JP2021530513A5 - - Google Patents

Info

Publication number
JP2021530513A5
JP2021530513A5 JP2021502436A JP2021502436A JP2021530513A5 JP 2021530513 A5 JP2021530513 A5 JP 2021530513A5 JP 2021502436 A JP2021502436 A JP 2021502436A JP 2021502436 A JP2021502436 A JP 2021502436A JP 2021530513 A5 JP2021530513 A5 JP 2021530513A5
Authority
JP
Japan
Prior art keywords
oxazepan
carboxamide
ethyl
cyano
phenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2021502436A
Other languages
English (en)
Japanese (ja)
Other versions
JP2021530513A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2019/042026 external-priority patent/WO2020018551A1/en
Publication of JP2021530513A publication Critical patent/JP2021530513A/ja
Publication of JP2021530513A5 publication Critical patent/JP2021530513A5/ja
Pending legal-status Critical Current

Links

JP2021502436A 2018-07-17 2019-07-16 炎症性腸疾患を処置するための特定の(2s)−n−[(1s)−1−シアノ−2−フェニルエチル]−1,4−オキサゼパン−2−カルボキサミド Pending JP2021530513A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201862699491P 2018-07-17 2018-07-17
US62/699,491 2018-07-17
PCT/US2019/042026 WO2020018551A1 (en) 2018-07-17 2019-07-16 Certain (2s)- n-[(1s)-1-cyano-2-phenylethyl]-1,4- oxazepane-2-carboxamides for treating inflammatory bowel disease

Publications (2)

Publication Number Publication Date
JP2021530513A JP2021530513A (ja) 2021-11-11
JP2021530513A5 true JP2021530513A5 (https=) 2022-07-21

Family

ID=69163563

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2021502436A Pending JP2021530513A (ja) 2018-07-17 2019-07-16 炎症性腸疾患を処置するための特定の(2s)−n−[(1s)−1−シアノ−2−フェニルエチル]−1,4−オキサゼパン−2−カルボキサミド

Country Status (7)

Country Link
US (1) US20210252015A1 (https=)
EP (1) EP3823628A4 (https=)
JP (1) JP2021530513A (https=)
KR (1) KR20210032439A (https=)
AU (1) AU2019305565A1 (https=)
CA (1) CA3106270A1 (https=)
WO (1) WO2020018551A1 (https=)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NO2699580T3 (https=) 2014-01-24 2018-02-24
HUE070049T2 (hu) 2018-03-01 2025-05-28 Astrazeneca Ab (2S)-{(1S)-1-ciano-2-[4-(3-metil-2-oxo-2,3-dihidro-1,3-benzoxazol-5-il)fenil]etil} -1,4-oxazepán-2-karboxamidot tartalmazó gyógyászati készítmények
WO2020018547A1 (en) 2018-07-17 2020-01-23 Insmed Incorporated Certain (2s)-n-[(1s)-1-cyano-2-phenylethyl]-1,4-oxazepane-2-carboxamides for treating lupus nephritis
CN114106005B (zh) * 2020-08-26 2025-08-01 西藏海思科制药有限公司 一种作为二肽基肽酶1抑制剂的腈衍生物及其用途
WO2022140516A1 (en) * 2020-12-22 2022-06-30 Insmed Incorporated Certain (25)-iv-[(ls')~ i-c yan0-2-phenylethyl·]- 1,4-oxazepane-2- carboxamides for treating behcet's disease
US20240150335A1 (en) * 2021-02-05 2024-05-09 Medshine Discovery Inc. Fused ring derivatives containing 1,4-oxazepane
EP4450497A4 (en) * 2022-01-11 2025-11-26 Shanghai Yidian Pharmaceutical Tech Development Co Ltd NITRILE PEPTIDYL COMPOUND AND ITS USES
EP4538271A4 (en) * 2022-06-07 2025-10-08 Reistone Biopharma Company Ltd POLYMORPH OF BENZO[C]CHROMANE COMPOUND, ITS PREPARATION METHOD AND ITS USE
JP2026503035A (ja) 2023-01-06 2026-01-27 インスメッド インコーポレイテッド 新規な可逆性dpp1阻害剤及びその用途
KR20250170710A (ko) * 2023-03-16 2025-12-05 인스메드 인코포레이티드 폴리사이클릭 링커를 갖는 dpp1 억제제 및 이의 용도

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20110236367A1 (en) * 2000-09-08 2011-09-29 Telenav, Inc. Rat cathespin dipeptidyl peptidase i (dppi): crystal structure and its uses
EP1633702B1 (en) * 2003-05-30 2008-07-02 Prozymex A/S Protease inhibitors
EP1745292A2 (en) * 2004-04-28 2007-01-24 Bayer HealthCare AG Diagnostics and therapeutics for diseases associated with dipeptidyl-peptidase 1 (dpp1)
MX2011011661A (es) * 2009-05-07 2011-11-18 Astrazeneca Ab Compuestos 1-cianoetilheterociclilcarboxamida sustituidos 750.
NO2699580T3 (https=) * 2014-01-24 2018-02-24
KR20240091302A (ko) * 2016-07-29 2024-06-21 인스메드 인코포레이티드 기관지확장증을 치료하기 위한 특정 (2s)-n-[(1s)-1-시아노-2-페닐에틸]-1,4-옥사제판-2-카르복스아미드
CA3089240A1 (en) * 2018-02-07 2019-08-15 Insmed Incorporated Certain (2s)-n-[(1s)-1-cyano-2-phenylethyl]-1,4-oxazepane-2-carboxamides for treating anca associated vasculitides

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