JP5475441B2 - 置換されたアミノピラゾロピリン類及びそれらの塩類、それらの調製及びそれらを含んで成る医薬組成物類 - Google Patents
置換されたアミノピラゾロピリン類及びそれらの塩類、それらの調製及びそれらを含んで成る医薬組成物類 Download PDFInfo
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- JP5475441B2 JP5475441B2 JP2009514714A JP2009514714A JP5475441B2 JP 5475441 B2 JP5475441 B2 JP 5475441B2 JP 2009514714 A JP2009514714 A JP 2009514714A JP 2009514714 A JP2009514714 A JP 2009514714A JP 5475441 B2 JP5475441 B2 JP 5475441B2
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- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
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Landscapes
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- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
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- Pharmacology & Pharmacy (AREA)
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- Urology & Nephrology (AREA)
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- Vascular Medicine (AREA)
- Ophthalmology & Optometry (AREA)
- Neurosurgery (AREA)
- Transplantation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP06090108.9 | 2006-06-13 | ||
| EP06090108A EP1867647A1 (en) | 2006-06-13 | 2006-06-13 | Substituted aminopyrazolopyridines and salts thereof, their preparations and pharmaceutical compositions comprising them. |
| EP07090024 | 2007-02-22 | ||
| EP07090024.6 | 2007-02-22 | ||
| PCT/EP2007/005430 WO2007144202A1 (en) | 2006-06-13 | 2007-06-12 | Substituted aminopyrazolopyridines and salts thereof, their preparations and pharmaceutical compositions comprising them |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2009539912A JP2009539912A (ja) | 2009-11-19 |
| JP2009539912A5 JP2009539912A5 (enExample) | 2013-05-16 |
| JP5475441B2 true JP5475441B2 (ja) | 2014-04-16 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2009514714A Expired - Fee Related JP5475441B2 (ja) | 2006-06-13 | 2007-06-12 | 置換されたアミノピラゾロピリン類及びそれらの塩類、それらの調製及びそれらを含んで成る医薬組成物類 |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US7825114B2 (enExample) |
| EP (1) | EP2032572B1 (enExample) |
| JP (1) | JP5475441B2 (enExample) |
| AR (1) | AR061345A1 (enExample) |
| CA (1) | CA2654987C (enExample) |
| CL (1) | CL2007001710A1 (enExample) |
| ES (1) | ES2467017T3 (enExample) |
| TW (1) | TW200815437A (enExample) |
| UY (1) | UY30410A1 (enExample) |
| WO (1) | WO2007144202A1 (enExample) |
Families Citing this family (17)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PE20061119A1 (es) * | 2005-01-19 | 2006-11-27 | Aventis Pharma Sa | PIRAZOLO PIRIDINAS SUSTITUIDAS COMO INHIBIDORES DE CINASAS FAK, KDR Y Tie |
| EP2452937A1 (en) * | 2007-04-30 | 2012-05-16 | Abbott Laboratories | Inhibitors of diacylglycerol o-acyltransferase type 1 enzyme |
| EP2307456B1 (en) | 2008-06-27 | 2014-10-15 | Amgen Inc. | Ang-2 inhibition to treat multiple sclerosis |
| JP5689069B2 (ja) | 2008-11-20 | 2015-03-25 | ジェネンテック， インコーポレイテッド | ピラゾロピリジンｐｉ３ｋ阻害剤化合物及び使用方法 |
| EP2464647B1 (en) | 2009-08-11 | 2016-09-21 | Bristol-Myers Squibb Company | Azaindazoles as btk kinase modulators and use thereof |
