JP2023538125A5 - - Google Patents

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Publication number
JP2023538125A5
JP2023538125A5 JP2023512428A JP2023512428A JP2023538125A5 JP 2023538125 A5 JP2023538125 A5 JP 2023538125A5 JP 2023512428 A JP2023512428 A JP 2023512428A JP 2023512428 A JP2023512428 A JP 2023512428A JP 2023538125 A5 JP2023538125 A5 JP 2023538125A5
Authority
JP
Japan
Prior art keywords
pharmaceutical product
product according
gsi
semagacestat
approximately
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023512428A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023538125A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/046742 external-priority patent/WO2022040447A2/en
Publication of JP2023538125A publication Critical patent/JP2023538125A/ja
Publication of JP2023538125A5 publication Critical patent/JP2023538125A5/ja
Pending legal-status Critical Current

Links

JP2023512428A 2020-08-20 2021-08-19 粘液過剰分泌を特徴とする呼吸器疾患を処置するための方法 Pending JP2023538125A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063068235P 2020-08-20 2020-08-20
US63/068,235 2020-08-20
PCT/US2021/046742 WO2022040447A2 (en) 2020-08-20 2021-08-19 Methods for treating respiratory diseases characterized by mucus hypersecretion

Publications (2)

Publication Number Publication Date
JP2023538125A JP2023538125A (ja) 2023-09-06
JP2023538125A5 true JP2023538125A5 (enExample) 2024-08-20

Family

ID=80323184

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023512428A Pending JP2023538125A (ja) 2020-08-20 2021-08-19 粘液過剰分泌を特徴とする呼吸器疾患を処置するための方法

Country Status (11)

Country Link
US (1) US20230277550A1 (enExample)
EP (1) EP4199914A4 (enExample)
JP (1) JP2023538125A (enExample)
KR (1) KR20230052954A (enExample)
CN (1) CN116033895A (enExample)
AU (1) AU2021329507A1 (enExample)
BR (1) BR112023002651A2 (enExample)
CA (1) CA3188234A1 (enExample)
IL (1) IL300405A (enExample)
MX (1) MX2023001993A (enExample)
WO (1) WO2022040447A2 (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP4268824A1 (en) * 2022-04-26 2023-11-01 Manros Therapeutics Imidazo[2,1-f][1,2,4]triazine derivatives useful as a medicament
WO2024112356A1 (en) * 2022-11-23 2024-05-30 The Board Of Trustees Of The Leland Stanford Junior University Methods for treating respiratory diseases characterized by mucus hypersecretion

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SE0101004D0 (sv) 2001-03-21 2001-03-21 Astrazeneca Ab New measuring technique
LT2502911T (lt) 2004-06-24 2017-09-11 Vertex Pharmaceuticals Incorporated Atp surišančios kasetės transporterių moduliatoriai
WO2007079139A2 (en) 2005-12-28 2007-07-12 Vertex Pharmaceuticals, Inc. Solid forms of n-[2,4-bis(1,1-dimethylethyl)-5-hydroxyphenyl]-1,4-dihydro-4-oxoquinoline-3-carboxamide
CA2644136A1 (en) * 2006-02-27 2007-09-07 The Johns Hopkins University Cancer treatment with gamma-secretase inhibitors
US7645789B2 (en) 2006-04-07 2010-01-12 Vertex Pharmaceuticals Incorporated Indole derivatives as CFTR modulators
NZ571803A (en) 2006-04-07 2011-12-22 Vertex Pharma Amide indole derivatives as modulators of ATP-binding cassette transporters
SI2225230T1 (sl) 2007-12-07 2017-03-31 Vertex Pharmaceuticals Incorporated Trdne oblike 3-(6-(1-2,2-difluorobenzo(d)(1,3)dioxol-5-il)ciklopropan- karboksamido)-3-metilpiridin-2-il) benzojske kisline
US8299059B2 (en) 2009-10-30 2012-10-30 Eli Lilly And Company Crystalline compound and a process for its preparation
HUE040366T2 (hu) 2013-08-08 2019-03-28 Galapagos Nv CFTR modulátor tieno[2,3-c]piránok
EP2932966A1 (en) * 2014-04-16 2015-10-21 Novartis AG Gamma secretase inhibitors for treating respiratory diseases
TWI735416B (zh) 2014-10-06 2021-08-11 美商維泰克斯製藥公司 囊腫纖維化症跨膜傳導調節蛋白之調節劑
CA2971850A1 (en) 2014-12-23 2016-06-30 Proteostasis Therapeutics, Inc. Derivatives of 5-phenyl- or 5-heteroarylthiazol-2-carboxylic amide useful for the treatment of inter alia cystic fibrosis
MA42488A (fr) 2015-07-24 2018-05-30 Proteostasis Therapeutics Inc Composés, compositions et procédés pour augmenter l'activité du cftr
CA3000483C (en) 2015-10-06 2024-02-13 Proteostasis Therapeutics, Inc. Compounds, compositions, and methods for modulating cftr
US9890149B2 (en) 2015-10-07 2018-02-13 NuBridge BioSciences Isothiazole derivatives as CFTR modulators
RU2724345C2 (ru) 2015-10-09 2020-06-23 Галапагос Нв N-СУЛЬФОНИЛИРОВАННЫЕ ПИРАЗОЛО[3,4-b]ПИРИДИН-6-КАРБОКСАМИДЫ И СПОСОБ ИХ ПРИМЕНЕНИЯ
AU2017256172A1 (en) 2016-04-26 2018-09-06 AbbVie S.à.r.l. Modulators of cystic fibrosis transmembrane conductance regulator protein
US10138227B2 (en) 2016-06-03 2018-11-27 Abbvie S.Á.R.L. Heteroaryl substituted pyridines and methods of use
TW201811766A (zh) 2016-08-29 2018-04-01 瑞士商諾華公司 N-(吡啶-2-基)吡啶-磺醯胺衍生物及其用於疾病治療之用途
US10399940B2 (en) 2016-10-07 2019-09-03 Abbvie S.Á.R.L. Substituted pyrrolidines and methods of use
AU2017362350B2 (en) 2016-11-18 2021-12-23 Cystic Fibrosis Foundation Pyrrolopyrimidines as CFTR potentiators
US10131670B2 (en) 2016-12-16 2018-11-20 Cystic Fibrosis Foundation Therapeutics, Inc. Bicyclic heteroaryl derivatives as CFTR potentiators
MX2019009552A (es) * 2017-02-17 2019-10-02 Hutchinson Fred Cancer Res Terapias de combinacion para el tratamiento de canceres relacionados con el antigeno de maduracion de celulas b (bcma) y trastornos autoinmunitarios.
TW201831471A (zh) 2017-02-24 2018-09-01 盧森堡商艾伯維公司 囊腫纖化症跨膜傳導調節蛋白的調節劑及其使用方法
PL4010322T3 (pl) 2019-08-09 2026-02-16 Pfizer Inc. Stałe postacie (s)-2-(((s)-6,8-difluoro-1,2,3,4-tetrahydronaftalen-2-ylo)amino)-n-(1-(2-metylo-1-(neopentyloamino)propan-2-ylo)-1h-imidazol-4-ilo)pentanamidu i ich zastosowanie

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