BRPI0613664B1 - Compostos antagonistas de beta-lactamil fenilalanina, cisteína e serina vasopressina, composição farmacêutica que compreende ditos compostos e usos terapêuticos dos mesmos - Google Patents

Compostos antagonistas de beta-lactamil fenilalanina, cisteína e serina vasopressina, composição farmacêutica que compreende ditos compostos e usos terapêuticos dos mesmos Download PDF

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Publication number
BRPI0613664B1
BRPI0613664B1 BRPI0613664-8A BRPI0613664A BRPI0613664B1 BR PI0613664 B1 BRPI0613664 B1 BR PI0613664B1 BR PI0613664 A BRPI0613664 A BR PI0613664A BR PI0613664 B1 BRPI0613664 B1 BR PI0613664B1
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Prior art keywords
alkyl
optionally substituted
group
substituted aryl
compounds
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BRPI0613664-8A
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English (en)
Portuguese (pt)
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Gary A. Koppel
Marvin J. Miller
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Azevan Pharmaceuticals, Inc
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Publication of BRPI0613664A2 publication Critical patent/BRPI0613664A2/pt
Publication of BRPI0613664A8 publication Critical patent/BRPI0613664A8/pt
Publication of BRPI0613664B1 publication Critical patent/BRPI0613664B1/pt

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    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
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BRPI0613664-8A 2005-07-19 2006-07-18 Compostos antagonistas de beta-lactamil fenilalanina, cisteína e serina vasopressina, composição farmacêutica que compreende ditos compostos e usos terapêuticos dos mesmos BRPI0613664B1 (pt)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US70067305P 2005-07-19 2005-07-19
US60/700.673 2005-07-19
PCT/US2006/027703 WO2007011878A2 (en) 2005-07-19 2006-07-18 Beta-lactamyl phenylalanine, cysteine, and serine vasopressin antagonists

Publications (3)

Publication Number Publication Date
BRPI0613664A2 BRPI0613664A2 (pt) 2011-01-25
BRPI0613664A8 BRPI0613664A8 (pt) 2018-06-19
BRPI0613664B1 true BRPI0613664B1 (pt) 2021-08-24

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BRPI0613664-8A BRPI0613664B1 (pt) 2005-07-19 2006-07-18 Compostos antagonistas de beta-lactamil fenilalanina, cisteína e serina vasopressina, composição farmacêutica que compreende ditos compostos e usos terapêuticos dos mesmos

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Country Link
US (2) US8048874B2 (enExample)
EP (1) EP1910346B1 (enExample)
JP (2) JP5328349B2 (enExample)
KR (2) KR101523776B1 (enExample)
CN (1) CN101268068B (enExample)
AU (1) AU2006270039B2 (enExample)
BR (1) BRPI0613664B1 (enExample)
CA (1) CA2615813C (enExample)
DK (1) DK1910346T3 (enExample)
ES (1) ES2726942T3 (enExample)
PL (1) PL1910346T3 (enExample)
RU (1) RU2466991C2 (enExample)
SI (1) SI1910346T1 (enExample)
TR (1) TR201907381T4 (enExample)
WO (1) WO2007011878A2 (enExample)

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CA2601709C (en) 2005-03-22 2017-02-14 Azevan Pharmaceuticals, Inc. Beta-lactamylalkanoic acids
AU2006270039B2 (en) * 2005-07-19 2013-07-04 Azevan Pharmaceuticals, Inc. Beta-lactamyl phenylalanine, cysteine, and serine vasopressin antagonists
US20100016274A1 (en) * 2006-09-14 2010-01-21 Koppel Gary A Beta-lactam cannabinoid receptor modulators
US9453042B2 (en) 2007-10-25 2016-09-27 Cempra Pharmaceuticals, Inc. Process for the preparation of macrolide antibacterial agents
HRP20160222T1 (hr) 2008-10-24 2016-04-08 Cempra Pharmaceuticals, Inc. Biozaštite uporabom makrolida koji sadrže triazol
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
WO2012003436A1 (en) * 2010-07-01 2012-01-05 Azevan Pharmaceuticals, Inc. Methods for treating post traumatic stress disorder
US9815863B2 (en) 2010-09-10 2017-11-14 Cempra Pharmaceuticals, Inc. Hydrogen bond forming fluoro ketolides for treating diseases
IN2014DN08939A (enExample) 2012-03-27 2015-05-22 Cempra Pharmaceuticals Inc
CA2905975A1 (en) 2013-03-14 2014-09-25 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor
EP2968384A4 (en) 2013-03-15 2017-02-15 Cempra Pharmaceuticals, Inc. Convergent processes for preparing macrolide antibacterial agents
CA2944211C (en) 2014-03-28 2022-10-04 Azevan Pharmaceuticals, Inc. Compositions and methods for treating neurodegenerative diseases
EP3681871A4 (en) 2017-09-15 2021-05-26 Azevan Pharmaceuticals, Inc. COMPOSITIONS AND METHODS FOR THE TREATMENT OF A BRAIN DAMAGE

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WO2007011878A2 (en) 2007-01-25
BRPI0613664A2 (pt) 2011-01-25
US8048874B2 (en) 2011-11-01
US20080280870A1 (en) 2008-11-13
AU2006270039A1 (en) 2007-01-25
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BRPI0613664A8 (pt) 2018-06-19
KR20140089430A (ko) 2014-07-14
US8426400B2 (en) 2013-04-23
RU2008106251A (ru) 2009-08-27
DK1910346T3 (da) 2019-05-27
CN101268068B (zh) 2015-12-02
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EP1910346B1 (en) 2019-02-27
CA2615813C (en) 2015-12-15
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US20120220765A1 (en) 2012-08-30
SI1910346T1 (sl) 2019-08-30
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PL1910346T3 (pl) 2019-09-30
JP5328349B2 (ja) 2013-10-30
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