JP2021530513A5 - - Google Patents
Info
- Publication number
- JP2021530513A5 JP2021530513A5 JP2021502436A JP2021502436A JP2021530513A5 JP 2021530513 A5 JP2021530513 A5 JP 2021530513A5 JP 2021502436 A JP2021502436 A JP 2021502436A JP 2021502436 A JP2021502436 A JP 2021502436A JP 2021530513 A5 JP2021530513 A5 JP 2021530513A5
- Authority
- JP
- Japan
- Prior art keywords
- oxazepan
- carboxamide
- ethyl
- cyano
- phenyl
- Prior art date
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201862699491P | 2018-07-17 | 2018-07-17 | |
| US62/699,491 | 2018-07-17 | ||
| PCT/US2019/042026 WO2020018551A1 (en) | 2018-07-17 | 2019-07-16 | Certain (2s)- n-[(1s)-1-cyano-2-phenylethyl]-1,4- oxazepane-2-carboxamides for treating inflammatory bowel disease |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2021530513A JP2021530513A (ja) | 2021-11-11 |
| JPWO2020018551A5 JPWO2020018551A5 (https=) | 2022-07-21 |
| JP2021530513A5 true JP2021530513A5 (https=) | 2022-07-21 |
Family
ID=69163563
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2021502436A Pending JP2021530513A (ja) | 2018-07-17 | 2019-07-16 | 炎症性腸疾患を処置するための特定の（２ｓ）−ｎ−［（１ｓ）−１−シアノ−２−フェニルエチル］−１，４−オキサゼパン−２−カルボキサミド |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US20210252015A1 (https=) |
| EP (1) | EP3823628A4 (https=) |
| JP (1) | JP2021530513A (https=) |
| KR (1) | KR20210032439A (https=) |
| AU (1) | AU2019305565A1 (https=) |
| CA (1) | CA3106270A1 (https=) |
| WO (1) | WO2020018551A1 (https=) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NO2699580T3 (https=) | 2014-01-24 | 2018-02-24 | ||
| KR20250002710A (ko) | 2018-03-01 | 2025-01-07 | 아스트라제네카 에이비이 | (2s)-n-｛(1s)-1-시아노-2-[4-(3-메틸-2-옥소-2,3-디하이드로-1,3-벤족사졸-5-일)페닐]에틸｝-1,4-옥사제판-2-카복스아미드를포함하는 약학 조성물 |
| AU2019306532A1 (en) | 2018-07-17 | 2021-03-04 | Insmed Incorporated | Certain (2S)-N-[(1S)-1-cyano-2-phenylethyl]-1,4-oxazepane-2-carboxamides for treating Lupus Nephritis |
| CN114106005B (zh) * | 2020-08-26 | 2025-08-01 | 西藏海思科制药有限公司 | 一种作为二肽基肽酶1抑制剂的腈衍生物及其用途 |
| WO2022140516A1 (en) * | 2020-12-22 | 2022-06-30 | Insmed Incorporated | Certain (25)-iv-[(ls')~ i-c yan0-2-phenylethyl·]- 1,4-oxazepane-2- carboxamides for treating behcet's disease |
| US20240150335A1 (en) * | 2021-02-05 | 2024-05-09 | Medshine Discovery Inc. | Fused ring derivatives containing 1,4-oxazepane |
| EP4450497A4 (en) * | 2022-01-11 | 2025-11-26 | Shanghai Yidian Pharmaceutical Tech Development Co Ltd | NITRILE PEPTIDYL COMPOUND AND ITS USES |
| CN119156384B (zh) * | 2022-06-07 | 2025-12-09 | 瑞石生物医药有限公司 | 苯并[c]色满化合物的多晶型及其制备方法和用途 |
| EP4646265A1 (en) | 2023-01-06 | 2025-11-12 | Insmed Incorporated | Novel, reversible dpp1 inhibitors and uses thereof |
| JP2026510867A (ja) * | 2023-03-16 | 2026-04-10 | インスメッド インコーポレイテッド | 多環式リンカーを有するｄｐｐ１阻害剤およびその使用 |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20110236367A1 (en) * | 2000-09-08 | 2011-09-29 | Telenav, Inc. | Rat cathespin dipeptidyl peptidase i (dppi): crystal structure and its uses |
| ATE399763T1 (de) * | 2003-05-30 | 2008-07-15 | Prozymex As | Proteasehemmer |
| EP2017620A3 (en) * | 2004-04-28 | 2009-04-22 | Bayer HealthCare AG | Diagnostics and therapeutics for diseases associated with dipeptidyl-peptidase 1 (DPP1) |
| CN102574830A (zh) * | 2009-05-07 | 2012-07-11 | 阿斯利康(瑞典)有限公司 | 取代的1-氰基乙基杂环基甲酰胺化合物750 |
| NO2699580T3 (https=) * | 2014-01-24 | 2018-02-24 | ||
| KR20250107292A (ko) * | 2016-07-29 | 2025-07-11 | 인스메드 인코포레이티드 | 기관지확장증을 치료하기 위한 특정 (2s)-n-[(1s)-1-시아노-2-페닐에틸]-1,4-옥사제판-2-카르복스아미드 |
| AU2019217870A1 (en) * | 2018-02-07 | 2020-08-27 | Insmed Incorporated | Certain (2S)-N-[(1S)-1-cyano-2-phenylethyl]-1,4-oxazepane-2-carboxamides for treating ANCA associated vasculitides |
-
2019
- 2019-07-16 US US17/260,602 patent/US20210252015A1/en not_active Abandoned
- 2019-07-16 JP JP2021502436A patent/JP2021530513A/ja active Pending
- 2019-07-16 AU AU2019305565A patent/AU2019305565A1/en not_active Abandoned
- 2019-07-16 EP EP19838400.0A patent/EP3823628A4/en not_active Withdrawn
- 2019-07-16 KR KR1020217004189A patent/KR20210032439A/ko not_active Ceased
- 2019-07-16 CA CA3106270A patent/CA3106270A1/en active Pending
- 2019-07-16 WO PCT/US2019/042026 patent/WO2020018551A1/en not_active Ceased
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