JP4783733B2 - バルサルタンを含む医薬組成物 - Google Patents
バルサルタンを含む医薬組成物 Download PDFInfo
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- JP4783733B2 JP4783733B2 JP2006529827A JP2006529827A JP4783733B2 JP 4783733 B2 JP4783733 B2 JP 4783733B2 JP 2006529827 A JP2006529827 A JP 2006529827A JP 2006529827 A JP2006529827 A JP 2006529827A JP 4783733 B2 JP4783733 B2 JP 4783733B2
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- valsartan
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Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D257/00—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms
- C07D257/02—Heterocyclic compounds containing rings having four nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D257/04—Five-membered rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/06—Antihyperlipidemics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Diabetes (AREA)
- Epidemiology (AREA)
- Cardiology (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Heart & Thoracic Surgery (AREA)
- Child & Adolescent Psychology (AREA)
- Emergency Medicine (AREA)
- Endocrinology (AREA)
- Hospice & Palliative Care (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US47113703P | 2003-05-16 | 2003-05-16 | |
| US60/471,137 | 2003-05-16 | ||
| PCT/EP2004/005204 WO2004101535A1 (en) | 2003-05-16 | 2004-05-14 | Pharmaceutical composition comprising valsartan |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2006528949A JP2006528949A (ja) | 2006-12-28 |
| JP2006528949A5 JP2006528949A5 (enExample) | 2007-06-28 |
| JP4783733B2 true JP4783733B2 (ja) | 2011-09-28 |
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2006529827A Expired - Fee Related JP4783733B2 (ja) | 2003-05-16 | 2004-05-14 | バルサルタンを含む医薬組成物 |
Country Status (10)
| Country | Link |
|---|---|
| US (2) | US20070054947A1 (enExample) |
| EP (1) | EP1631556A1 (enExample) |
| JP (1) | JP4783733B2 (enExample) |
| CN (1) | CN1816533A (enExample) |
| AU (2) | AU2004238546A1 (enExample) |
| BR (1) | BRPI0410374A (enExample) |
| CA (1) | CA2525665A1 (enExample) |
| MX (1) | MXPA05012299A (enExample) |
| TW (1) | TW200509909A (enExample) |
| WO (1) | WO2004101535A1 (enExample) |
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| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20080261958A1 (en) * | 2005-11-08 | 2008-10-23 | Randy Lee Webb | Combination of Organic Compounds |
| AR057882A1 (es) * | 2005-11-09 | 2007-12-26 | Novartis Ag | Compuestos de accion doble de bloqueadores del receptor de angiotensina e inhibidores de endopeptidasa neutra |
| EP2638013A4 (en) | 2010-11-12 | 2014-03-26 | Hetero Research Foundation | NEW POLYMORPHS OF CALCIUM PIVASTATIN |
| JPWO2013147137A1 (ja) * | 2012-03-30 | 2015-12-14 | 味の素株式会社 | 心不全の治療剤 |
| PL2887961T3 (pl) | 2012-08-24 | 2021-11-08 | Novartis Ag | Inhibitory nep do leczenia chorób charakteryzujących się powiększeniem lub przebudową przedsionka |
| WO2015028941A1 (en) * | 2013-08-26 | 2015-03-05 | Novartis Ag | New use |
| WO2016037552A1 (zh) * | 2014-09-09 | 2016-03-17 | 上海翰森生物医药科技有限公司 | 结晶型ARB-NEPi复合物及其制备方法和应用 |
| JP7470647B2 (ja) * | 2018-06-14 | 2024-04-18 | アストラゼネカ・ユーケイ・リミテッド | ジヒドロピリジン型カルシウムチャネル遮断薬医薬組成物を用いて血圧を低下させるための方法 |
| AU2019287551A1 (en) * | 2018-06-14 | 2021-01-28 | Astrazeneca Uk Limited | Methods for treatment of hypertension with an angiotensin II receptor blocker pharmaceutical composition |
| CN115317478B (zh) * | 2022-08-26 | 2023-05-02 | 宁波大学 | 沙库巴曲缬沙坦类物质在制备药物成瘾和复吸药物的应用 |
Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2002015933A2 (en) * | 2000-08-22 | 2002-02-28 | Novartis Ag | Combination comprising an at1-receptor antagonist and an insulin secretion enhancer or an insulin sensitiser |
| JP2002520274A (ja) * | 1998-07-10 | 2002-07-09 | ノバルティス アクチエンゲゼルシャフト | バルサルタンとカルシウムチャンネルブロッカーの抗高血圧組合わせ |
