JP5684896B2 - ピラゾールカルボン酸アミドの調製方法 - Google Patents

ピラゾールカルボン酸アミドの調製方法 Download PDF

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JP5684896B2
JP5684896B2 JP2013505409A JP2013505409A JP5684896B2 JP 5684896 B2 JP5684896 B2 JP 5684896B2 JP 2013505409 A JP2013505409 A JP 2013505409A JP 2013505409 A JP2013505409 A JP 2013505409A JP 5684896 B2 JP5684896 B2 JP 5684896B2
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formula
compound
chloro
bromo
palladium
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JP2013525317A5 (enExample
JP2013525317A (ja
Inventor
ドゥムニアー ラファエル
ドゥムニアー ラファエル
シュレト フロリアン
シュレト フロリアン
フェティガー トマス
フェティガー トマス
ロメル ミヒャエル
ロメル ミヒャエル
トラー シュテファン
トラー シュテファン
Original Assignee
シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト
シンジェンタ パーティシペーションズ アクチェンゲゼルシャフト
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00—Preparation of halogenated hydrocarbons
    • C07C17/23—Preparation of halogenated hydrocarbons by dehalogenation
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00—Preparation of halogenated hydrocarbons
    • C07C17/26—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton
    • C07C17/30—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton by a Diels-Alder synthesis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C209/00—Preparation of compounds containing amino groups bound to a carbon skeleton
    • C07C209/04—Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups
    • C07C209/06—Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups by substitution of halogen atoms
    • C07C209/10—Preparation of compounds containing amino groups bound to a carbon skeleton by substitution of functional groups by amino groups by substitution of halogen atoms with formation of amino groups bound to carbon atoms of six-membered aromatic rings or from amines having nitrogen atoms bound to carbon atoms of six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C25/00—Compounds containing at least one halogen atom bound to a six-membered aromatic ring
    • C07C25/24—Halogenated aromatic hydrocarbons with unsaturated side chains
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C29/00—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring
    • C07C29/132—Preparation of compounds having hydroxy or O-metal groups bound to a carbon atom not belonging to a six-membered aromatic ring by reduction of an oxygen containing functional group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C35/00—Compounds having at least one hydroxy or O-metal group bound to a carbon atom of a ring other than a six-membered aromatic ring
    • C07C35/48—Halogenated derivatives
    • C07C35/52—Alcohols with a condensed ring system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
    • C07C45/27—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by oxidation
    • C07C45/29—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by oxidation of hydroxy groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D303/00—Compounds containing three-membered rings having one oxygen atom as the only ring hetero atom
    • C07D303/02—Compounds containing oxirane rings
    • C07D303/12—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms
    • C07D303/16—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms by esterified hydroxyl radicals
    • C07D303/17—Compounds containing oxirane rings with hydrocarbon radicals, substituted by singly or doubly bound oxygen atoms by esterified hydroxyl radicals containing oxirane rings condensed with carbocyclic ring systems having three or more relevant rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/56—Ring systems containing bridged rings
    • C07C2603/58—Ring systems containing bridged rings containing three rings
    • C07C2603/60—Ring systems containing bridged rings containing three rings containing at least one ring with less than six members
    • C07C2603/66—Ring systems containing bridged rings containing three rings containing at least one ring with less than six members containing five-membered rings

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Catalysts (AREA)
  • Epoxy Compounds (AREA)
JP2013505409A 2010-04-20 2011-04-14 ピラゾールカルボン酸アミドの調製方法 Active JP5684896B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP10160438 2010-04-20
EP10160438.7 2010-04-20
PCT/EP2011/055871 WO2011131545A1 (en) 2010-04-20 2011-04-14 Process for the preparation of pyrazole carboxylic acid amides

Publications (3)

Publication Number Publication Date
JP2013525317A JP2013525317A (ja) 2013-06-20
JP2013525317A5 JP2013525317A5 (enExample) 2014-03-13
JP5684896B2 true JP5684896B2 (ja) 2015-03-18

Family

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Family Applications (1)

Application Number Title Priority Date Filing Date
JP2013505409A Active JP5684896B2 (ja) 2010-04-20 2011-04-14 ピラゾールカルボン酸アミドの調製方法

Country Status (12)

Country Link
US (1) US8519152B2 (enExample)
EP (1) EP2560959B1 (enExample)
JP (1) JP5684896B2 (enExample)
CN (1) CN102906072B (enExample)
AR (1) AR080922A1 (enExample)
BR (1) BR112012026631B1 (enExample)
ES (1) ES2513540T3 (enExample)
IL (1) IL222398A (enExample)
MX (1) MX2012012005A (enExample)
TW (1) TWI428325B (enExample)
UY (1) UY33340A (enExample)
WO (1) WO2011131545A1 (enExample)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2011131544A1 (en) * 2010-04-20 2011-10-27 Syngenta Participations Ag Process for the preparation of pyrazole carboxylic acid amides
TWI534126B (zh) * 2011-01-25 2016-05-21 先正達合夥公司 用於製備吡唑羧酸醯胺之方法
GB201403438D0 (en) 2014-02-27 2014-04-16 Syngenta Participations Ag Polymorphs
AU2023309261A1 (en) 2022-07-22 2024-12-12 Syngenta Crop Protection Ag Solid form of a heterocyclic amide derivative
CN116143635B (zh) * 2022-12-01 2025-02-25 江苏七洲绿色科技研究院有限公司 一种9-二氯亚甲基-5-氨基-苯并降冰片烯的制备方法
WO2025157998A1 (en) 2024-01-26 2025-07-31 Syngenta Crop Protection Ag Chemical process

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH075487B2 (ja) 1985-11-14 1995-01-25 住友化学工業株式会社 １―ブロモ―２―クロロ―４―フルオロベンゼンの製造法
US5093347A (en) 1991-01-28 1992-03-03 Monsanto Company 3-difluoromethylpyrazolecarboxamide fungicides, compositions and use
US7223879B2 (en) 1998-07-10 2007-05-29 Massachusetts Institute Of Technology Ligands for metals and improved metal-catalyzed processes based thereon
GEP20115161B (en) * 2005-10-25 2011-02-10 Syngenta Participations Ag Heterocyclic amide derivatives useful as microbiocides
WO2007124907A2 (en) 2006-04-27 2007-11-08 Syngenta Participations Ag Heterocyclyl-carboxylic acid (benzonorbornene-5-yl)amide derivatives as fungicides for agrochemical use
EP2076123B1 (en) 2006-10-25 2011-06-01 Syngenta Limited Process for the production of substituted bromobenzenes
EP2370412A1 (en) * 2008-12-24 2011-10-05 Syngenta Limited Methods for the preparation of fungicides

Also Published As

Publication number Publication date
MX2012012005A (es) 2012-12-17
IL222398A (en) 2017-01-31
BR112012026631B1 (pt) 2017-07-25
EP2560959A1 (en) 2013-02-27
CN102906072A (zh) 2013-01-30
UY33340A (es) 2011-12-01
ES2513540T3 (es) 2014-10-27
US8519152B2 (en) 2013-08-27
JP2013525317A (ja) 2013-06-20
EP2560959B1 (en) 2014-08-20
CN102906072B (zh) 2014-07-02
WO2011131545A1 (en) 2011-10-27
TWI428325B (zh) 2014-03-01
BR112012026631A2 (pt) 2015-09-15
AR080922A1 (es) 2012-05-16
US20130035496A1 (en) 2013-02-07
TW201204704A (en) 2012-02-01

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