JP2025160175A5 - - Google Patents
Info
- Publication number
- JP2025160175A5 JP2025160175A5 JP2025107301A JP2025107301A JP2025160175A5 JP 2025160175 A5 JP2025160175 A5 JP 2025160175A5 JP 2025107301 A JP2025107301 A JP 2025107301A JP 2025107301 A JP2025107301 A JP 2025107301A JP 2025160175 A5 JP2025160175 A5 JP 2025160175A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- pharmaceutically acceptable
- acceptable salt
- independently selected
- haloalkyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202163143245P | 2021-01-29 | 2021-01-29 | |
| US63/143,245 | 2021-01-29 | ||
| JP2023544674A JP7777596B2 (ja) | 2021-01-29 | 2022-01-28 | Cd38阻害剤としてのキノリン及びアザキノリン |
| PCT/US2022/014221 WO2022165114A1 (en) | 2021-01-29 | 2022-01-28 | Quinolines and azaquinolines as inhibitors of cd38 |
Related Parent Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023544674A Division JP7777596B2 (ja) | 2021-01-29 | 2022-01-28 | Cd38阻害剤としてのキノリン及びアザキノリン |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2025160175A JP2025160175A (ja) | 2025-10-22 |
| JP2025160175A5 true JP2025160175A5 (https=) | 2026-03-13 |
Family
ID=80446310
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023544674A Active JP7777596B2 (ja) | 2021-01-29 | 2022-01-28 | Cd38阻害剤としてのキノリン及びアザキノリン |
| JP2025107301A Pending JP2025160175A (ja) | 2021-01-29 | 2025-06-25 | Cd38阻害剤としてのキノリン及びアザキノリン |
Family Applications Before (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023544674A Active JP7777596B2 (ja) | 2021-01-29 | 2022-01-28 | Cd38阻害剤としてのキノリン及びアザキノリン |
Country Status (25)
| Country | Link |
|---|---|
| US (2) | US11952377B2 (https=) |
| EP (2) | EP4674415A3 (https=) |
| JP (2) | JP7777596B2 (https=) |
| KR (1) | KR20230141799A (https=) |
| CN (1) | CN117580829A (https=) |
| AR (1) | AR124718A1 (https=) |
| AU (1) | AU2022212035A1 (https=) |
| BR (1) | BR112023014898A2 (https=) |
| CA (1) | CA3208851A1 (https=) |
| CL (2) | CL2023002163A1 (https=) |
| CO (1) | CO2023009803A2 (https=) |
| CR (1) | CR20230323A (https=) |
| DO (1) | DOP2023000142A (https=) |
| EC (1) | ECSP23056223A (https=) |
| ES (1) | ES3042412T3 (https=) |
| HR (1) | HRP20251111T1 (https=) |
| HU (1) | HUE072981T2 (https=) |
| IL (1) | IL304466A (https=) |
| JO (1) | JOP20230160A1 (https=) |
| MX (1) | MX2023008701A (https=) |
| PE (1) | PE20232047A1 (https=) |
| PL (1) | PL4284511T3 (https=) |
| RS (1) | RS67253B1 (https=) |
| TW (1) | TW202241418A (https=) |
| WO (1) | WO2022165114A1 (https=) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2021021986A1 (en) | 2019-07-31 | 2021-02-04 | Ribon Therapeutics, Inc. | Heterobicyclic amides as inhibitors of cd38 |
| WO2024217995A1 (en) | 2023-04-20 | 2024-10-24 | Syngenta Crop Protection Ag | Pesticidally active dihydropyridinone derivatives |
| WO2026000074A1 (en) * | 2024-06-25 | 2026-01-02 | Welnx Company Inc. | Use of cd38 inhibitors for reducing th2 inflammation |
| WO2026075971A1 (en) | 2024-10-01 | 2026-04-09 | Neolaia Inc. | Combination therapy for treatment of metabolic disorders and inflamation related disorders using incretin compounds and cd38 inhibitors |
