JP2024509981A5 - - Google Patents
Info
- Publication number
- JP2024509981A5 JP2024509981A5 JP2023556474A JP2023556474A JP2024509981A5 JP 2024509981 A5 JP2024509981 A5 JP 2024509981A5 JP 2023556474 A JP2023556474 A JP 2023556474A JP 2023556474 A JP2023556474 A JP 2023556474A JP 2024509981 A5 JP2024509981 A5 JP 2024509981A5
- Authority
- JP
- Japan
- Prior art keywords
- alkyl
- membered
- pharmaceutically acceptable
- hydrogen
- tautomer
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| JP2025056015A JP2025106341A (ja) | 2021-03-15 | 2025-03-28 | ピラゾロピリジン誘導体及びその使用 |
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US202163161139P | 2021-03-15 | 2021-03-15 | |
| US63/161,139 | 2021-03-15 | ||
| US202163164130P | 2021-03-22 | 2021-03-22 | |
| US63/164,130 | 2021-03-22 | ||
| PCT/IB2022/052281 WO2022195454A1 (en) | 2021-03-15 | 2022-03-14 | Pyrazolopyridine derivatives and uses thereof |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025056015A Division JP2025106341A (ja) | 2021-03-15 | 2025-03-28 | ピラゾロピリジン誘導体及びその使用 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| JP2024509981A JP2024509981A (ja) | 2024-03-05 |
| JP2024509981A5 true JP2024509981A5 (https=) | 2024-03-28 |
| JP7659648B2 JP7659648B2 (ja) | 2025-04-09 |
Family
ID=80819999
Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023556474A Active JP7659648B2 (ja) | 2021-03-15 | 2022-03-14 | ピラゾロピリジン誘導体及びその使用 |
| JP2025056015A Pending JP2025106341A (ja) | 2021-03-15 | 2025-03-28 | ピラゾロピリジン誘導体及びその使用 |
Family Applications After (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2025056015A Pending JP2025106341A (ja) | 2021-03-15 | 2025-03-28 | ピラゾロピリジン誘導体及びその使用 |
Country Status (19)
| Country | Link |
|---|---|
| US (4) | US11787785B2 (https=) |
| EP (1) | EP4308562A1 (https=) |
| JP (2) | JP7659648B2 (https=) |
| KR (1) | KR102902295B1 (https=) |
| AU (2) | AU2022239950B2 (https=) |
| CA (1) | CA3208951A1 (https=) |
| CL (1) | CL2023002726A1 (https=) |
| CO (1) | CO2023013486A2 (https=) |
| CR (1) | CR20230486A (https=) |
| DO (1) | DOP2023000188A (https=) |
| EC (1) | ECSP23076800A (https=) |
| IL (1) | IL305931A (https=) |
| JO (1) | JOP20230218A1 (https=) |
| MX (1) | MX2023010827A (https=) |
| PE (1) | PE20242203A1 (https=) |
| PY (1) | PY2217419A (https=) |
| UY (1) | UY39671A (https=) |
| WO (1) | WO2022195454A1 (https=) |
| ZA (1) | ZA202307290B (https=) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PY2217419A (es) | 2021-03-15 | 2022-09-27 | Novartis Ag | Derivados de pirazolopiridina y sus usos |
| WO2022195355A1 (en) * | 2021-03-15 | 2022-09-22 | Novartis Ag | Benzisoxazole derivatives and uses thereof |
| EP4612128A4 (en) | 2022-11-04 | 2025-09-10 | Bristol Myers Squibb Co | COMPOUNDS AND THEIR USE FOR THE TREATMENT OF HEMOGLOBINOPATHIES |
| WO2024255810A1 (en) * | 2023-06-15 | 2024-12-19 | Hangzhou Glubio Pharmaceutical Co., Ltd | Dihydropyrimidine-2, 4 (1h, 3h) -dione-containing polycyclic derivatives and pharmaceutical composition thereof, preparation method thereof and use thereof |
Family Cites Families (19)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2007524596A (ja) | 2003-02-28 | 2007-08-30 | トランスフォーム・ファーマシューティカルズ・インコーポレイテッド | 共結晶医薬組成物 |
| KR20060109979A (ko) | 2003-12-02 | 2006-10-23 | 셀진 코포레이션 | 혈색소병증 및 빈혈의 치료 및 관리를 위한 방법및 조성물 |
| EP1604988A1 (en) | 2004-05-18 | 2005-12-14 | Sanofi-Aventis Deutschland GmbH | Pyridazinone derivatives, methods for producing them and their use as pharmaceuticals |
