JP2024518685A5 - - Google Patents

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Publication number
JP2024518685A5
JP2024518685A5 JP2023560623A JP2023560623A JP2024518685A5 JP 2024518685 A5 JP2024518685 A5 JP 2024518685A5 JP 2023560623 A JP2023560623 A JP 2023560623A JP 2023560623 A JP2023560623 A JP 2023560623A JP 2024518685 A5 JP2024518685 A5 JP 2024518685A5
Authority
JP
Japan
Prior art keywords
salt
cancer
compound
dose
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2023560623A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024518685A (ja
JP7839803B2 (ja
Filing date
Publication date
Priority claimed from GBGB2104416.9A external-priority patent/GB202104416D0/en
Priority claimed from GBGB2117511.2A external-priority patent/GB202117511D0/en
Application filed filed Critical
Priority claimed from PCT/EP2022/058283 external-priority patent/WO2022207646A1/en
Publication of JP2024518685A publication Critical patent/JP2024518685A/ja
Publication of JP2024518685A5 publication Critical patent/JP2024518685A5/ja
Application granted granted Critical
Publication of JP7839803B2 publication Critical patent/JP7839803B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2023560623A 2021-03-29 2022-03-29 治療レジメンで使用するためのpi3k-デルタ阻害剤 Active JP7839803B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GBGB2104416.9A GB202104416D0 (en) 2021-03-29 2021-03-29 Treatment reginmens
GB2104416.9 2021-03-29
GBGB2117511.2A GB202117511D0 (en) 2021-12-03 2021-12-03 Treatment regimens
GB2117511.2 2021-12-03
PCT/EP2022/058283 WO2022207646A1 (en) 2021-03-29 2022-03-29 A pi3k-delta inhibitor for use in treatment regimens

Publications (3)

Publication Number Publication Date
JP2024518685A JP2024518685A (ja) 2024-05-02
JP2024518685A5 true JP2024518685A5 (https=) 2025-04-04
JP7839803B2 JP7839803B2 (ja) 2026-04-02

Family

ID=81388915

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023560623A Active JP7839803B2 (ja) 2021-03-29 2022-03-29 治療レジメンで使用するためのpi3k-デルタ阻害剤

Country Status (17)

Country Link
US (1) US12605389B2 (https=)
EP (1) EP4313058B1 (https=)
JP (1) JP7839803B2 (https=)
AU (1) AU2022251843B2 (https=)
CA (1) CA3212731A1 (https=)
DK (1) DK4313058T3 (https=)
ES (1) ES3031295T3 (https=)
FI (1) FI4313058T3 (https=)
HR (1) HRP20250516T1 (https=)
HU (1) HUE071610T2 (https=)
LT (1) LT4313058T (https=)
MX (1) MX2023011442A (https=)
PL (1) PL4313058T3 (https=)
PT (1) PT4313058T (https=)
RS (1) RS66754B1 (https=)
SI (1) SI4313058T1 (https=)
WO (1) WO2022207646A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2026510567A (ja) * 2023-03-03 2026-04-08 アイオンクチュラ・ソシエテ・アノニム 血液悪性腫瘍の治療におけるロギノリシブ及びbcl-2阻害剤の組み合わせ
AU2024231699A1 (en) * 2023-03-03 2025-09-11 Ionctura Sa Combination of roginolisib and hdac inhibitor in the treatment of haematological malignancy

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EA201290305A1 (ru) 2009-11-13 2012-12-28 Мерк Сероно С.А. Производные трициклического пиразоламина
WO2014121901A1 (en) 2013-02-07 2014-08-14 Merck Patent Gmbh Polymorphic forms
US9986723B2 (en) 2014-10-22 2018-06-05 The Board Of Regents Of The University Of Texas System Screen and use of therapeutics for pancreatic ductal adenocarcinoma
GB201502020D0 (en) 2015-02-06 2015-03-25 Cancer Rec Tech Ltd Autotaxin inhibitory compounds
EP3610264A1 (en) 2017-04-13 2020-02-19 INSERM (Institut National de la Santé et de la Recherche Médicale) Methods for the diagnosis and treatment of pancreatic ductal adenocarcinoma

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