JP2024514338A - 複素環式誘導体阻害剤及びその調製方法及びその用途 - Google Patents

複素環式誘導体阻害剤及びその調製方法及びその用途 Download PDF

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JP2024514338A
JP2024514338A JP2023564007A JP2023564007A JP2024514338A JP 2024514338 A JP2024514338 A JP 2024514338A JP 2023564007 A JP2023564007 A JP 2023564007A JP 2023564007 A JP2023564007 A JP 2023564007A JP 2024514338 A JP2024514338 A JP 2024514338A
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amino
cycloalkyl
alkoxy
haloalkyl
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JPWO2022223025A5 (https=
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▲鵬▼ 高
蜜 曾
少宝 王
文▲勝▼ ▲兪▼
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Jiangsu Hansoh Pharmaceutical Group Co Ltd
Shanghai Hansoh Biomedical Co Ltd
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Jiangsu Hansoh Pharmaceutical Group Co Ltd
Shanghai Hansoh Biomedical Co Ltd
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JP2023564007A 2021-04-23 2022-04-22 複素環式誘導体阻害剤及びその調製方法及びその用途 Pending JP2024514338A (ja)

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CN202110443582.0 2021-04-23
CN202110443582 2021-04-23
CN202110653169.7 2021-06-11
CN202110653169 2021-06-11
CN202110808316.3 2021-07-16
CN202110808316 2021-07-16
CN202110926676.3 2021-08-12
CN202110926676 2021-08-12
CN202210072358 2022-01-21
CN202210072358.X 2022-01-21
PCT/CN2022/088466 WO2022223025A1 (zh) 2021-04-23 2022-04-22 杂环类衍生物抑制剂、其制备方法和应用

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CN (2) CN115232154A (https=)
AU (1) AU2022261029A1 (https=)
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JP2025502373A (ja) * 2022-01-27 2025-01-24 シンセラ, インコーポレイテッド Parp1阻害薬及びその使用

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TW202309025A (zh) 2021-04-19 2023-03-01 美商辛瑟拉股份有限公司 Parp1抑制劑及其用途
WO2022222965A1 (zh) * 2021-04-23 2022-10-27 成都百裕制药股份有限公司 吡啶衍生物及其在医药上的应用
US20230159525A1 (en) 2021-10-01 2023-05-25 Xinthera, Inc. Azetidine and pyrrolidine parp1 inhibitors and uses thereof
JP7762306B2 (ja) * 2021-11-19 2025-10-29 康百達(四川)生物医薬科技有限公司 選択的parp1阻害剤およびその用途
CN116143776A (zh) * 2021-11-22 2023-05-23 南京圣和药业股份有限公司 Parp1抑制剂及其应用
CA3241338A1 (en) * 2021-12-17 2023-06-22 Yongqi Deng Parp inhibitor, pharmaceutical composition comprising same, and use thereof
WO2023138541A1 (zh) * 2022-01-20 2023-07-27 微境生物医药科技(上海)有限公司 吡啶酰胺类parp抑制剂、及其制备方法和医药用途
AU2023209820B2 (en) 2022-01-21 2024-10-10 Xinthera, Inc. Parp1 inhibitors and uses thereof
KR20240161147A (ko) 2022-03-14 2024-11-12 슬랩 파마슈티컬스 엘엘씨 다중 사이클릭 화합물
FI4497438T3 (fi) 2022-04-28 2025-10-20 Xinthera Inc Trisyklisiä parp1:n estäjiä ja niiden käyttötapoja
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