JP5627038B2 - ピリジン環含有化合物 - Google Patents
ピリジン環含有化合物 Download PDFInfo
- Publication number
- JP5627038B2 JP5627038B2 JP2012504543A JP2012504543A JP5627038B2 JP 5627038 B2 JP5627038 B2 JP 5627038B2 JP 2012504543 A JP2012504543 A JP 2012504543A JP 2012504543 A JP2012504543 A JP 2012504543A JP 5627038 B2 JP5627038 B2 JP 5627038B2
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- JP
- Japan
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- unsubstituted
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- reaction
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
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- 0 *N(*)c1nc(CBr)ccc1 Chemical compound *N(*)c1nc(CBr)ccc1 0.000 description 2
- RTLXKGJMDMNDDA-UHFFFAOYSA-N CCc1nc(N(C(C)=O)C(OC(C)(C)C)=O)ccc1 Chemical compound CCc1nc(N(C(C)=O)C(OC(C)(C)C)=O)ccc1 RTLXKGJMDMNDDA-UHFFFAOYSA-N 0.000 description 1
- IHGPXLROZCMMHE-UHFFFAOYSA-N C[n]1nnnc1C(c1ccccc1)=N Chemical compound C[n]1nnnc1C(c1ccccc1)=N IHGPXLROZCMMHE-UHFFFAOYSA-N 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
- C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
- C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pyridine Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2012504543A JP5627038B2 (ja) | 2010-03-12 | 2011-03-11 | ピリジン環含有化合物 |
Applications Claiming Priority (8)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2010056718 | 2010-03-12 | ||
| JP2010056718 | 2010-03-12 | ||
| JP2010115703 | 2010-05-19 | ||
| JP2010115703 | 2010-05-19 | ||
| JP2010127207 | 2010-06-02 | ||
| JP2010127207 | 2010-06-02 | ||
| JP2012504543A JP5627038B2 (ja) | 2010-03-12 | 2011-03-11 | ピリジン環含有化合物 |
| PCT/JP2011/055809 WO2011111831A1 (ja) | 2010-03-12 | 2011-03-11 | ピリジン環含有化合物、及びハロゲン化ピコリン誘導体及びテトラゾリルオキシム誘導体の製造方法 |
Related Child Applications (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014025954A Division JP5793589B2 (ja) | 2010-03-12 | 2014-02-13 | 臭化ピコリン誘導体の製造方法 |
| JP2014025952A Division JP5695233B2 (ja) | 2010-03-12 | 2014-02-13 | テトラゾリルオキシム誘導体の製造方法 |
| JP2014025953A Division JP5793588B2 (ja) | 2010-03-12 | 2014-02-13 | ハロゲン化ピコリン誘導体の製造方法 |
| JP2014025955A Division JP5695234B2 (ja) | 2010-03-12 | 2014-02-13 | テトラゾリルオキシム誘導体及びテトラゾリルオキシム誘導体の製造方法 |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JPWO2011111831A1 JPWO2011111831A1 (ja) | 2013-06-27 |
| JP5627038B2 true JP5627038B2 (ja) | 2014-11-19 |
Family
ID=44563629
Family Applications (5)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2012504543A Active JP5627038B2 (ja) | 2010-03-12 | 2011-03-11 | ピリジン環含有化合物 |
| JP2014025954A Active JP5793589B2 (ja) | 2010-03-12 | 2014-02-13 | 臭化ピコリン誘導体の製造方法 |
| JP2014025952A Active JP5695233B2 (ja) | 2010-03-12 | 2014-02-13 | テトラゾリルオキシム誘導体の製造方法 |
| JP2014025955A Active JP5695234B2 (ja) | 2010-03-12 | 2014-02-13 | テトラゾリルオキシム誘導体及びテトラゾリルオキシム誘導体の製造方法 |
| JP2014025953A Active JP5793588B2 (ja) | 2010-03-12 | 2014-02-13 | ハロゲン化ピコリン誘導体の製造方法 |
Family Applications After (4)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2014025954A Active JP5793589B2 (ja) | 2010-03-12 | 2014-02-13 | 臭化ピコリン誘導体の製造方法 |
