JP2025508435A5 - - Google Patents

Info

Publication number
JP2025508435A5
JP2025508435A5 JP2024548743A JP2024548743A JP2025508435A5 JP 2025508435 A5 JP2025508435 A5 JP 2025508435A5 JP 2024548743 A JP2024548743 A JP 2024548743A JP 2024548743 A JP2024548743 A JP 2024548743A JP 2025508435 A5 JP2025508435 A5 JP 2025508435A5
Authority
JP
Japan
Prior art keywords
pharmaceutical composition
cancer
disorders
solvate
pharmaceutically acceptable
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024548743A
Other languages
English (en)
Japanese (ja)
Other versions
JP2025508435A (ja
Filing date
Publication date
Priority claimed from GBGB2202199.2A external-priority patent/GB202202199D0/en
Application filed filed Critical
Publication of JP2025508435A publication Critical patent/JP2025508435A/ja
Publication of JP2025508435A5 publication Critical patent/JP2025508435A5/ja
Pending legal-status Critical Current

Links

JP2024548743A 2022-02-18 2023-02-17 Erk5媒介性疾患を治療するのに有用な複素環式化合物 Pending JP2025508435A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB2202199.2 2022-02-18
GBGB2202199.2A GB202202199D0 (en) 2022-02-18 2022-02-18 Compounds
PCT/GB2023/050369 WO2023156791A1 (en) 2022-02-18 2023-02-17 Heterocyclic compounds useful for treating a erk5-mediated disease

Publications (2)

Publication Number Publication Date
JP2025508435A JP2025508435A (ja) 2025-03-26
JP2025508435A5 true JP2025508435A5 (enExample) 2026-01-08

Family

ID=80934460

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024548743A Pending JP2025508435A (ja) 2022-02-18 2023-02-17 Erk5媒介性疾患を治療するのに有用な複素環式化合物

Country Status (8)

Country Link
US (1) US20250154157A1 (enExample)
EP (1) EP4479400A1 (enExample)
JP (1) JP2025508435A (enExample)
CN (1) CN119053604A (enExample)
AU (1) AU2023220934A1 (enExample)
CA (1) CA3251985A1 (enExample)
GB (1) GB202202199D0 (enExample)
WO (1) WO2023156791A1 (enExample)

Family Cites Families (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB9624482D0 (en) 1995-12-18 1997-01-15 Zeneca Phaema S A Chemical compounds
WO1997030035A1 (en) 1996-02-13 1997-08-21 Zeneca Limited Quinazoline derivatives as vegf inhibitors
ES2169355T3 (es) 1996-03-05 2002-07-01 Astrazeneca Ab Derivados de 4-anilinoquinazolina.
GB9718972D0 (en) 1996-09-25 1997-11-12 Zeneca Ltd Chemical compounds
GB9714249D0 (en) 1997-07-08 1997-09-10 Angiogene Pharm Ltd Vascular damaging agents
GB9900334D0 (en) 1999-01-07 1999-02-24 Angiogene Pharm Ltd Tricylic vascular damaging agents
GB9900752D0 (en) 1999-01-15 1999-03-03 Angiogene Pharm Ltd Benzimidazole vascular damaging agents
BRPI0017548B8 (pt) 1999-02-10 2023-05-02 Astrazeneca Ab Composto
IL152682A0 (en) 2000-05-31 2003-06-24 Astrazeneca Ab Indole derivatives with vascular damaging activity
UA73993C2 (uk) 2000-06-06 2005-10-17 Астразенека Аб Хіназолінові похідні для лікування пухлин та фармацевтична композиція
HUP0301742A3 (en) 2000-07-07 2005-08-29 Angiogene Pharm Ltd Colchinol derivatives as angiogenesis inhibitors, process for producing them, pharmaceutical compositions containing them and their use
BR0112224A (pt) 2000-07-07 2003-06-10 Angiogene Pharm Ltd Composto, composição farmacêutica, uso de um composto ou de um sal, solvato ou pró-droga farmaceuticamente aceitável do mesmo, e, processo para preparar um composto
JP2017504650A (ja) * 2014-01-31 2017-02-09 ダナ−ファーバー キャンサー インスティテュート, インコーポレイテッド ジアゼパン誘導体およびその使用
WO2015117087A1 (en) * 2014-01-31 2015-08-06 Dana-Farber Cancer Institute, Inc. Uses of diazepane derivatives
WO2015129927A1 (en) * 2014-02-26 2015-09-03 Kyorin Pharmaceutical Co., Ltd. Heterocyclic compounds
EP4034132B1 (en) 2019-09-27 2026-02-25 Dana-Farber Cancer Institute, Inc. Erk5 degraders as therapeutics in cancer and inflammatory diseases

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