JP2022541311A5 - - Google Patents

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Publication number
JP2022541311A5
JP2022541311A5 JP2022504089A JP2022504089A JP2022541311A5 JP 2022541311 A5 JP2022541311 A5 JP 2022541311A5 JP 2022504089 A JP2022504089 A JP 2022504089A JP 2022504089 A JP2022504089 A JP 2022504089A JP 2022541311 A5 JP2022541311 A5 JP 2022541311A5
Authority
JP
Japan
Application number
JP2022504089A
Other languages
Japanese (ja)
Other versions
JP7583022B2 (ja
JP2022541311A (ja
JPWO2021014166A5 (https=
Filing date
Publication date
Priority claimed from GBGB1910607.9A external-priority patent/GB201910607D0/en
Priority claimed from GBGB2005739.4A external-priority patent/GB202005739D0/en
Application filed filed Critical
Priority claimed from PCT/GB2020/051778 external-priority patent/WO2021014166A1/en
Publication of JP2022541311A publication Critical patent/JP2022541311A/ja
Publication of JP2022541311A5 publication Critical patent/JP2022541311A5/ja
Publication of JPWO2021014166A5 publication Critical patent/JPWO2021014166A5/ja
Application granted granted Critical
Publication of JP7583022B2 publication Critical patent/JP7583022B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2022504089A 2019-07-24 2020-07-24 呼吸器症状の治療における使用のためのtmem16aモジュレータとしてのピリジン誘導体 Active JP7583022B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GB1910607.9 2019-07-24
GBGB1910607.9A GB201910607D0 (en) 2019-07-24 2019-07-24 Compounds
GB2005739.4 2020-04-20
GBGB2005739.4A GB202005739D0 (en) 2020-04-20 2020-04-20 Compounds
PCT/GB2020/051778 WO2021014166A1 (en) 2019-07-24 2020-07-24 Pyridine derivatives as tmem16a modulators for use in the treatment of respiratory conditions

Publications (4)

Publication Number Publication Date
JP2022541311A JP2022541311A (ja) 2022-09-22
JP2022541311A5 true JP2022541311A5 (https=) 2023-07-25
JPWO2021014166A5 JPWO2021014166A5 (https=) 2023-07-25
JP7583022B2 JP7583022B2 (ja) 2024-11-13

Family

ID=71948615

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2022504089A Active JP7583022B2 (ja) 2019-07-24 2020-07-24 呼吸器症状の治療における使用のためのtmem16aモジュレータとしてのピリジン誘導体

Country Status (16)

Country Link
US (1) US20220235006A1 (https=)
EP (1) EP4003516A1 (https=)
JP (1) JP7583022B2 (https=)
KR (1) KR20220063162A (https=)
CN (1) CN114616226B (https=)
AU (1) AU2020317036A1 (https=)
BR (1) BR112022001164A2 (https=)
CA (1) CA3145120A1 (https=)
CL (1) CL2022000147A1 (https=)
CO (1) CO2022002022A2 (https=)
CR (1) CR20220072A (https=)
IL (1) IL290035A (https=)
MX (1) MX2022000841A (https=)
PE (1) PE20221441A1 (https=)
PH (1) PH12022550181A1 (https=)
WO (1) WO2021014166A1 (https=)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PE20221441A1 (es) * 2019-07-24 2022-09-21 Tmem16A Ltd Derivados de piridina como moduladores de tmem16a para su uso en el tratamiento de afecciones respiratorias
WO2026038890A1 (ko) * 2024-08-13 2026-02-19 광주과학기술원 신규한 치환된 피리딘 유도체 화합물, 이의 제조방법, 및 이를 유효성분으로 포함하는 호흡기 질환의 예방 또는 치료용 약학적 조성물

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20050176767A1 (en) 2003-10-30 2005-08-11 Laval Chan Chun Kong Pyridine carboxamide and methods for inhibiting HIV integrase
US11358947B2 (en) * 2017-04-17 2022-06-14 The Regents Of The University Of California Substituted 2-acylamino-cycloalkylthiophene-3-carboxylic acid arylamides as inhibitors of calcium-activated chloride channel TMEM16A
GB201801355D0 (en) * 2018-01-26 2018-03-14 Enterprise Therapeutics Ltd Compounds
PE20221441A1 (es) * 2019-07-24 2022-09-21 Tmem16A Ltd Derivados de piridina como moduladores de tmem16a para su uso en el tratamiento de afecciones respiratorias

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