| JP2014025952A Active JP5695233B2 (ja) | 2010-03-12 | 2014-02-13 | テトラゾリルオキシム誘導体の製造方法 |
| JP2014025955A Active JP5695234B2 (ja) | 2010-03-12 | 2014-02-13 | テトラゾリルオキシム誘導体及びテトラゾリルオキシム誘導体の製造方法 |
| JP2014025953A Active JP5793588B2 (ja) | 2010-03-12 | 2014-02-13 | ハロゲン化ピコリン誘導体の製造方法 |
Country Status (10)
| Country | Link |
|---|---|
| US (5) | US8841458B2 (enExample) |
| EP (4) | EP2546236A4 (enExample) |
| JP (5) | JP5627038B2 (enExample) |
| KR (1) | KR101409137B1 (enExample) |
| CN (5) | CN104072408B (enExample) |
| AU (1) | AU2011225122B8 (enExample) |
| BR (4) | BR122017023123B1 (enExample) |
| IL (3) | IL221847A (enExample) |
| RU (1) | RU2512344C1 (enExample) |
| WO (1) | WO2011111831A1 (enExample) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| KR101633575B1 (ko) | 2012-03-13 | 2016-06-24 | 닛뽕소다 가부시키가이샤 | 화합물, 화합물의 제조 방법, 및 화합물의 정제 방법 |
| CN108935454A (zh) * | 2012-07-19 | 2018-12-07 | 日本曹达株式会社 | 水分散粒剂 |
| US20180265481A1 (en) | 2015-03-10 | 2018-09-20 | Lonza Ltd | Method for preparation of certain 1,5 disubstituted tetrazoles |
| EP3112344A1 (en) | 2015-06-30 | 2017-01-04 | Lonza Ltd | Method for preparation of certain thioacetamides |
| CN110452220B (zh) * | 2018-04-26 | 2020-08-14 | 东莞市东阳光农药研发有限公司 | 肟衍生物及其在农业中的应用 |
| CN113825747B (zh) * | 2019-05-13 | 2025-04-25 | 大金工业株式会社 | 氟代内酯及其制造方法 |
| EP3782985A1 (en) | 2019-08-19 | 2021-02-24 | BASF Agrochemical Products B.V. | Process for manufacturing 5-methoxymethylpyridine-2,3-dicarboxylic acid derivatives |
Citations (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2279346A (en) * | 1993-07-01 | 1995-01-04 | Glaxo Group Ltd | Benzofuran intermediates |
| US5872136A (en) * | 1996-04-03 | 1999-02-16 | Merck & Co., Inc. | Arylheteroaryl inhibitors of farnesyl-protein transferase |
| WO2008106692A1 (en) * | 2007-03-01 | 2008-09-04 | Novartis Vaccines And Diagnostics, Inc. | Pim kinase inhibitors and methods of their use |
| WO2009014100A1 (ja) * | 2007-07-20 | 2009-01-29 | Chugai Seiyaku Kabushiki Kaisha | p27蛋白質誘導剤 |
| JP2009040711A (ja) * | 2007-08-08 | 2009-02-26 | Kyorin Pharmaceut Co Ltd | カルボスティリル誘導体及びそれらを有効成分とするpde阻害剤 |
| US20090098189A1 (en) * | 2007-09-05 | 2009-04-16 | Bernd Buchmann | Azaindoles as inhibitors of soluble adenylate cyclase |
Family Cites Families (31)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JPS5643268A (en) | 1979-09-17 | 1981-04-21 | Seitetsu Kagaku Co Ltd | 6-chloro-2-(chloromethyl)pyridine and its preparation |
| IL96436A0 (en) | 1989-11-28 | 1991-08-16 | Ishihara Sangyo Kaisha | Pyridylcarbamates,their preparation and biocidal compositions containing them |
| DE4322054A1 (de) | 1993-07-02 | 1995-01-12 | Bayer Ag | Verfahren zur Herstellung von Chlormethylpyridinen |
| DE4446338A1 (de) | 1994-12-23 | 1996-06-27 | Bayer Ag | Verfahren zur Herstellung von Chlormethylpyridinen |
| JPH09268178A (ja) | 1996-04-01 | 1997-10-14 | Shiratori Seiyaku Kk | 光学活性な4,5−ジフェニル−2−イミダゾリジノン誘導体 |
| DE19815946A1 (de) | 1998-04-09 | 1999-10-14 | Basf Ag | N-Vinyleinheiten enthaltende polymere Gerbstoffe |
| JP4330313B2 (ja) | 2001-08-20 | 2009-09-16 | 日本曹達株式会社 | テトラゾイルオキシム誘導体及びこれを有効成分とする農薬 |
