JP2024510778A5 - - Google Patents

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Publication number
JP2024510778A5
JP2024510778A5 JP2023558324A JP2023558324A JP2024510778A5 JP 2024510778 A5 JP2024510778 A5 JP 2024510778A5 JP 2023558324 A JP2023558324 A JP 2023558324A JP 2023558324 A JP2023558324 A JP 2023558324A JP 2024510778 A5 JP2024510778 A5 JP 2024510778A5
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JP
Japan
Prior art keywords
independently selected
alkyl
corneal
pharmaceutically acceptable
acceptable salt
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Application number
JP2023558324A
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English (en)
Japanese (ja)
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JP7887908B2 (ja
JP2024510778A (ja
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Application filed filed Critical
Priority claimed from PCT/IB2022/052720 external-priority patent/WO2022201097A1/en
Publication of JP2024510778A publication Critical patent/JP2024510778A/ja
Publication of JP2024510778A5 publication Critical patent/JP2024510778A5/ja
Application granted granted Critical
Publication of JP7887908B2 publication Critical patent/JP7887908B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

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JP2023558324A 2021-03-26 2022-03-24 1,3-置換シクロブチル誘導体及びその使用 Active JP7887908B2 (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202163166289P 2021-03-26 2021-03-26
US63/166,289 2021-03-26
PCT/IB2022/052720 WO2022201097A1 (en) 2021-03-26 2022-03-24 1,3-substituted cyclobutyl derivatives and uses thereof

Publications (3)

Publication Number Publication Date
JP2024510778A JP2024510778A (ja) 2024-03-11
JP2024510778A5 true JP2024510778A5 (enExample) 2026-05-19
JP7887908B2 JP7887908B2 (ja) 2026-07-10

Family

ID=80999265

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023558324A Active JP7887908B2 (ja) 2021-03-26 2022-03-24 1,3-置換シクロブチル誘導体及びその使用

Country Status (14)

Country Link
US (2) US11845730B2 (enExample)
EP (1) EP4313951A1 (enExample)
JP (1) JP7887908B2 (enExample)
KR (1) KR20230162660A (enExample)
CN (1) CN117062804A (enExample)
AR (1) AR125196A1 (enExample)
AU (1) AU2022244467A1 (enExample)
CA (1) CA3214066A1 (enExample)
IL (1) IL307189B1 (enExample)
MX (1) MX2023011377A (enExample)
PY (1) PY2221203A (enExample)
TW (1) TWI924820B (enExample)
UY (1) UY39681A (enExample)
WO (1) WO2022201097A1 (enExample)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AR125196A1 (es) * 2021-03-26 2023-06-21 Novartis Ag Derivados de ciclobutilo 1,3-sustituidos y sus usos
JP2025531367A (ja) * 2022-09-21 2025-09-19 ボシュ + ロム アイルランド リミテッド Trpv1アンタゴニストの結晶多形形態およびその製剤
US20240148709A1 (en) * 2022-11-08 2024-05-09 Aisa Pharma, Inc. Methods of treating eye pain and eye disorders

Family Cites Families (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2004078163A2 (en) 2003-02-28 2004-09-16 Transform Pharmaceuticals, Inc. Pharmaceutical co-crystal compositions of drugs such as carbamazepine, celecoxib, olanzapine, itraconazole, topiramate, modafinil, 5-fluorouracil, hydrochlorothiazide, acetaminophen, aspirin, flurbiprofen, phenytoin and ibuprofen
US6933311B2 (en) 2003-02-11 2005-08-23 Abbott Laboratories Fused azabicyclic compounds that inhibit vanilloid receptor subtype 1 (VR1) receptor
US7514562B2 (en) 2003-03-07 2009-04-07 Glaxo Group Limited Urea derivatives and their use as vanilloid receptor antagonists in the treatment of pain
GB0412769D0 (en) 2004-06-08 2004-07-07 Novartis Ag Organic compounds
RU2451014C2 (ru) 2005-07-22 2012-05-20 Мотида Фармасьютикал Ко., Лтд. Новое производное гетероциклиден ацетамида
KR20090031898A (ko) * 2006-07-13 2009-03-30 교와 핫꼬 기린 가부시키가이샤 펜타디엔아미드 유도체
CN101595094B (zh) 2006-12-27 2013-02-20 塞诺菲-安万特股份有限公司 环烷基胺取代的异喹诺酮衍生物
WO2012072512A1 (en) * 2010-11-29 2012-06-07 Glaxo Group Limited N-cyclobutyl-imidazopyridine or -pyrazolopyridine carboxamides as trpv1 antagonists
DE102010052781A1 (de) * 2010-11-30 2012-05-31 Trw Automotive Gmbh Befestigungsvorrichtung und Befestigungsbaugruppe zur Befestigung eines Gasgenerators und Fahrzeuginsassenrückhaltesystem
WO2012134943A1 (en) 2011-03-25 2012-10-04 Abbott Laboratories Trpv1 antagonists
US8754101B2 (en) 2011-04-11 2014-06-17 Glaxo Group Limited N-cyclobutyl-imidazopyridine-methylamine as TRPV1 antagonists
WO2017079162A1 (en) 2015-11-02 2017-05-11 Castar, Inc Method of immersive rendering for wide field of view
US10269906B2 (en) * 2016-11-30 2019-04-23 Taiwan Semiconductor Manufacturing Co., Ltd. Semiconductor device having two spacers
WO2018151678A1 (en) 2017-02-15 2018-08-23 Agency For Science, Technology And Research Compounds for treatment of cancer and epigenetics
US11542248B2 (en) 2017-06-08 2023-01-03 Kura Oncology, Inc. Methods and compositions for inhibiting the interaction of menin with MLL proteins
JP7594787B2 (ja) 2018-12-07 2024-12-05 ユニバーシティ オブ メリーランド、ボルチモア 非ATP/触媒部位p38マイトジェン活性化プロテインキナーゼ阻害剤
AR125196A1 (es) * 2021-03-26 2023-06-21 Novartis Ag Derivados de ciclobutilo 1,3-sustituidos y sus usos

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