JP4709378B2 - 水不溶性物質のマイクロ粒子を製造するための組成物及び方法 - Google Patents

水不溶性物質のマイクロ粒子を製造するための組成物及び方法 Download PDF

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Publication number
JP4709378B2
JP4709378B2 JP2000540812A JP2000540812A JP4709378B2 JP 4709378 B2 JP4709378 B2 JP 4709378B2 JP 2000540812 A JP2000540812 A JP 2000540812A JP 2000540812 A JP2000540812 A JP 2000540812A JP 4709378 B2 JP4709378 B2 JP 4709378B2
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Prior art keywords
particles
phospholipid
water
phospholipids
composition
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Expired - Fee Related
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JP2000540812A
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Japanese (ja)
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JP2002509876A5 (enExample
JP2002509876A (ja
Inventor
カン，シーマ
ペース，ゲイリー・ダブリュー
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オバン・エナジー・リミテッド
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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
    • A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
    • A61K9/51—Nanocapsules; Nanoparticles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/146—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/145—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic compounds
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S977/00—Nanotechnology
    • Y10S977/902—Specified use of nanostructure
    • Y10S977/904—Specified use of nanostructure for medical, immunological, body treatment, or diagnosis
    • Y10S977/926—Topical chemical, e.g. cosmetic or sunscreen

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  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Physics & Mathematics (AREA)
  • Biomedical Technology (AREA)
  • Nanotechnology (AREA)
  • Optics & Photonics (AREA)
  • Medicinal Preparation (AREA)
  • Manufacturing Of Micro-Capsules (AREA)
JP2000540812A 1998-03-30 1999-03-29 水不溶性物質のマイクロ粒子を製造するための組成物及び方法 Expired - Fee Related JP4709378B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US7980998P 1998-03-30 1998-03-30
US60/079,809 1998-03-30
PCT/US1999/006746 WO1999049846A2 (en) 1998-03-30 1999-03-29 Compositions containing microparticles of water-insoluble substances and method for their preparation

Related Child Applications (1)

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JP2010232130A Division JP5539839B2 (ja) 1998-03-30 2010-10-15 水不溶性物質のマイクロ粒子を製造するための組成物及び方法

Publications (3)

Publication Number Publication Date
JP2002509876A JP2002509876A (ja) 2002-04-02
JP2002509876A5 JP2002509876A5 (enExample) 2006-04-27
JP4709378B2 true JP4709378B2 (ja) 2011-06-22

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Family Applications (2)

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JP2000540812A Expired - Fee Related JP4709378B2 (ja) 1998-03-30 1999-03-29 水不溶性物質のマイクロ粒子を製造するための組成物及び方法
JP2010232130A Expired - Fee Related JP5539839B2 (ja) 1998-03-30 2010-10-15 水不溶性物質のマイクロ粒子を製造するための組成物及び方法

Family Applications After (1)

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JP2010232130A Expired - Fee Related JP5539839B2 (ja) 1998-03-30 2010-10-15 水不溶性物質のマイクロ粒子を製造するための組成物及び方法

Country Status (14)

Country Link
US (1) US6387409B1 (enExample)
EP (1) EP1067914B1 (enExample)
JP (2) JP4709378B2 (enExample)
KR (1) KR100628341B1 (enExample)
CN (1) CN1303278B (enExample)
AT (1) ATE318132T1 (enExample)
AU (1) AU761205B2 (enExample)
CA (1) CA2326456C (enExample)
DE (1) DE69929959T2 (enExample)
ES (1) ES2257041T3 (enExample)
IL (3) IL138765A0 (enExample)
SE (1) SE0003429L (enExample)
TW (1) TWI267383B (enExample)
WO (1) WO1999049846A2 (enExample)

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Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2011037889A (ja) * 1998-03-30 2011-02-24 Oban Energy Ltd 水不溶性物質のマイクロ粒子を製造するための組成物及び方法

Also Published As

Publication number Publication date
TWI267383B (en) 2006-12-01
CN1303278A (zh) 2001-07-11
IL138765A0 (en) 2001-10-31
ATE318132T1 (de) 2006-03-15
WO1999049846A3 (en) 1999-11-18
ES2257041T3 (es) 2006-07-16
CN1303278B (zh) 2010-06-23
KR100628341B1 (ko) 2006-09-27
JP2011037889A (ja) 2011-02-24
AU761205B2 (en) 2003-05-29
US6387409B1 (en) 2002-05-14
SE0003429L (sv) 2000-11-23
IL162023A0 (en) 2005-11-20
JP5539839B2 (ja) 2014-07-02
EP1067914A2 (en) 2001-01-17
JP2002509876A (ja) 2002-04-02
WO1999049846A2 (en) 1999-10-07
DE69929959D1 (de) 2006-04-27
DE69929959T2 (de) 2006-11-02
CA2326456C (en) 2008-12-23
IL138765A (en) 2007-09-20
SE0003429D0 (sv) 2000-09-26
AU3118599A (en) 1999-10-18
KR20010042103A (ko) 2001-05-25
CA2326456A1 (en) 1999-10-07
EP1067914B1 (en) 2006-02-22

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