| CN103214479A (zh) * | 2012-01-18 | 2013-07-24 | 武汉东宇生物医药科技有限公司 | 吡唑类萘脲类酪氨酸激酶抑制剂及其应用 |
| CN103923078A (zh) * | 2013-01-15 | 2014-07-16 | 华东理工大学 | 3,4-二取代(1H-吡唑[3,4-b]吡啶)类化合物及其用途 |
| CN103524421B (zh) * | 2013-09-29 | 2015-04-01 | 镇江蓝德特药业科技有限公司 | 新型萘脲类衍生物及其医疗应用 |
| JOP20190024A1 (ar) | 2016-08-26 | 2019-02-19 | Gilead Sciences Inc | مركبات بيروليزين بها استبدال واستخداماتها |
| CA3072362A1 (en) | 2017-10-06 | 2019-04-11 | Forma Therapeutics, Inc. | Inhibiting ubiquitin specific peptidase 30 |
| JP7050165B2 (ja) | 2018-02-26 | 2022-04-07 | ギリアード サイエンシーズ， インコーポレイテッド | Ｈｂｖ複製阻害剤としての置換ピロリジン化合物 |
| SG11202011299PA (en) | 2018-05-17 | 2020-12-30 | Forma Therapeutics Inc | Fused bicyclic compounds useful as ubiquitin-specific peptidase 30 inhibitors |
| MY209034A (en) | 2018-10-05 | 2025-06-17 | Forma Therapeutics Inc | Fused pyrrolines which act as ubiquitin-specific protease 30 (usp30) inhibitors |
| TW202330519A (zh) * | 2021-09-29 | 2023-08-01 | 香港商德琪研發有限公司 | 作為ｔａｍ抑制劑的吡唑并吡啶化合物 |
| KR20240148322A (ko) * | 2021-12-22 | 2024-10-11 | 아낙시스 파마 피티와이 엘티디 | 이작용성 아릴설폰아미드 화합물 |
| AU2022421952A1 (en) * | 2021-12-22 | 2024-07-04 | Anaxis Pharma Pty Ltd | Arylsulphonamide compounds |
| WO2023155886A1 (en) * | 2022-02-17 | 2023-08-24 | Shanghai Antengene Corporation Limited | Pyrazolopyridine compounds as tam inhibitors |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU7491400A (en) * | 1999-09-17 | 2001-04-17 | Abbott Gmbh & Co. Kg | Kinase inhibitors as therapeutic agents |
| JP4810427B2 (ja) | 2003-05-22 | 2011-11-09 | アボット・ラボラトリーズ | インダゾール、ベンズイソオキサゾールおよびベンズイソチアゾールキナーゼ阻害剤 |
| MX2007005120A (es) * | 2004-10-29 | 2007-07-16 | Abbott Lab | Nuevos inhibidores de cinasa. |
-
2007
- 2007-06-11 TW TW096120982A patent/TW200815437A/zh unknown
- 2007-06-12 WO PCT/EP2007/005430 patent/WO2007144202A1/en not_active Ceased
- 2007-06-12 JP JP2009514714A patent/JP5475441B2/ja not_active Expired - Fee Related
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- 2007-06-12 CL CL2007001710A patent/CL2007001710A1/es unknown
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- 2007-06-12 US US11/761,621 patent/US7825114B2/en not_active Expired - Fee Related
- 2007-06-12 UY UY30410A patent/UY30410A1/es not_active Application Discontinuation
- 2007-06-12 AR ARP070102551A patent/AR061345A1/es unknown
- 2007-06-12 EP EP07764751.9A patent/EP2032572B1/en not_active Not-in-force
Also Published As
| Publication number | Publication date |
|---|---|
| AR061345A1 (es) | 2008-08-20 |
| ES2467017T3 (es) | 2014-06-11 |
| UY30410A1 (es) | 2008-01-31 |
| US7825114B2 (en) | 2010-11-02 |
| CA2654987A1 (en) | 2007-12-21 |
| EP2032572B1 (en) | 2014-03-12 |
| TW200815437A (en) | 2008-04-01 |
| EP2032572A1 (en) | 2009-03-11 |
| CL2007001710A1 (es) | 2008-01-04 |
| JP2009539912A (ja) | 2009-11-19 |
| US20090018129A1 (en) | 2009-01-15 |
| CA2654987C (en) | 2014-08-05 |
| WO2007144202A1 (en) | 2007-12-21 |
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