JP2025511404A5 - - Google Patents

Info

Publication number
JP2025511404A5
JP2025511404A5 JP2024559037A JP2024559037A JP2025511404A5 JP 2025511404 A5 JP2025511404 A5 JP 2025511404A5 JP 2024559037 A JP2024559037 A JP 2024559037A JP 2024559037 A JP2024559037 A JP 2024559037A JP 2025511404 A5 JP2025511404 A5 JP 2025511404A5
Authority
JP
Japan
Prior art keywords
compound
formula
salt
process according
reaction
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024559037A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025511404A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/EP2023/059132 external-priority patent/WO2023194531A1/en
Publication of JP2025511404A publication Critical patent/JP2025511404A/ja
Publication of JP2025511404A5 publication Critical patent/JP2025511404A5/ja
Pending legal-status Critical Current

Links

JP2024559037A 2022-04-07 2023-04-06 オシメルチニブを製造するための改善されたプロセス Pending JP2025511404A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202263362622P 2022-04-07 2022-04-07
US63/362,622 2022-04-07
PCT/EP2023/059132 WO2023194531A1 (en) 2022-04-07 2023-04-06 Improved process for the manufacture of osimertinib

Publications (2)

Publication Number Publication Date
JP2025511404A JP2025511404A (ja) 2025-04-15
JP2025511404A5 true JP2025511404A5 (https=) 2026-04-14

Family

ID=86142780

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024559037A Pending JP2025511404A (ja) 2022-04-07 2023-04-06 オシメルチニブを製造するための改善されたプロセス

Country Status (14)

Country Link
US (1) US20250250255A1 (https=)
EP (1) EP4504718A1 (https=)
JP (1) JP2025511404A (https=)
KR (1) KR20250002363A (https=)
CN (1) CN119317624A (https=)
AR (1) AR128999A1 (https=)
AU (1) AU2023250220A1 (https=)
CA (1) CA3255378A1 (https=)
CO (1) CO2024015096A2 (https=)
IL (1) IL316018A (https=)
MX (1) MX2024012370A (https=)
TW (1) TW202404955A (https=)
WO (1) WO2023194531A1 (https=)
ZA (1) ZA202408113B (https=)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN120717920A (zh) * 2025-08-18 2025-09-30 爱斯特(成都)生物制药股份有限公司 一种微通道连续合成3-硝基-4-氟苯腈的方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4119551A1 (en) 2011-07-27 2023-01-18 Astrazeneca AB 2-(2,4,5-substituted-anilino)pyrimidine compounds
CN106883216B (zh) * 2017-04-06 2020-03-13 张家港威胜生物医药有限公司 一种奥希替尼的制备方法
IN201741031902A (https=) * 2017-09-08 2019-03-15 Msn Laboratories Private Ltd
CN109134435B (zh) 2018-10-29 2023-01-03 湖南大学 一种奥希替尼azd9291的合成方法

Similar Documents

Publication Publication Date Title
JP5513508B2 (ja) アミノスルホン化合物を調製するためのプロセス
JP7379567B2 (ja) (2r,6r)-ヒドロキシノルケタミンおよび(2s,6s)-ヒドロキシノルケタミンの結晶形態および合成方法
JP2025511404A5 (https=)
US20100081807A1 (en) Method for producing 5-cloro-n-(methyl)-2-thiophenecarboxamide
JP2019048806A5 (https=)
JP2020519583A5 (https=)
JPWO2009125841A1 (ja) 5−メチルウリジンを出発原料とするエチニルチミジン化合物の製造方法
CN106029641B (zh) 1,1-二取代肼化合物的制造方法
JP4890267B2 (ja) 無水プロパンホスホン酸の脱水反応によるニトリルおよびイソニトリルの製造法
RU2006139128A (ru) Способ получения фторированных олефинов
JP5629260B2 (ja) トリフルオロメチルチオフェニウム誘導体塩、その製造方法並びにそれを用いたトリフルオロメチル基含有化合物類の製造法
US9663505B2 (en) Process for the preparation of rivaroxaban
JP2013530948A5 (https=)
CN108373453A (zh) 三氮唑衍生物及其制备方法
García-Egido et al. Synthesis of cyanoformamides from primary amines and carbon dioxide under mild conditions. Synthesis of ceratinamine
JP2023513186A (ja) (r)-2-アミノブタン酸からのs-ベフルブタミドの合成プロセス
JP6257115B2 (ja) 3−アルキルチオ−2−ブロモピリジンの製造方法
CN102203111B (zh) 2,4-二取代的1,3 -氧硫杂环戊烷核苷的对映体拆分
JP2001354597A (ja) シクロプロペン類の製造方法
US20250250255A1 (en) Improved process for the manufacture of osimertinib
JP2022528611A5 (https=)
JP2022528612A5 (https=)
Inoue et al. Stereoselective aldol reactions using pseudo C 2 symmetric 1-benzyl-4-(trifluoromethyl) piperidine-2, 6-dione
CN108699049A (zh) 用于制备苯并噁唑化合物的方法
CN113429411A (zh) 一种1-烃基-6-氯-1H-吡唑并[3,4-d]嘧啶化合物的制备方法