| BRPI0212034B1 (pt) * | 2001-08-20 | 2018-01-30 | Nippon Soda Co., Ltd. | Derivado de tetrazoiloxima, produto químico agrícola e agente controlador de doença de planta contendo o mesmo como ingrediente ativo |
| US6784294B2 (en) * | 2002-03-12 | 2004-08-31 | Wyeth | Preparation of N1-(2′-pyridyl)-1,2-propanediamine sulfamic acid and its use in the synthesis of biologically active piperazines |
| JP2004131392A (ja) | 2002-10-08 | 2004-04-30 | Sumitomo Chem Co Ltd | テトラゾール化合物およびその用途 |
| JP2004131416A (ja) | 2002-10-10 | 2004-04-30 | Sumitomo Chem Co Ltd | テトラゾール化合物およびその植物病害防除用途 |
| TWI346108B (en) * | 2004-08-23 | 2011-08-01 | Bristol Myers Squibb Co | A method for preparing irbesartan and intermediates thereof |
| AR059339A1 (es) * | 2006-02-09 | 2008-03-26 | Chugai Pharmaceutical Co Ltd | Derivados de la cumarina para trastornos proliferativos de celulas, composicion farmaceutica y agente terapeutico que los contiene |
| WO2007141473A1 (en) | 2006-06-09 | 2007-12-13 | Astrazeneca Ab | N-(benzoyl)-o- [2- (pyridin- 2 -ylamino) ethyl] -l-tyrosine derivatives and related compounds as a5b1 antagonists for the treatment of solid tumors |
| CA2653698A1 (en) | 2006-07-13 | 2008-01-17 | Bayer Cropscience Sa | Fungicide hydroximoyl-tetrazole derivatives |
| US8084613B2 (en) | 2007-05-14 | 2011-12-27 | Nippon Soda Co., Ltd. | Tetrazoyloxime derivative and plant disease control agent |
| JPWO2008156102A1 (ja) | 2007-06-19 | 2010-08-26 | 杏林製薬株式会社 | ピラゾロン誘導体及びそれらを有効成分とするpde阻害剤 |
| EP2168959A1 (en) * | 2007-06-19 | 2010-03-31 | Kyorin Pharmaceutical Co., Ltd. | Pyridazinone derivative and pde inhibitor containing the same as active ingredient |
| EP2669282A1 (en) * | 2007-08-08 | 2013-12-04 | Nippon Soda Co., Ltd. | Tetrazoyloxime derivative and plant disease control agent |
| US8084477B2 (en) | 2007-10-31 | 2011-12-27 | Bristol-Myers Squibb Company | Alpha-(N-sulfonamido)acetamide compound as an inhibitor of beta amyloid peptide production |
| US8648097B2 (en) | 2008-03-12 | 2014-02-11 | Ube Industries, Ltd. | Pyridylaminoacetic acid compound |
| MX2010010135A (es) * | 2008-03-19 | 2010-10-25 | Bayer Cropscience Ag | Derivados de hidroximoil-tetrazol fungicidas. |
| JPWO2009130900A1 (ja) * | 2008-04-24 | 2011-08-11 | 日本曹達株式会社 | オキシム誘導体、中間体化合物および植物病害防除剤 |
| CA2728469A1 (en) | 2008-07-04 | 2010-01-07 | Bayer Cropscience Ag | Fungicide hydroximoyl-tetrazole derivatives |
| EP2318415B1 (en) | 2008-07-15 | 2013-02-20 | Sanofi | Oxazolopyrimidines as edg-1 receptor agonists |
| JP4926141B2 (ja) | 2008-08-27 | 2012-05-09 | 京セラ株式会社 | 誘電体アンテナ及びこれを用いた通信機器装置 |
| CN101362730B (zh) * | 2008-09-25 | 2011-09-21 | 北京赛科药业有限责任公司 | 一种制备沙坦侧链化合物的方法 |
| JP2010115703A (ja) | 2008-11-13 | 2010-05-27 | Shuichi Matsunaga | 閉塞鍛造装置 |
| JP2010127207A (ja) | 2008-11-28 | 2010-06-10 | Toyota Motor Corp | 過給器用エアホース膨張防止装置 |
| AU2011236155B2 (en) | 2010-04-06 | 2014-01-16 | Nippon Soda Co., Ltd. | Nitrogen-containing heterocyclic compound and method for producing same |
| JP2010248273A (ja) * | 2010-08-10 | 2010-11-04 | Nippon Soda Co Ltd | オキシム化合物またはその塩、ならびに殺菌剤 |
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2011