| WO2003035046A2 (en) * | 2001-10-18 | 2003-05-01 | Novartis Ag | Salts formed of an at1-receptor antagonist and a cardiovascular agent |
Family Cites Families (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6201002B1 (en) * | 1997-01-10 | 2001-03-13 | Merck & Co., Inc. | Method for reducing mortality with an angiotensin II antagonist |
| US6204281B1 (en) * | 1998-07-10 | 2001-03-20 | Novartis Ag | Method of treatment and pharmaceutical composition |
| US6596747B2 (en) * | 1998-10-29 | 2003-07-22 | Bristol-Myers Squibb Company | Compounds derived from an amine nucleus and pharmaceutical compositions comprising same |
| CA2360305A1 (en) * | 1999-02-09 | 2000-08-17 | Bristol-Myers Squibb Company | Lactam inhibitors of fxa and method |
| US6395728B2 (en) * | 1999-07-08 | 2002-05-28 | Novartis Ag | Method of treatment and pharmaceutical composition |
| US6544981B2 (en) * | 2000-06-09 | 2003-04-08 | Bristol-Myers Squibb Company | Lactam inhibitors of factor Xa and method |
| US6642252B2 (en) * | 2000-11-07 | 2003-11-04 | Bristol-Myers Squibb Company | Acid derivatives useful as serine protease inhibitors |
| WO2002053161A1 (en) * | 2000-12-29 | 2002-07-11 | Alteon, Inc. | Method for treating fibrotic diseases or other indications |
| US6395782B1 (en) * | 2001-03-02 | 2002-05-28 | Wisconsin Alumni Research Foundation | Method of increasing longevity and preventing body weight wasting in autoimmune disease by using conjugated linoleic acid |
| CA2448306A1 (en) * | 2001-05-30 | 2002-12-05 | Alteon Inc. | Method for treating fibrotic diseases or other indications |
| US6869970B2 (en) * | 2002-02-04 | 2005-03-22 | Novartis Ag | Crystalline salt forms of valsartan |
| EG24716A (en) * | 2002-05-17 | 2010-06-07 | Novartis Ag | Combination of organic compounds |
-
2004
- 2004-05-14 TW TW093113753A patent/TW200509909A/zh unknown
- 2004-05-14 CN CNA2004800186113A patent/CN1816533A/zh active Pending
- 2004-05-14 WO PCT/EP2004/005204 patent/WO2004101535A1/en not_active Ceased
- 2004-05-14 AU AU2004238546A patent/AU2004238546A1/en not_active Abandoned
- 2004-05-14 MX MXPA05012299A patent/MXPA05012299A/es unknown
- 2004-05-14 EP EP04732990A patent/EP1631556A1/en not_active Withdrawn
- 2004-05-14 JP JP2006529827A patent/JP4783733B2/ja not_active Expired - Fee Related
- 2004-05-14 US US10/556,260 patent/US20070054947A1/en not_active Abandoned
- 2004-05-14 CA CA002525665A patent/CA2525665A1/en not_active Abandoned
- 2004-05-14 BR BRPI0410374-2A patent/BRPI0410374A/pt not_active IP Right Cessation
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2008
- 2008-11-20 AU AU2008246267A patent/AU2008246267B2/en not_active Ceased
- 2008-12-22 US US12/341,669 patent/US20090105322A1/en not_active Abandoned
Patent Citations (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2002520274A (ja) * | 1998-07-10 | 2002-07-09 | ノバルティス アクチエンゲゼルシャフト | バルサルタンとカルシウムチャンネルブロッカーの抗高血圧組合わせ |
| WO2002015933A2 (en) * | 2000-08-22 | 2002-02-28 | Novartis Ag | Combination comprising an at1-receptor antagonist and an insulin secretion enhancer or an insulin sensitiser |
| WO2003035046A2 (en) * | 2001-10-18 | 2003-05-01 | Novartis Ag | Salts formed of an at1-receptor antagonist and a cardiovascular agent |
Also Published As
| Publication number | Publication date |
|---|---|
| CA2525665A1 (en) | 2004-11-25 |
| AU2008246267A1 (en) | 2008-12-11 |
| BRPI0410374A (pt) | 2006-06-13 |
| AU2008246267B2 (en) | 2011-02-17 |
| AU2004238546A1 (en) | 2004-11-25 |
| US20070054947A1 (en) | 2007-03-08 |
| EP1631556A1 (en) | 2006-03-08 |
| JP2006528949A (ja) | 2006-12-28 |
| TW200509909A (en) | 2005-03-16 |
| CN1816533A (zh) | 2006-08-09 |
| MXPA05012299A (es) | 2006-01-30 |
| US20090105322A1 (en) | 2009-04-23 |
| WO2004101535A1 (en) | 2004-11-25 |
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