JP5036557B2 - 抗炎症活性デクラジノシル−マクロライド - Google Patents
抗炎症活性デクラジノシル−マクロライド Download PDFInfo
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- JP5036557B2 JP5036557B2 JP2007550875A JP2007550875A JP5036557B2 JP 5036557 B2 JP5036557 B2 JP 5036557B2 JP 2007550875 A JP2007550875 A JP 2007550875A JP 2007550875 A JP2007550875 A JP 2007550875A JP 5036557 B2 JP5036557 B2 JP 5036557B2
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/04—Drugs for skeletal disorders for non-specific disorders of the connective tissue
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/06—Antigout agents, e.g. antihyperuricemic or uricosuric agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/08—Plasma substitutes; Perfusion solutions; Dialytics or haemodialytics; Drugs for electrolytic or acid-base disorders, e.g. hypovolemic shock
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Pulmonology (AREA)
- Dermatology (AREA)
- Rheumatology (AREA)
- Physical Education & Sports Medicine (AREA)
- Genetics & Genomics (AREA)
- Biotechnology (AREA)
- Molecular Biology (AREA)
- Biochemistry (AREA)
- Pain & Pain Management (AREA)
- Vascular Medicine (AREA)
- Otolaryngology (AREA)
- Immunology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Ophthalmology & Optometry (AREA)
- Heart & Thoracic Surgery (AREA)
- Biomedical Technology (AREA)
- Cardiology (AREA)
- Urology & Nephrology (AREA)
- Hematology (AREA)
- Diabetes (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US64384005P | 2005-01-13 | 2005-01-13 | |
| US60/643,840 | 2005-01-13 | ||
| PCT/IB2006/001097 WO2006077501A2 (en) | 2005-01-13 | 2006-01-13 | Decladinosyl-macrolides with anti-inflammatory activity |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2008526946A JP2008526946A (ja) | 2008-07-24 |
| JP2008526946A5 JP2008526946A5 (https=) | 2009-02-26 |
| JP5036557B2 true JP5036557B2 (ja) | 2012-09-26 |
Family
ID=36692605
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2007550875A Expired - Fee Related JP5036557B2 (ja) | 2005-01-13 | 2006-01-13 | 抗炎症活性デクラジノシル−マクロライド |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US7910559B2 (https=) |
| EP (1) | EP1841776B1 (https=) |
| JP (1) | JP5036557B2 (https=) |
| AT (1) | ATE419261T1 (https=) |
| DE (1) | DE602006004555D1 (https=) |
| ES (1) | ES2317527T3 (https=) |
| WO (1) | WO2006077501A2 (https=) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PT1851236E (pt) | 2005-01-13 | 2010-10-25 | Glaxosmithkline Zagreb | Macrólidos com actividade anti-inflamatória |
| US20090075916A1 (en) * | 2005-11-23 | 2009-03-19 | Upadhyay Dilip J | Use of Macrolide Derivatives for Treating Acne |
| PL2056858T3 (pl) | 2006-08-11 | 2015-01-30 | Csl Ltd | Leczenie stanów chorobowych płuc |
| CN102378763A (zh) * | 2009-01-30 | 2012-03-14 | 葛兰素集团有限公司 | 消炎的大环内酯 |
| US20160031925A1 (en) * | 2013-04-10 | 2016-02-04 | Probiotic Pharmaceuticals Aps | Azithromycin antimicrobial derivatives with non-antibiotic pharmaceutical effect |
| GB201520419D0 (en) | 2015-11-19 | 2016-01-06 | Epi Endo Pharmaceuticals Ehf | Compounds |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IL99995A (en) | 1990-11-21 | 1997-11-20 | Roussel Uclaf | Erythromycin derivatives, their preparation and pharmaceutical compositions containing them |
| US5523399A (en) * | 1991-12-27 | 1996-06-04 | Taisho Pharmaceutical Co., Ltd. | 5-O-desosaminylerythronolide derivatives |
| AU3192695A (en) | 1994-08-12 | 1996-03-07 | Taisho Pharmaceutical Co., Ltd. | Interleukin-5 production inhibitor |
| WO1996004919A1 (en) | 1994-08-12 | 1996-02-22 | Taisho Pharmaceutical Co., Ltd. | Interleukin-5 production inhibitor |
| US20020115621A1 (en) | 2000-08-07 | 2002-08-22 | Wei-Gu Su | Macrolide antibiotics |
| ITMI20021726A1 (it) * | 2002-08-01 | 2004-02-02 | Zambon Spa | Macrolidi ad attivita' antiinfiammatoria. |
| ITMI20022292A1 (it) | 2002-10-29 | 2004-04-30 | Zambon Spa | 9a-azalidi ad attivita' antiinfiammatoria. |
-
2006
- 2006-01-13 DE DE602006004555T patent/DE602006004555D1/de not_active Expired - Lifetime
- 2006-01-13 ES ES06727561T patent/ES2317527T3/es not_active Expired - Lifetime
- 2006-01-13 JP JP2007550875A patent/JP5036557B2/ja not_active Expired - Fee Related
- 2006-01-13 AT AT06727561T patent/ATE419261T1/de not_active IP Right Cessation
- 2006-01-13 US US11/813,876 patent/US7910559B2/en not_active Expired - Fee Related
- 2006-01-13 WO PCT/IB2006/001097 patent/WO2006077501A2/en not_active Ceased
- 2006-01-13 EP EP06727561A patent/EP1841776B1/en not_active Expired - Lifetime
Also Published As
| Publication number | Publication date |
|---|---|
| WO2006077501A3 (en) | 2006-11-09 |
| EP1841776A2 (en) | 2007-10-10 |
| WO2006077501A2 (en) | 2006-07-27 |
| EP1841776B1 (en) | 2008-12-31 |
| US20080234211A1 (en) | 2008-09-25 |
| JP2008526946A (ja) | 2008-07-24 |
| ES2317527T3 (es) | 2009-04-16 |
| ATE419261T1 (de) | 2009-01-15 |
| DE602006004555D1 (de) | 2009-02-12 |
| US7910559B2 (en) | 2011-03-22 |
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