JP2025502210A5 - - Google Patents
Info
- Publication number
- JP2025502210A5 JP2025502210A5 JP2024541811A JP2024541811A JP2025502210A5 JP 2025502210 A5 JP2025502210 A5 JP 2025502210A5 JP 2024541811 A JP2024541811 A JP 2024541811A JP 2024541811 A JP2024541811 A JP 2024541811A JP 2025502210 A5 JP2025502210 A5 JP 2025502210A5
- Authority
- JP
- Japan
- Prior art keywords
- formula
- methyl
- dimethylbenzoyl
- butoxycarbonyl
- oxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202263298751P | 2022-01-12 | 2022-01-12 | |
| US63/298,751 | 2022-01-12 | ||
| PCT/US2022/079176 WO2023136942A1 (en) | 2022-01-12 | 2022-11-02 | Synthetic intermediates and improved processes for preparing rock inhibitors |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2025502210A JP2025502210A (ja) | 2025-01-24 |
| JP2025502210A5 true JP2025502210A5 (cg-RX-API-DMAC7.html) | 2025-10-01 |
Family
ID=84462734
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024541811A Pending JP2025502210A (ja) | 2022-01-12 | 2022-11-02 | Rock阻害剤を調製するための合成中間体および改善したプロセス |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US20250109106A1 (cg-RX-API-DMAC7.html) |
| EP (1) | EP4463439A1 (cg-RX-API-DMAC7.html) |
| JP (1) | JP2025502210A (cg-RX-API-DMAC7.html) |
| KR (1) | KR20240134342A (cg-RX-API-DMAC7.html) |
| CN (1) | CN118696027A (cg-RX-API-DMAC7.html) |
| AU (1) | AU2022433635B2 (cg-RX-API-DMAC7.html) |
| CA (1) | CA3247774A1 (cg-RX-API-DMAC7.html) |
| IL (1) | IL314262A (cg-RX-API-DMAC7.html) |
| MX (1) | MX2024008610A (cg-RX-API-DMAC7.html) |
| WO (1) | WO2023136942A1 (cg-RX-API-DMAC7.html) |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP4191829B2 (ja) * | 1998-11-05 | 2008-12-03 | 大日本住友製薬株式会社 | 光学活性カルボン酸の製造方法 |
| WO2010126626A2 (en) | 2009-05-01 | 2010-11-04 | Aerie Pharmaceuticals, Inc. | Dual mechanism inhibitors for the treatment of disease |
| WO2017086941A1 (en) * | 2015-11-17 | 2017-05-26 | Aerie Pharmaceuticals, Inc. | Process for the preparation of kinase inhibitors and intermediates thereof |
| JP2021517137A (ja) * | 2018-03-23 | 2021-07-15 | フォチョン・ファーマシューティカルズ・リミテッドFochon Pharmaceuticals, Ltd. | Rock阻害剤としての重水素化合物 |
| EP3852790A4 (en) * | 2018-09-19 | 2022-08-10 | Forma Therapeutics, Inc. | INHIBITION OF UBIQUITIN-SPECIFIC PEPTIDASE 9X |
-
2022
- 2022-11-02 EP EP22821805.3A patent/EP4463439A1/en active Pending
- 2022-11-02 MX MX2024008610A patent/MX2024008610A/es unknown
- 2022-11-02 AU AU2022433635A patent/AU2022433635B2/en active Active
- 2022-11-02 US US18/728,421 patent/US20250109106A1/en active Pending
- 2022-11-02 CN CN202280088641.XA patent/CN118696027A/zh active Pending
- 2022-11-02 IL IL314262A patent/IL314262A/en unknown
- 2022-11-02 JP JP2024541811A patent/JP2025502210A/ja active Pending
- 2022-11-02 KR KR1020247026239A patent/KR20240134342A/ko active Pending
- 2022-11-02 WO PCT/US2022/079176 patent/WO2023136942A1/en not_active Ceased
- 2022-11-02 CA CA3247774A patent/CA3247774A1/en active Pending
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