JP2024543973A5 - - Google Patents

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Publication number
JP2024543973A5
JP2024543973A5 JP2024532491A JP2024532491A JP2024543973A5 JP 2024543973 A5 JP2024543973 A5 JP 2024543973A5 JP 2024532491 A JP2024532491 A JP 2024532491A JP 2024532491 A JP2024532491 A JP 2024532491A JP 2024543973 A5 JP2024543973 A5 JP 2024543973A5
Authority
JP
Japan
Prior art keywords
pharmaceutically acceptable
acceptable salt
compound according
alkyl
pharmaceutical composition
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2024532491A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024543973A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/051493 external-priority patent/WO2023102100A1/en
Publication of JP2024543973A publication Critical patent/JP2024543973A/ja
Publication of JP2024543973A5 publication Critical patent/JP2024543973A5/ja
Pending legal-status Critical Current

Links

JP2024532491A 2021-12-01 2022-12-01 ムスカリン性アセチルコリン受容体m4のアンタゴニスト Pending JP2024543973A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202163284750P 2021-12-01 2021-12-01
US63/284,750 2021-12-01
PCT/US2022/051493 WO2023102100A1 (en) 2021-12-01 2022-12-01 Antagonists of the muscarinic acetylcholine receptor m4

Publications (2)

Publication Number Publication Date
JP2024543973A JP2024543973A (ja) 2024-11-26
JP2024543973A5 true JP2024543973A5 (https=) 2025-12-08

Family

ID=84943708

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2024532491A Pending JP2024543973A (ja) 2021-12-01 2022-12-01 ムスカリン性アセチルコリン受容体m4のアンタゴニスト

Country Status (10)

Country Link
US (1) US20250145595A1 (https=)
EP (1) EP4441046A1 (https=)
JP (1) JP2024543973A (https=)
KR (1) KR20240112343A (https=)
CN (2) CN116669737A (https=)
AU (1) AU2022400780A1 (https=)
CA (1) CA3241298A1 (https=)
IL (1) IL313219A (https=)
MX (1) MX2024006718A (https=)
WO (1) WO2023102100A1 (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2018300980A1 (en) 2017-07-12 2020-01-02 Vanderbilt University Antagonists of the muscarinic acetylcholine receptor M4
IL273924B2 (en) 2017-10-20 2024-07-01 Univ Vanderbilt Antagonists of the muscarinic acetylcholine receptor m4
CA3155864A1 (en) 2019-10-04 2021-04-08 Vanderbilt University Antagonists of the muscarinic acetylcholine receptor m4
EP4491228A3 (en) * 2020-12-22 2025-04-23 Vanderbilt University Antagonists of the muscarinic acetylcholine receptor m4

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112018003417B1 (pt) * 2016-06-22 2023-10-24 Vanderbilt University Composto modulador alostérico positivo do receptor muscarínico de acetilcolina m4 e composição farmacêutica que o compreende
JP2020530451A (ja) * 2017-08-08 2020-10-22 ヴァンダービルト ユニバーシティー ムスカリン性アセチルコリン受容体m4のアンタゴニスト
IL273924B2 (en) * 2017-10-20 2024-07-01 Univ Vanderbilt Antagonists of the muscarinic acetylcholine receptor m4
WO2021119254A1 (en) * 2019-12-10 2021-06-17 Vanderbilt University Antagonists of the muscarinic acetylcholine receptor m4
US20230183218A1 (en) * 2020-04-24 2023-06-15 Vanderbilt University Condensed substituted hydropyrroles as antagonists of the muscarinic acetylcholine receptor m4
EP4139303A1 (en) * 2020-04-24 2023-03-01 Vanderbilt University Condensed substituted hydropyrroles as antagonists of the muscarinic acetylcholine receptor m4

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