JP4386729B2 - オレフィンのアリール化法 - Google Patents

オレフィンのアリール化法 Download PDF

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Publication number
JP4386729B2
JP4386729B2 JP2003549274A JP2003549274A JP4386729B2 JP 4386729 B2 JP4386729 B2 JP 4386729B2 JP 2003549274 A JP2003549274 A JP 2003549274A JP 2003549274 A JP2003549274 A JP 2003549274A JP 4386729 B2 JP4386729 B2 JP 4386729B2
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JP
Japan
Prior art keywords
alkyl
aryl
group
general formula
palladium
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
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JP2003549274A
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English (en)
Japanese (ja)
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JP2005511667A5 (enExample
JP2005511667A (ja
Inventor
ラムプフ フローリアン
エッケルト マルクス
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Lanxess Deutschland GmbH
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Lanxess Deutschland GmbH
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Publication of JP2005511667A5 publication Critical patent/JP2005511667A5/ja
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C253/00—Preparation of carboxylic acid nitriles
    • C07C253/30—Preparation of carboxylic acid nitriles by reactions not involving the formation of cyano groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B37/00—Reactions without formation or introduction of functional groups containing hetero atoms, involving either the formation of a carbon-to-carbon bond between two carbon atoms not directly linked already or the disconnection of two directly linked carbon atoms
    • C07B37/04—Substitution
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C17/00—Preparation of halogenated hydrocarbons
    • C07C17/26—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton
    • C07C17/263—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton by condensation reactions
    • C07C17/266—Preparation of halogenated hydrocarbons by reactions involving an increase in the number of carbon atoms in the skeleton by condensation reactions of hydrocarbons and halogenated hydrocarbons
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C231/00—Preparation of carboxylic acid amides
    • C07C231/12—Preparation of carboxylic acid amides by reactions not involving the formation of carboxamide groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C67/00—Preparation of carboxylic acid esters
    • C07C67/30—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group
    • C07C67/333—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by isomerisation; by change of size of the carbon skeleton
    • C07C67/343—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
JP2003549274A 2001-12-03 2002-11-20 オレフィンのアリール化法 Expired - Fee Related JP4386729B2 (ja)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10159270A DE10159270A1 (de) 2001-12-03 2001-12-03 Verfahren zur Arylierung von Olefinen
PCT/EP2002/012993 WO2003048079A2 (de) 2001-12-03 2002-11-20 Verfahren zur arylierung von olefinen

Publications (3)

Publication Number Publication Date
JP2005511667A JP2005511667A (ja) 2005-04-28
JP2005511667A5 JP2005511667A5 (enExample) 2006-01-05
JP4386729B2 true JP4386729B2 (ja) 2009-12-16

Family

ID=7707839

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2003549274A Expired - Fee Related JP4386729B2 (ja) 2001-12-03 2002-11-20 オレフィンのアリール化法

Country Status (9)

Country Link
US (1) US7102046B2 (enExample)
EP (1) EP1453774B1 (enExample)
JP (1) JP4386729B2 (enExample)
AT (1) ATE421491T1 (enExample)
AU (1) AU2002356692A1 (enExample)
DE (2) DE10159270A1 (enExample)
ES (1) ES2318065T3 (enExample)
IL (2) IL162237A0 (enExample)
WO (1) WO2003048079A2 (enExample)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8193182B2 (en) 2008-01-04 2012-06-05 Intellikine, Inc. Substituted isoquinolin-1(2H)-ones, and methods of use thereof
DK2240451T3 (da) 2008-01-04 2017-11-20 Intellikine Llc Isoquinolinonderivater substitueret med en purin, der er anvendelig som pi3k-inhibitorer
PE20180318A1 (es) 2011-01-10 2018-02-09 Infinity Pharmaceuticals Inc Procedimiento para preparar isoquinolinonas y formas solidas de isoquinolinonas
US8828998B2 (en) 2012-06-25 2014-09-09 Infinity Pharmaceuticals, Inc. Treatment of lupus, fibrotic conditions, and inflammatory myopathies and other disorders using PI3 kinase inhibitors
LT2914296T (lt) 2012-11-01 2018-09-25 Infinity Pharmaceuticals, Inc. Vėžio gydymas, panaudojant p13 kinazės izoformos moduliatorius
FR2997696B1 (fr) * 2012-11-08 2014-12-05 Servier Lab Nouveau procede de synthese du (2e)-3-(3,4-dimethoxyphenyl)prop-2-enenitrile, et application a la synthese de l'ivabradine et de ses sels d'addition a un acide pharmaceutiquement acceptable
US20150320755A1 (en) 2014-04-16 2015-11-12 Infinity Pharmaceuticals, Inc. Combination therapies
UA125216C2 (uk) 2016-06-24 2022-02-02 Інфініті Фармасьютікалз, Інк. Комбінована терапія
EP3945105A1 (en) 2020-07-30 2022-02-02 Basf Se Process for preparing a hydroxy group functionalized thioether

Also Published As

Publication number Publication date
WO2003048079A2 (de) 2003-06-12
WO2003048079A3 (de) 2003-12-18
DE10159270A1 (de) 2003-06-12
AU2002356692A1 (en) 2003-06-17
IL162237A0 (en) 2005-11-20
IL162237A (en) 2010-06-16
ATE421491T1 (de) 2009-02-15
EP1453774A2 (de) 2004-09-08
DE50213245D1 (de) 2009-03-12
ES2318065T3 (es) 2009-05-01
EP1453774B1 (de) 2009-01-21
JP2005511667A (ja) 2005-04-28
US7102046B2 (en) 2006-09-05
AU2002356692A8 (en) 2003-06-17
US20030105353A1 (en) 2003-06-05

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