| CN119775288B (zh) * | 2024-12-31 | 2025-10-10 | 浙江工业大学 | 一种cd38抑制化合物及应用 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ES2607064T3 (es) | 2010-12-01 | 2017-03-29 | Glaxosmithkline Llc | Indoles |
| BR112014010803A2 (pt) | 2011-11-04 | 2017-04-25 | Glaxosmithkline Intellectual Property (No 2) Ltd | método de tratamento |
| JP6464139B2 (ja) * | 2013-03-14 | 2019-02-06 | コンバージーン・リミテッド・ライアビリティ・カンパニーConvergene Llc | ブロモドメイン含有タンパク質の阻害のための方法および組成物 |
| AU2015356721B2 (en) | 2014-12-03 | 2018-03-15 | Glaxosmithkline Intellectual Property (No.2) Limited | CD38 inhibitors and methods of treatment |
| WO2017053604A1 (en) | 2015-09-23 | 2017-03-30 | The Regents Of The University Of California | Potent antiviral pyrazolopyridine compounds |
| WO2018151830A1 (en) | 2017-02-17 | 2018-08-23 | Fronthera U.S. Pharmaceuticals Llc | Pyridinyl based apoptosis signal-regulation kinase inhibitors |
| EP3434692A1 (en) | 2017-07-24 | 2019-01-30 | Encefa | Compounds which specifically binds to cd38 for use in the treatment of neurodegenerative diseases |
| WO2021021986A1 (en) | 2019-07-31 | 2021-02-04 | Ribon Therapeutics, Inc. | Heterobicyclic amides as inhibitors of cd38 |
| US20230025807A1 (en) | 2019-10-30 | 2023-01-26 | Mitobridge Inc. | Cd38 inhibitors |
| BR112022020291A2 (pt) | 2020-04-07 | 2022-12-06 | Mitobridge Inc | Inibidores de cd38 |
-
2022
- 2022-01-28 HR HRP20251111TT patent/HRP20251111T1/hr unknown
- 2022-01-28 CA CA3208851A patent/CA3208851A1/en active Pending
- 2022-01-28 CR CR20230323A patent/CR20230323A/es unknown
- 2022-01-28 RS RS20250955A patent/RS67253B1/sr unknown
- 2022-01-28 PL PL22704226.4T patent/PL4284511T3/pl unknown
- 2022-01-28 MX MX2023008701A patent/MX2023008701A/es unknown
- 2022-01-28 AR ARP220100173A patent/AR124718A1/es unknown
- 2022-01-28 TW TW111103880A patent/TW202241418A/zh unknown
- 2022-01-28 EP EP25188747.7A patent/EP4674415A3/en active Pending
- 2022-01-28 EP EP22704226.4A patent/EP4284511B1/en active Active
- 2022-01-28 AU AU2022212035A patent/AU2022212035A1/en active Pending
- 2022-01-28 BR BR112023014898A patent/BR112023014898A2/pt unknown
- 2022-01-28 CN CN202280022060.6A patent/CN117580829A/zh active Pending
- 2022-01-28 PE PE2023002190A patent/PE20232047A1/es unknown
- 2022-01-28 KR KR1020237027359A patent/KR20230141799A/ko active Pending
- 2022-01-28 HU HUE22704226A patent/HUE072981T2/hu unknown
- 2022-01-28 ES ES22704226T patent/ES3042412T3/es active Active
- 2022-01-28 JP JP2023544674A patent/JP7777596B2/ja active Active
- 2022-01-28 WO PCT/US2022/014221 patent/WO2022165114A1/en not_active Ceased
- 2022-01-28 US US17/586,939 patent/US11952377B2/en active Active
-
2023
- 2023-07-13 IL IL304466A patent/IL304466A/en unknown
- 2023-07-20 JO JOJO/P/2023/0160A patent/JOP20230160A1/ar unknown
- 2023-07-24 CL CL2023002163A patent/CL2023002163A1/es unknown
- 2023-07-25 DO DO2023000142A patent/DOP2023000142A/es unknown
- 2023-07-25 EC ECSENADI202356223A patent/ECSP23056223A/es unknown
- 2023-07-25 CO CONC2023/0009803A patent/CO2023009803A2/es unknown
-
2024
- 2024-02-28 US US18/590,300 patent/US20240279224A1/en active Pending
- 2024-05-22 CL CL2024001535A patent/CL2024001535A1/es unknown
-
2025
- 2025-06-25 JP JP2025107301A patent/JP2025160175A/ja active Pending
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