JP2024536858A5 - - Google Patents
Info
- Publication number
- JP2024536858A5 JP2024536858A5 JP2024518772A JP2024518772A JP2024536858A5 JP 2024536858 A5 JP2024536858 A5 JP 2024536858A5 JP 2024518772 A JP2024518772 A JP 2024518772A JP 2024518772 A JP2024518772 A JP 2024518772A JP 2024536858 A5 JP2024536858 A5 JP 2024536858A5
- Authority
- JP
- Japan
- Prior art keywords
- phenyl
- amino
- methyl
- pyrrolo
- pyridine
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CNPCT/CN2021/119861 | 2021-09-23 | ||
| CN2021119861 | 2021-09-23 | ||
| CN2022096894 | 2022-06-02 | ||
| CNPCT/CN2022/096894 | 2022-06-02 | ||
| PCT/CN2022/121076 WO2023046117A1 (en) | 2021-09-23 | 2022-09-23 | Fgfr inhibitors and methods of use thereof |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2024536858A JP2024536858A (ja) | 2024-10-08 |
| JP2024536858A5 true JP2024536858A5 (https=) | 2025-06-25 |
Family
ID=85720119
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2024518772A Pending JP2024536858A (ja) | 2021-09-23 | 2022-09-23 | Fgfr阻害剤及びその使用方法 |
Country Status (8)
| Country | Link |
|---|---|
| US (1) | US20240383905A1 (https=) |
| EP (1) | EP4405358A4 (https=) |
| JP (1) | JP2024536858A (https=) |
| KR (1) | KR20240075952A (https=) |
| CN (1) | CN118043327A (https=) |
| AU (1) | AU2022350571A1 (https=) |
| CA (1) | CA3231948A1 (https=) |
| WO (1) | WO2023046117A1 (https=) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN117402161A (zh) * | 2022-07-06 | 2024-01-16 | 上海科恩泰生物医药科技有限公司 | 一种具有fgfr抑制作用的亚砜亚胺类化合物、包含其的药物组合物及其用途 |
| CN115232147B (zh) * | 2022-08-09 | 2023-10-13 | 南方科技大学 | 一种作为HIF-2α激动剂的杂环衍生物 |
| CN120344533A (zh) * | 2022-11-22 | 2025-07-18 | 海思科医药集团股份有限公司 | 一种嘧啶衍生物及其在医药上的应用 |
| WO2024208315A1 (zh) * | 2023-04-07 | 2024-10-10 | 中国医药研究开发中心有限公司 | 芳香杂环类化合物及其制备方法和医药用途 |
| CN121002017A (zh) * | 2023-05-04 | 2025-11-21 | 株式会社大熊制药 | 新颖的杂环胺衍生物以及包含其的药物组合物 |
| CN121263414A (zh) * | 2023-05-26 | 2026-01-02 | 上海艾力斯医药科技股份有限公司 | 杂芳环类化合物、其药物组合物及其应用 |
| CN121693505A (zh) * | 2023-11-17 | 2026-03-17 | 上海齐鲁制药研究中心有限公司 | 含氮杂芳基衍生物、其制备方法及其在医药上的应用 |
| WO2025149021A1 (zh) * | 2024-01-10 | 2025-07-17 | 海思科医药集团股份有限公司 | 一种吡啶并吡咯衍生物及其在医药上的应用 |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| TR199902301T2 (xx) * | 1997-03-19 | 1999-12-21 | Basf Aktiengesellschaft | Pirilo $2,3D]pirimidinler ve onlar�n kullan�m�. |
| GB0031080D0 (en) * | 2000-12-20 | 2001-01-31 | Novartis Ag | Organic compounds |
| US7232823B2 (en) * | 2003-06-09 | 2007-06-19 | Pfizer, Inc. | Cannabinoid receptor ligands and uses thereof |
| WO2005061504A1 (en) * | 2003-12-16 | 2005-07-07 | Pfizer Products Inc. | Bicyclic pyridazinone cannabinoid receptor ligands and uses thereof |
| DE102008052943A1 (de) * | 2008-10-23 | 2010-04-29 | Merck Patent Gmbh | Azaindolderivate |
| CN105837576B (zh) * | 2015-01-14 | 2019-03-26 | 湖北生物医药产业技术研究院有限公司 | Btk抑制剂 |
| CN107417687A (zh) * | 2016-05-24 | 2017-12-01 | 中国科学院上海药物研究所 | 五元杂环并[3,4‑d]哒嗪酮类化合物、其制备方法、药物组合物及其应用 |
| CN108997380A (zh) * | 2018-07-26 | 2018-12-14 | 长春海谱润斯科技有限公司 | 一种嘌呤化合物及其有机电致发光器件 |
| WO2020231990A1 (en) * | 2019-05-13 | 2020-11-19 | Relay Therapeutics, Inc. | Fgfr inhibitors and methods of use thereof |
-
2022
- 2022-09-23 KR KR1020247013425A patent/KR20240075952A/ko active Pending
- 2022-09-23 JP JP2024518772A patent/JP2024536858A/ja active Pending
- 2022-09-23 US US18/693,543 patent/US20240383905A1/en active Pending
- 2022-09-23 CA CA3231948A patent/CA3231948A1/en active Pending
- 2022-09-23 AU AU2022350571A patent/AU2022350571A1/en active Pending
- 2022-09-23 WO PCT/CN2022/121076 patent/WO2023046117A1/en not_active Ceased
- 2022-09-23 EP EP22872161.9A patent/EP4405358A4/en active Pending
- 2022-09-23 CN CN202280064436.XA patent/CN118043327A/zh active Pending
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