JP2024516826A5 - - Google Patents

Info

Publication number
JP2024516826A5
JP2024516826A5 JP2023566480A JP2023566480A JP2024516826A5 JP 2024516826 A5 JP2024516826 A5 JP 2024516826A5 JP 2023566480 A JP2023566480 A JP 2023566480A JP 2023566480 A JP2023566480 A JP 2023566480A JP 2024516826 A5 JP2024516826 A5 JP 2024516826A5
Authority
JP
Japan
Prior art keywords
oxazepan
carboxamide
ethyl
cyano
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023566480A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024516826A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2022/027026 external-priority patent/WO2022232573A1/en
Publication of JP2024516826A publication Critical patent/JP2024516826A/ja
Publication of JP2024516826A5 publication Critical patent/JP2024516826A5/ja
Pending legal-status Critical Current

Links

JP2023566480A 2021-04-29 2022-04-29 嚢胞性線維症を治療するためのある特定のn-(1-シアノ-2-フェニルエチル)-1,4-オキサゼパン-2-カルボキサミド Pending JP2024516826A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202163181817P 2021-04-29 2021-04-29
US63/181,817 2021-04-29
PCT/US2022/027026 WO2022232573A1 (en) 2021-04-29 2022-04-29 Certain n-(1-cyano-2-phenylethyl)-1,4-oxazepane-2-carboxamides for treating cystic fibrosis

Publications (2)

Publication Number Publication Date
JP2024516826A JP2024516826A (ja) 2024-04-17
JP2024516826A5 true JP2024516826A5 (https=) 2025-05-09

Family

ID=83848696

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023566480A Pending JP2024516826A (ja) 2021-04-29 2022-04-29 嚢胞性線維症を治療するためのある特定のn-(1-シアノ-2-フェニルエチル)-1,4-オキサゼパン-2-カルボキサミド

Country Status (6)

Country Link
US (1) US20240226112A1 (https=)
EP (1) EP4329767A4 (https=)
JP (1) JP2024516826A (https=)
KR (1) KR20240004691A (https=)
CA (1) CA3215375A1 (https=)
WO (1) WO2022232573A1 (https=)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NO2699580T3 (https=) 2014-01-24 2018-02-24
HUE070049T2 (hu) 2018-03-01 2025-05-28 Astrazeneca Ab (2S)-{(1S)-1-ciano-2-[4-(3-metil-2-oxo-2,3-dihidro-1,3-benzoxazol-5-il)fenil]etil} -1,4-oxazepán-2-karboxamidot tartalmazó gyógyászati készítmények
WO2020018547A1 (en) 2018-07-17 2020-01-23 Insmed Incorporated Certain (2s)-n-[(1s)-1-cyano-2-phenylethyl]-1,4-oxazepane-2-carboxamides for treating lupus nephritis
JP2026503035A (ja) * 2023-01-06 2026-01-27 インスメッド インコーポレイテッド 新規な可逆性dpp1阻害剤及びその用途
JP2026510407A (ja) * 2023-03-23 2026-04-02 ハイスコ ファーマスーティカル プライベート リミテッド ジペプチジルペプチダーゼ小分子阻害剤を含む医薬組成物

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004076434A1 (en) * 2003-02-28 2004-09-10 Aic Dipeptidyl peptidase inhibitors
ES2845473T3 (es) * 2013-03-14 2021-07-26 Boehringer Ingelheim Int (Bencil-ciano-metil)-amidas sustituidas de ácido 2-aza-biciclo[2.2.1]heptano-3-carboxílico inhibidores de la catepsina- C
NO2699580T3 (https=) * 2014-01-24 2018-02-24
JP6783426B2 (ja) * 2015-03-05 2020-11-11 ニュープロザイム・セラピューティクス・アンパルトセルスカブNeuprozyme Therapeutics ApS ジペプチジルペプチダーゼi阻害剤としてのペプチジルニトリル化合物
KR20240091302A (ko) * 2016-07-29 2024-06-21 인스메드 인코포레이티드 기관지확장증을 치료하기 위한 특정 (2s)-n-[(1s)-1-시아노-2-페닐에틸]-1,4-옥사제판-2-카르복스아미드
HUE070049T2 (hu) * 2018-03-01 2025-05-28 Astrazeneca Ab (2S)-{(1S)-1-ciano-2-[4-(3-metil-2-oxo-2,3-dihidro-1,3-benzoxazol-5-il)fenil]etil} -1,4-oxazepán-2-karboxamidot tartalmazó gyógyászati készítmények

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