JP4386729B2 - オレフィンのアリール化法 - Google Patents

オレフィンのアリール化法 Download PDF

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Publication number
JP4386729B2
JP4386729B2 JP2003549274A JP2003549274A JP4386729B2 JP 4386729 B2 JP4386729 B2 JP 4386729B2 JP 2003549274 A JP2003549274 A JP 2003549274A JP 2003549274 A JP2003549274 A JP 2003549274A JP 4386729 B2 JP4386729 B2 JP 4386729B2
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JP
Japan
Prior art keywords
alkyl
aryl
group
general formula
palladium
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
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JP2003549274A
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English (en)
Japanese (ja)
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JP2005511667A (ja
JP2005511667A5 (https=
Inventor
ラムプフ フローリアン
エッケルト マルクス
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Lanxess Deutschland GmbH
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Lanxess Deutschland GmbH
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Publication date
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Publication of JP2005511667A publication Critical patent/JP2005511667A/ja
Publication of JP2005511667A5 publication Critical patent/JP2005511667A5/ja
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C253/00—Preparation of carboxylic acid nitriles
    • C07C253/30—Preparation of carboxylic acid nitriles by reactions not involving the formation of cyano groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B37/00—Reactions without formation or introduction of functional groups containing hetero atoms, involving either the formation of a carbon-to-carbon bond between two carbon atoms not directly linked already or the disconnection of two directly linked carbon atoms
    • C07B37/04—Substitution
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00—Preparation of halogenated hydrocarbons
    • C07C17/26—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton
    • C07C17/263—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton by condensation reactions
    • C07C17/266—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton by condensation reactions of hydrocarbons and halogenated hydrocarbons
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C67/00—Preparation of carboxylic acid esters
    • C07C67/30—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group
    • C07C67/333—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by isomerisation; by change of size of the carbon skeleton
    • C07C67/343—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
JP2003549274A 2001-12-03 2002-11-20 オレフィンのアリール化法 Expired - Fee Related JP4386729B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10159270A DE10159270A1 (de) 2001-12-03 2001-12-03 Verfahren zur Arylierung von Olefinen
PCT/EP2002/012993 WO2003048079A2 (de) 2001-12-03 2002-11-20 Verfahren zur arylierung von olefinen

Publications (3)

Publication Number Publication Date
JP2005511667A JP2005511667A (ja) 2005-04-28
JP2005511667A5 JP2005511667A5 (https=) 2006-01-05
JP4386729B2 true JP4386729B2 (ja) 2009-12-16

Family

ID=7707839

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2003549274A Expired - Fee Related JP4386729B2 (ja) 2001-12-03 2002-11-20 オレフィンのアリール化法

Country Status (9)

Country Link
US (1) US7102046B2 (https=)
EP (1) EP1453774B1 (https=)
JP (1) JP4386729B2 (https=)
AT (1) ATE421491T1 (https=)
AU (1) AU2002356692A1 (https=)
DE (2) DE10159270A1 (https=)
ES (1) ES2318065T3 (https=)
IL (2) IL162237A0 (https=)
WO (1) WO2003048079A2 (https=)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3613743B1 (en) 2008-01-04 2022-03-16 Intellikine, LLC Processes for the preparation of 1h-pyrazolo[3,4-d]pyrimidin-4-amine derivatives
US8193182B2 (en) 2008-01-04 2012-06-05 Intellikine, Inc. Substituted isoquinolin-1(2H)-ones, and methods of use thereof
TWI674262B (zh) 2011-01-10 2019-10-11 美商英菲尼提製藥股份有限公司 製備異喹啉酮之方法及異喹啉酮之固體形式
US8828998B2 (en) 2012-06-25 2014-09-09 Infinity Pharmaceuticals, Inc. Treatment of lupus, fibrotic conditions, and inflammatory myopathies and other disorders using PI3 kinase inhibitors
EP2914296B2 (en) 2012-11-01 2021-09-29 Infinity Pharmaceuticals, Inc. Treatment of cancers using pi3 kinase isoform modulators
FR2997696B1 (fr) * 2012-11-08 2014-12-05 Servier Lab Nouveau procede de synthese du (2e)-3-(3,4-dimethoxyphenyl)prop-2-enenitrile, et application a la synthese de l'ivabradine et de ses sels d'addition a un acide pharmaceutiquement acceptable
WO2015160975A2 (en) 2014-04-16 2015-10-22 Infinity Pharmaceuticals, Inc. Combination therapies
RU2754507C2 (ru) 2016-06-24 2021-09-02 Инфинити Фармасьютикалз, Инк. Комбинированная терапия
EP3945105A1 (en) 2020-07-30 2022-02-02 Basf Se Process for preparing a hydroxy group functionalized thioether

Also Published As

Publication number Publication date
EP1453774A2 (de) 2004-09-08
JP2005511667A (ja) 2005-04-28
IL162237A0 (en) 2005-11-20
AU2002356692A8 (en) 2003-06-17
US20030105353A1 (en) 2003-06-05
ES2318065T3 (es) 2009-05-01
ATE421491T1 (de) 2009-02-15
DE50213245D1 (de) 2009-03-12
WO2003048079A2 (de) 2003-06-12
US7102046B2 (en) 2006-09-05
AU2002356692A1 (en) 2003-06-17
DE10159270A1 (de) 2003-06-12
WO2003048079A3 (de) 2003-12-18
IL162237A (en) 2010-06-16
EP1453774B1 (de) 2009-01-21

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