- 2011-03-11 CN CN201410283380.4A patent/CN104072408B/zh active Active
- 2011-03-11 US US13/583,733 patent/US8841458B2/en active Active
- 2011-03-11 JP JP2012504543A patent/JP5627038B2/ja active Active
- 2011-03-11 WO PCT/JP2011/055809 patent/WO2011111831A1/ja not_active Ceased
- 2011-03-11 CN CN201180012762.8A patent/CN102791691B/zh active Active
- 2011-03-11 KR KR1020127023288A patent/KR101409137B1/ko active Active
- 2011-03-11 EP EP11753489.1A patent/EP2546236A4/en not_active Withdrawn
- 2011-03-11 CN CN201410283225.2A patent/CN104072483B/zh active Active
- 2011-03-11 AU AU2011225122A patent/AU2011225122B8/en active Active
- 2011-03-11 EP EP14000070.4A patent/EP2719687B1/en active Active
- 2011-03-11 EP EP14000069.6A patent/EP2719686B1/en active Active
- 2011-03-11 BR BR122017023123-5A patent/BR122017023123B1/pt active IP Right Grant
- 2011-03-11 RU RU2012138410/04A patent/RU2512344C1/ru active
- 2011-03-11 BR BR122017023130-8A patent/BR122017023130B1/pt active IP Right Grant
- 2011-03-11 EP EP14000071.2A patent/EP2719688B1/en active Active
- 2011-03-11 CN CN201410283542.4A patent/CN104130184B/zh active Active
- 2011-03-11 CN CN201410283563.6A patent/CN104109150B/zh active Active
- 2011-03-11 BR BR122017023128-6A patent/BR122017023128B1/pt active IP Right Grant
- 2011-03-11 BR BR112012022823-4A patent/BR112012022823B1/pt active IP Right Grant
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2012
- 2012-09-09 IL IL221847A patent/IL221847A/en active IP Right Grant
-
2013
- 2013-12-17 IL IL229967A patent/IL229967A/en active IP Right Grant
- 2013-12-17 IL IL229968A patent/IL229968A/en active IP Right Grant
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2014
- 2014-02-05 US US14/173,323 patent/US9018385B2/en active Active
- 2014-02-05 US US14/173,352 patent/US9000178B2/en active Active
- 2014-02-05 US US14/173,330 patent/US9012653B2/en active Active
- 2014-02-05 US US14/173,338 patent/US8962848B2/en active Active
- 2014-02-13 JP JP2014025954A patent/JP5793589B2/ja active Active
- 2014-02-13 JP JP2014025952A patent/JP5695233B2/ja active Active
- 2014-02-13 JP JP2014025955A patent/JP5695234B2/ja active Active
- 2014-02-13 JP JP2014025953A patent/JP5793588B2/ja active Active
Patent Citations (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB2279346A (en) * | 1993-07-01 | 1995-01-04 | Glaxo Group Ltd | Benzofuran intermediates |
| US5872136A (en) * | 1996-04-03 | 1999-02-16 | Merck & Co., Inc. | Arylheteroaryl inhibitors of farnesyl-protein transferase |
| WO2008106692A1 (en) * | 2007-03-01 | 2008-09-04 | Novartis Vaccines And Diagnostics, Inc. | Pim kinase inhibitors and methods of their use |
| WO2009014100A1 (ja) * | 2007-07-20 | 2009-01-29 | Chugai Seiyaku Kabushiki Kaisha | p27蛋白質誘導剤 |
| JP2009040711A (ja) * | 2007-08-08 | 2009-02-26 | Kyorin Pharmaceut Co Ltd | カルボスティリル誘導体及びそれらを有効成分とするpde阻害剤 |
| US20090098189A1 (en) * | 2007-09-05 | 2009-04-16 | Bernd Buchmann | Azaindoles as inhibitors of soluble adenylate cyclase |
Non-Patent Citations (1)
| Title |
|---|
| JPN6013062387; 新実験化学講座14 有機化合物の合成と反応V , 1978, pp.2555-2569, 丸善株式会社 * |
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