PL1910346T3 - Beta-laktamowy antagonista wazopresyny fenyloalaniny, cysteiny i seryny - Google Patents

Beta-laktamowy antagonista wazopresyny fenyloalaniny, cysteiny i seryny

Info

Publication number
PL1910346T3
PL1910346T3 PL06787593T PL06787593T PL1910346T3 PL 1910346 T3 PL1910346 T3 PL 1910346T3 PL 06787593 T PL06787593 T PL 06787593T PL 06787593 T PL06787593 T PL 06787593T PL 1910346 T3 PL1910346 T3 PL 1910346T3
Authority
PL
Poland
Prior art keywords
lactamyl
phenylalanine
cysteine
serine
beta
Prior art date
Application number
PL06787593T
Other languages
English (en)
Inventor
Gary A. Koppel
Marvin J. Miller
Original Assignee
Azevan Pharmaceuticals, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Azevan Pharmaceuticals, Inc. filed Critical Azevan Pharmaceuticals, Inc.
Publication of PL1910346T3 publication Critical patent/PL1910346T3/pl

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A61K31/422—Oxazoles not condensed and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61P1/08—Drugs for disorders of the alimentary tract or the digestive system for nausea, cinetosis or vertigo; Antiemetics
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond

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  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pulmonology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Urology & Nephrology (AREA)
  • Diabetes (AREA)
  • Psychiatry (AREA)
  • Immunology (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Hematology (AREA)
  • Hospice & Palliative Care (AREA)
  • Otolaryngology (AREA)
  • Addiction (AREA)
  • Ophthalmology & Optometry (AREA)
  • Obesity (AREA)
  • Vascular Medicine (AREA)
  • Endocrinology (AREA)
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PL06787593T 2005-07-19 2006-07-18 Beta-laktamowy antagonista wazopresyny fenyloalaniny, cysteiny i seryny PL1910346T3 (pl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US70067305P 2005-07-19 2005-07-19
EP06787593.0A EP1910346B1 (en) 2005-07-19 2006-07-18 Beta-lactamyl phenylalanine, cysteine, and serine vasopressin antagonist
PCT/US2006/027703 WO2007011878A2 (en) 2005-07-19 2006-07-18 Beta-lactamyl phenylalanine, cysteine, and serine vasopressin antagonists

Publications (1)

Publication Number Publication Date
PL1910346T3 true PL1910346T3 (pl) 2019-09-30

Family

ID=37529732

Family Applications (1)

Application Number Title Priority Date Filing Date
PL06787593T PL1910346T3 (pl) 2005-07-19 2006-07-18 Beta-laktamowy antagonista wazopresyny fenyloalaniny, cysteiny i seryny

Country Status (15)

Country Link
US (2) US8048874B2 (pl)
EP (1) EP1910346B1 (pl)
JP (2) JP5328349B2 (pl)
KR (2) KR101521405B1 (pl)
CN (1) CN101268068B (pl)
AU (1) AU2006270039B2 (pl)
BR (1) BRPI0613664B1 (pl)
CA (1) CA2615813C (pl)
DK (1) DK1910346T3 (pl)
ES (1) ES2726942T3 (pl)
PL (1) PL1910346T3 (pl)
RU (1) RU2466991C2 (pl)
SI (1) SI1910346T1 (pl)
TR (1) TR201907381T4 (pl)
WO (1) WO2007011878A2 (pl)

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AU2002342045C1 (en) * 2001-10-12 2009-07-30 Azevan Pharmaceuticals, Inc. Beta-lactamyl vasopressin Vla antagonists
EP3738591A3 (en) 2003-03-10 2021-03-24 Merck Sharp & Dohme Corp. Novel antibacterial agents
WO2006102283A2 (en) 2005-03-22 2006-09-28 Azevan Pharmaceuticals, Inc. Beta-lactamylalkanoic acids for treating premenstrual disorders
PL1910346T3 (pl) * 2005-07-19 2019-09-30 Azevan Pharmaceuticals, Inc. Beta-laktamowy antagonista wazopresyny fenyloalaniny, cysteiny i seryny
US20100016274A1 (en) * 2006-09-14 2010-01-21 Koppel Gary A Beta-lactam cannabinoid receptor modulators
CN101917850B (zh) 2007-10-25 2016-01-13 森普拉制药公司 大环内酯类抗菌剂的制备方法
DK2358379T3 (en) 2008-10-24 2016-03-07 Cempra Pharmaceuticals Inc BIOFORSVAR USING TRIAZOLHOLDIGE macrolides
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
RU2623209C9 (ru) 2010-07-01 2018-01-22 Азеван Фармасьютикалз, Инк. Способы лечения посттравматического стрессового расстройства
US9815863B2 (en) 2010-09-10 2017-11-14 Cempra Pharmaceuticals, Inc. Hydrogen bond forming fluoro ketolides for treating diseases
MX2014011537A (es) 2012-03-27 2015-02-10 Cempra Pharmaceuticals Inc Formulaciones parenterales para la administracion de antibioticos macrolidos.
WO2014152326A1 (en) 2013-03-14 2014-09-25 Cempra Pharmaceuticals, Inc. Methods for treating respiratory diseases and formulations therefor
BR112015023670A2 (pt) 2013-03-15 2017-07-18 Cempra Pharmaceuticals Inc processo para preparar um composto
BR112016022575A2 (pt) 2014-03-28 2017-08-15 Azevan Pharmaceuticals Inc Composições e métodos para o tratamento de doenças neurodegenerativas
MX2020002762A (es) * 2017-09-15 2020-09-17 Azevan Pharmaceuticals Inc Composiciones y métodos para tratar una lesión cerebral.

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BRPI0613664A8 (pt) 2018-06-19
AU2006270039B2 (en) 2013-07-04
US20120220765A1 (en) 2012-08-30
ES2726942T3 (es) 2019-10-10
US8426400B2 (en) 2013-04-23
EP1910346B1 (en) 2019-02-27
JP2013151520A (ja) 2013-08-08
CA2615813C (en) 2015-12-15
EP1910346A2 (en) 2008-04-16
CN101268068A (zh) 2008-09-17
RU2008106251A (ru) 2009-08-27
US20080280870A1 (en) 2008-11-13
JP2009502788A (ja) 2009-01-29
SI1910346T1 (sl) 2019-08-30
WO2007011878A3 (en) 2007-09-07
BRPI0613664A2 (pt) 2011-01-25
DK1910346T3 (da) 2019-05-27
CN101268068B (zh) 2015-12-02
WO2007011878A2 (en) 2007-01-25
CA2615813A1 (en) 2007-01-25
AU2006270039A1 (en) 2007-01-25
WO2007011878A8 (en) 2007-04-26
KR20140089430A (ko) 2014-07-14
KR20080036193A (ko) 2008-04-25
JP5328349B2 (ja) 2013-10-30
US8048874B2 (en) 2011-11-01
BRPI0613664B1 (pt) 2021-08-24
RU2466991C2 (ru) 2012-11-20
KR101523776B1 (ko) 2015-05-28
KR101521405B1 (ko) 2015-05-18

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