JP2021518379A5 - - Google Patents
Info
- Publication number
- JP2021518379A5 JP2021518379A5 JP2020550114A JP2020550114A JP2021518379A5 JP 2021518379 A5 JP2021518379 A5 JP 2021518379A5 JP 2020550114 A JP2020550114 A JP 2020550114A JP 2020550114 A JP2020550114 A JP 2020550114A JP 2021518379 A5 JP2021518379 A5 JP 2021518379A5
- Authority
- JP
- Japan
- Prior art keywords
- methyl
- pyrimidine
- pyrrolo
- azaspiro
- amino
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862646167P | 2018-03-21 | 2018-03-21 | |
| US62/646,167 | 2018-03-21 | ||
| PCT/US2019/022657 WO2019182924A1 (en) | 2018-03-21 | 2019-03-18 | Jak inhibitors |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2021518379A JP2021518379A (ja) | 2021-08-02 |
| JP2021518379A5 true JP2021518379A5 (https=) | 2022-03-30 |
| JP7462951B2 JP7462951B2 (ja) | 2024-04-08 |
Family
ID=67986579
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2020550114A Active JP7462951B2 (ja) | 2018-03-21 | 2019-03-18 | Ｊａｋ阻害剤 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US11365188B2 (https=) |
| EP (1) | EP3768272B1 (https=) |
| JP (1) | JP7462951B2 (https=) |
| CN (1) | CN111936144B (https=) |
| AU (1) | AU2019237991B2 (https=) |
| CA (1) | CA3093706A1 (https=) |
| WO (1) | WO2019182924A1 (https=) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX388576B (es) | 2016-06-07 | 2025-03-20 | Jacobio Pharmaceuticals Co Ltd | Derivados heterociclicos novedosos utiles como inhibidores de shp2. |
| EA202190196A1 (ru) | 2017-03-23 | 2021-08-31 | Джакобио Фармасьютикалс Ко., Лтд. | Новые гетероциклические производные, применимые в качестве ингибиторов shp2 |
| US20210393623A1 (en) | 2018-09-26 | 2021-12-23 | Jacobio Pharmaceuticals Co., Ltd. | Novel Heterocyclic Derivatives Useful as SHP2 Inhibitors |
| BR112021008742A2 (pt) * | 2018-11-05 | 2021-08-10 | Avista Pharma Solutions, Inc. | compostos químicos |
| CN113498352A (zh) | 2019-01-23 | 2021-10-12 | 施万生物制药研发Ip有限责任公司 | 作为jak抑制剂的咪唑并[1,5-a]吡啶、1,2,4-三唑并[4,3-a]吡啶和咪唑并[1,5-a]吡嗪 |
| MX2021008984A (es) | 2019-01-30 | 2021-09-08 | Felicamed Biotechnology Co Ltd | Inhibidor jak y metodo de preparacion del mismo. |
| WO2022117075A1 (zh) * | 2020-12-04 | 2022-06-09 | 广州费米子科技有限责任公司 | 氮杂并环化合物、其制备方法及其用途 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PT2796460T (pt) | 2011-12-21 | 2018-11-05 | Shanghai hengrui pharmaceutical co ltd | Derivado pirrole de anel heteroarilo de seis membros, método de preparação do mesmo e suas utilizações médicas |
| SI3077395T1 (en) * | 2013-12-05 | 2018-03-30 | Pfizer Inc. | Pyrrolo(2,3-d)pyrimidinyl, pyrrolo(2,3-b)pyrazinyl and pyrrolo(2,3-d)pyridinyl acrylamides |
| WO2015131080A1 (en) * | 2014-02-28 | 2015-09-03 | Nimbus Lakshmi, Inc. | Tyk2 inhibitors and uses thereof |
| WO2016024185A1 (en) * | 2014-08-12 | 2016-02-18 | Pfizer Inc. | Pyrrolo[2,3-d]pyrimidine derivatives useful for inhibiting janus kinase |
| EA036122B1 (ru) * | 2015-01-20 | 2020-09-30 | Уси Форчун Фармасьютикал Ко., Лтд | Ингибитор jak |
| WO2018169700A1 (en) * | 2017-03-14 | 2018-09-20 | Sunshine Lake Pharma Co., Ltd. | Substituted heteroaryl compounds and methods of use |
-
2019
- 2019-03-18 EP EP19770607.0A patent/EP3768272B1/en active Active
- 2019-03-18 WO PCT/US2019/022657 patent/WO2019182924A1/en not_active Ceased
- 2019-03-18 CA CA3093706A patent/CA3093706A1/en active Pending
- 2019-03-18 AU AU2019237991A patent/AU2019237991B2/en active Active
- 2019-03-18 CN CN201980020463.5A patent/CN111936144B/zh active Active
- 2019-03-18 JP JP2020550114A patent/JP7462951B2/ja active Active
- 2019-03-18 US US16/979,455 patent/US11365188B2/en active Active
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