| KR101608259B1 (ko) | 2008-04-28 | 2016-04-01 | 교린 세이야꾸 가부시키 가이샤 | 시클로펜틸아크릴산아미드 유도체 |
| EP2165707A1 (en) | 2008-09-23 | 2010-03-24 | Genkyo Tex Sa | Pyrazolo pyridine derivatives as NADPH oxidase inhibitors |
| PL3202460T3 (pl) * | 2010-02-11 | 2019-12-31 | Celgene Corporation | Pochodne arylometoksyizoindoliny i zawierające je kompozycje oraz sposoby ich zastosowania |
| CN104619709B (zh) | 2012-07-13 | 2016-11-09 | Ucb生物制药私人有限公司 | 作为tnf活性调节剂的咪唑并吡啶衍生物 |
| US9845308B2 (en) | 2014-11-05 | 2017-12-19 | Vitae Pharmaceuticals, Inc. | Isoindoline inhibitors of ROR-gamma |
| TWI793151B (zh) * | 2017-08-23 | 2023-02-21 | 瑞士商諾華公司 | 3-(1-氧異吲哚啉-2-基)之氫吡啶-2,6-二酮衍生物及其用途 |
| WO2019140387A1 (en) | 2018-01-12 | 2019-07-18 | Kymera Therapeutics, Inc. | Crbn ligands and uses thereof |
| JP2020009513A (ja) * | 2018-07-10 | 2020-01-16 | キオクシア株式会社 | メモリシステム |
| AR116109A1 (es) * | 2018-07-10 | 2021-03-31 | Novartis Ag | Derivados de 3-(5-amino-1-oxoisoindolin-2-il)piperidina-2,6-diona y usos de los mismos |
| CN120698983A (zh) | 2018-12-20 | 2025-09-26 | C4医药公司 | 靶向蛋白降解 |
| CN120574283A (zh) | 2019-04-05 | 2025-09-02 | 凯麦拉医疗公司 | Stat降解剂和其用途 |
| EP3969458A4 (en) | 2019-05-13 | 2023-05-17 | Borah, Inc. | CHEMICAL COMPOUNDS |
| PH12022551482A1 (en) | 2019-12-18 | 2023-11-29 | Novartis Ag | 3-(5-methoxy-1-oxoisoindolin-2-yl)piperidine-2,6-dione derivatives and uses thereof |
| KR20220138399A (ko) | 2020-02-04 | 2022-10-12 | 스팅레이 테라퓨릭스, 인크. | 엑토뉴클레오티드 피로포스파타제/포스포디에스테라제 1(enpp1)의 억제제 및 이의 사용 방법 |
| US20230089530A1 (en) | 2020-02-09 | 2023-03-23 | Newave Pharmaceutical Inc. | Quinuclidinone analogues as anticancer agents |
| PY2217419A (es) | 2021-03-15 | 2022-09-27 | Novartis Ag | Derivados de pirazolopiridina y sus usos |
-
2022
- 2022-03-11 PY PY202202217419A patent/PY2217419A/es unknown
- 2022-03-11 UY UY0001039671A patent/UY39671A/es unknown
- 2022-03-14 CR CR20230486A patent/CR20230486A/es unknown
- 2022-03-14 KR KR1020237034868A patent/KR102902295B1/ko active Active
- 2022-03-14 CA CA3208951A patent/CA3208951A1/en active Pending
- 2022-03-14 JP JP2023556474A patent/JP7659648B2/ja active Active
- 2022-03-14 IL IL305931A patent/IL305931A/en unknown
- 2022-03-14 AU AU2022239950A patent/AU2022239950B2/en active Active
- 2022-03-14 WO PCT/IB2022/052281 patent/WO2022195454A1/en not_active Ceased
- 2022-03-14 MX MX2023010827A patent/MX2023010827A/es unknown
- 2022-03-14 PE PE2023002595A patent/PE20242203A1/es unknown
- 2022-03-14 US US17/693,759 patent/US11787785B2/en active Active
- 2022-03-14 EP EP22711643.1A patent/EP4308562A1/en active Pending
-
2023
- 2023-07-21 ZA ZA2023/07290A patent/ZA202307290B/en unknown
- 2023-09-01 US US18/460,428 patent/US12172984B2/en active Active
- 2023-09-13 DO DO2023000188A patent/DOP2023000188A/es unknown
- 2023-09-13 CL CL2023002726A patent/CL2023002726A1/es unknown
- 2023-09-14 JO JOJO/P/2023/0218A patent/JOP20230218A1/ar unknown
- 2023-10-12 CO CONC2023/0013486A patent/CO2023013486A2/es unknown
- 2023-10-12 EC ECSENADI202376800A patent/ECSP23076800A/es unknown
-
2024
- 2024-09-06 US US18/826,887 patent/US12252482B2/en active Active
- 2024-11-06 US US18/939,314 patent/US20250282762A1/en active Pending
- 2024-12-09 AU AU2024278210A patent/AU2024278210B2/en active Active
-
2025
- 2025-03-28 JP JP2025056015A patent/JP2025106341A/ja active Pending
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