JP5328349B2 - ベータ−ラクタミルフェニルアラニン、システイン、およびセリン・バソプレッシン拮抗剤 - Google Patents

ベータ−ラクタミルフェニルアラニン、システイン、およびセリン・バソプレッシン拮抗剤 Download PDF

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JP5328349B2
JP5328349B2 JP2008522861A JP2008522861A JP5328349B2 JP 5328349 B2 JP5328349 B2 JP 5328349B2 JP 2008522861 A JP2008522861 A JP 2008522861A JP 2008522861 A JP2008522861 A JP 2008522861A JP 5328349 B2 JP5328349 B2 JP 5328349B2
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JP2009502788A (ja
JP2009502788A5 (enExample
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コッペル，ゲリー，エー．
ミラー，マーヴィン，ジェイ．
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Azevan Pharmaceuticals Inc
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Azevan Pharmaceuticals Inc
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    • C07—ORGANIC CHEMISTRY
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    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Neurosurgery (AREA)
  • Pulmonology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Dermatology (AREA)
  • Diabetes (AREA)
  • Psychiatry (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Addiction (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Anesthesiology (AREA)
  • Endocrinology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Emergency Medicine (AREA)
  • Vascular Medicine (AREA)
  • Obesity (AREA)
JP2008522861A 2005-07-19 2006-07-18 ベータ−ラクタミルフェニルアラニン、システイン、およびセリン・バソプレッシン拮抗剤 Expired - Fee Related JP5328349B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US70067305P 2005-07-19 2005-07-19
US60/700,673 2005-07-19
PCT/US2006/027703 WO2007011878A2 (en) 2005-07-19 2006-07-18 Beta-lactamyl phenylalanine, cysteine, and serine vasopressin antagonists

Related Child Applications (1)

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JP2013044654A Division JP2013151520A (ja) 2005-07-19 2013-03-06 ベータ−ラクタミルフェニルアラニン、システイン、およびセリン・バソプレッシン拮抗剤

Publications (3)

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JP2009502788A JP2009502788A (ja) 2009-01-29
JP2009502788A5 JP2009502788A5 (enExample) 2009-10-08
JP5328349B2 true JP5328349B2 (ja) 2013-10-30

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JP2008522861A Expired - Fee Related JP5328349B2 (ja) 2005-07-19 2006-07-18 ベータ−ラクタミルフェニルアラニン、システイン、およびセリン・バソプレッシン拮抗剤
JP2013044654A Pending JP2013151520A (ja) 2005-07-19 2013-03-06 ベータ−ラクタミルフェニルアラニン、システイン、およびセリン・バソプレッシン拮抗剤

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US (2) US8048874B2 (enExample)
EP (1) EP1910346B1 (enExample)
JP (2) JP5328349B2 (enExample)
KR (2) KR101523776B1 (enExample)
CN (1) CN101268068B (enExample)
AU (1) AU2006270039B2 (enExample)
BR (1) BRPI0613664B1 (enExample)
CA (1) CA2615813C (enExample)
DK (1) DK1910346T3 (enExample)
ES (1) ES2726942T3 (enExample)
PL (1) PL1910346T3 (enExample)
RU (1) RU2466991C2 (enExample)
SI (1) SI1910346T1 (enExample)
TR (1) TR201907381T4 (enExample)
WO (1) WO2007011878A2 (enExample)

Families Citing this family (15)

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Publication number Priority date Publication date Assignee Title
AU2002342045C1 (en) * 2001-10-12 2009-07-30 Azevan Pharmaceuticals, Inc. Beta-lactamyl vasopressin Vla antagonists
EP1638549A4 (en) 2003-03-10 2011-06-15 Optimer Pharmaceuticals Inc NEW ANTIBACTERIAL AGENTS
CA2601709C (en) 2005-03-22 2017-02-14 Azevan Pharmaceuticals, Inc. Beta-lactamylalkanoic acids
AU2006270039B2 (en) * 2005-07-19 2013-07-04 Azevan Pharmaceuticals, Inc. Beta-lactamyl phenylalanine, cysteine, and serine vasopressin antagonists
US20100016274A1 (en) * 2006-09-14 2010-01-21 Koppel Gary A Beta-lactam cannabinoid receptor modulators
US9453042B2 (en) 2007-10-25 2016-09-27 Cempra Pharmaceuticals, Inc. Process for the preparation of macrolide antibacterial agents
HRP20160222T1 (hr) 2008-10-24 2016-04-08 Cempra Pharmaceuticals, Inc. Biozaštite uporabom makrolida koji sadrže triazol
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
WO2012003436A1 (en) * 2010-07-01 2012-01-05 Azevan Pharmaceuticals, Inc. Methods for treating post traumatic stress disorder
US9815863B2 (en) 2010-09-10 2017-11-14 Cempra Pharmaceuticals, Inc. Hydrogen bond forming fluoro ketolides for treating diseases
IN2014DN08939A (enExample) 2012-03-27 2015-05-22 Cempra Pharmaceuticals Inc
CA2905975A1 (en) 2013-03-14 2014-09-25 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor
EP2968384A4 (en) 2013-03-15 2017-02-15 Cempra Pharmaceuticals, Inc. Convergent processes for preparing macrolide antibacterial agents
CA2944211C (en) 2014-03-28 2022-10-04 Azevan Pharmaceuticals, Inc. Compositions and methods for treating neurodegenerative diseases
EP3681871A4 (en) 2017-09-15 2021-05-26 Azevan Pharmaceuticals, Inc. COMPOSITIONS AND METHODS FOR THE TREATMENT OF A BRAIN DAMAGE

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JPS6033439B2 (ja) * 1980-03-07 1985-08-02 財団法人相模中央化学研究所 ジペプチドの製造方法
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US8048874B2 (en) 2011-11-01
US20080280870A1 (en) 2008-11-13
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BRPI0613664A8 (pt) 2018-06-19
KR20140089430A (ko) 2014-07-14
US8426400B2 (en) 2013-04-23
RU2008106251A (ru) 2009-08-27
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CA2615813C (en) 2015-12-15
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US20120220765A1 (en) 2012-08-30
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PL1910346T3 (pl) 2019-09-30
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