Makhteshim Ltd. Mixtures and compositions comprising 5-fluoro-4-imino-3- methyl-1-tosyl-3,4-dihydropyrimidin-2-one, and methods of use thereof

Family Cites Families (24)

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US3309359A (en) * 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) * 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (OSRAM) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
EP0139613A1 (de) 1983-08-29 1985-05-02 Ciba-Geigy Ag N-(2-Nitrophenyl)-4-aminopyrimidin-Derivate, deren Herstellung und Verwendung
JPS60123486A (ja) * 1983-12-09 1985-07-02 Asahi Glass Co Ltd フルオロブラストサイジンsおよびその製法
US4845081A (en) * 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
DE58908159D1 (de) 1988-03-09 1994-09-15 Ciba Geigy Ag Mittel zum Schutz von Pflanzen gegen Krankheiten.
DE3821711A1 (de) * 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3109012B2 (ja) 1992-06-18 2000-11-13 クミアイ化学工業株式会社 チアゾロ[5,4−d]ピリミジン誘導体及び農園芸用殺菌剤
JP3217191B2 (ja) * 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
EP0836602B1 (en) * 1995-07-05 2002-01-30 E.I. Du Pont De Nemours And Company Fungicidal pyrimidinones
TR199801813T2 (xx) 1996-03-11 1998-12-21 Novartis Ag B�cek �ld�r�c� olarak pirimidin-4- on t�revleri.
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) * 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
US7914799B2 (en) * 2001-08-27 2011-03-29 Immunitor USA, Inc. Anti-fungal composition
EP1731523A4 (en) * 2004-04-01 2009-08-12 Takeda Pharmaceutical THIAZOLOPYRIMIDINDERIVAT
EP2044086A2 (en) * 2006-06-30 2009-04-08 Janssen Pharmaceutica N.V. Thiazolopyrimidine modulators of trpv1
EP2562175A1 (en) * 2008-01-22 2013-02-27 Dow AgroSciences LLC 5-fluoro pyrimidine derivatives as fungicides
ES2456272T3 (es) 2008-08-01 2014-04-21 Dow Agrosciences Llc Uso de 5-fluorocitosina como un fungicida
SI2389375T1 (sl) * 2009-01-23 2015-11-30 Euro-Celtique S.A. Derivati hidroksamske kisline
ES2471371T3 (es) * 2009-08-07 2014-06-26 Dow Agrosciences Llc Derivados de N1-sulfonil-5-fluoropirimidinona
UA107671C2 (en) * 2009-08-07 2015-02-10 Dow Agrosciences Llc N1-substityted-5-fluoro-2-oxopyrimidinone-1(2h)-carboxamide derivatives

Also Published As

Publication number Publication date
CA2769656A1 (en) 2011-02-10
ZA201200813B (en) 2013-05-29
ES2552097T3 (es) 2015-11-25
NI201200021A (es) 2012-05-22
EP2461686A4 (en) 2013-02-13
MX2012001617A (es) 2012-04-11
US20110034492A1 (en) 2011-02-10
BR112012002757A2 (pt) 2019-12-17
IL217950A (en) 2015-04-30
AU2010279409A1 (en) 2012-02-02
US9000002B2 (en) 2015-04-07
JP2013501727A (ja) 2013-01-17
IN2012DN00369A (OSRAM) 2015-08-21
WO2011017545A1 (en) 2011-02-10
CR20120032A (es) 2012-03-22
HUE027390T2 (en) 2016-10-28
UA107671C2 (en) 2015-02-10
EP2461686A1 (en) 2012-06-13
ECSP12011652A (es) 2012-03-30
PL2461686T3 (pl) 2016-04-29
CA2769656C (en) 2018-05-15
PE20120692A1 (es) 2012-06-08
CN102497781A (zh) 2012-06-13
BR112012002757B1 (pt) 2020-10-06
NZ597483A (en) 2014-02-28
IL217950A0 (en) 2012-03-29
DK2461686T3 (en) 2016-01-18
EA201270256A1 (ru) 2012-07-30
US8552020B2 (en) 2013-10-08
EA020910B1 (ru) 2015-02-27
KR101792284B1 (ko) 2017-10-31
CN102497781B (zh) 2014-12-10
HK1171915A1 (en) 2013-04-12
KR20120052281A (ko) 2012-05-23
CL2012000312A1 (es) 2012-10-05
CO6491115A2 (es) 2012-07-31
EP2461686B1 (en) 2015-10-07
JP5735510B2 (ja) 2015-06-17
US20140011824A1 (en) 2014-01-09

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