JP2024506047A5 - - Google Patents
Info
- Publication number
- JP2024506047A5 JP2024506047A5 JP2023547798A JP2023547798A JP2024506047A5 JP 2024506047 A5 JP2024506047 A5 JP 2024506047A5 JP 2023547798 A JP2023547798 A JP 2023547798A JP 2023547798 A JP2023547798 A JP 2023547798A JP 2024506047 A5 JP2024506047 A5 JP 2024506047A5
- Authority
- JP
- Japan
- Prior art keywords
- thiazole
- carboxamide
- benzo
- ring
- alkoxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
Links
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB2102088.8 | 2021-02-15 | ||
| GBGB2102088.8A GB202102088D0 (en) | 2021-02-15 | 2021-02-15 | Compounds and their use as pde4 activators |
| PCT/GB2022/050402 WO2022172037A1 (en) | 2021-02-15 | 2022-02-15 | Compounds and their use as pde4 activators |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| JP2024506047A JP2024506047A (ja) | 2024-02-08 |
| JP2024506047A5 true JP2024506047A5 (https=) | 2025-02-03 |
Family
ID=75338983
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| JP2023547798A Pending JP2024506047A (ja) | 2021-02-15 | 2022-02-15 | 化合物およびｐｄｅ４活性剤としてのそれらの使用 |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US20240150339A1 (https=) |
| EP (1) | EP4291557A1 (https=) |
| JP (1) | JP2024506047A (https=) |
| CN (1) | CN116848107A (https=) |
| CA (1) | CA3206667A1 (https=) |
| GB (1) | GB202102088D0 (https=) |
| WO (1) | WO2022172037A1 (https=) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MX2024001294A (es) * | 2021-08-03 | 2024-02-13 | Cytokinetics Inc | Proceso para la preparacion de aficamten. |
| GB202211999D0 (en) * | 2022-08-17 | 2022-09-28 | Mironid Ltd | Compounds and their use as PDE4 activators |
| WO2025194063A1 (en) * | 2024-03-15 | 2025-09-18 | Board Of Trustees Of Northern Illinois University | Benzothiazole derivatives for treating diseases |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN101454318A (zh) * | 2006-03-22 | 2009-06-10 | 阿斯利康(瑞典)有限公司 | 吡啶并嘧啶衍生物及其作为pde4抑制剂的用途 |
| US20090130076A1 (en) * | 2007-11-21 | 2009-05-21 | Decode Genetics Ehf | Substituted benzoazole pde4 inhibitors for treating pulmonary and cardiovascular disorders |
| TW201215607A (en) * | 2010-07-02 | 2012-04-16 | Lundbeck & Co As H | Aryl-and heteroarylamid derivatives as PDE10A enzyme inhibitor |
| KR102214222B1 (ko) * | 2013-07-10 | 2021-02-08 | 메이지 세이카 파루마 가부시키가이샤 | 신규 pde4 저해제 |
| TWI652014B (zh) * | 2013-09-13 | 2019-03-01 | 美商艾佛艾姆希公司 | 雜環取代之雙環唑殺蟲劑 |
| BR112017011661A2 (pt) * | 2014-12-02 | 2018-03-06 | Bayer Cropscience Aktiengesellschaft | compostos bicíclicos como agentes de controle de pragas. |
| GB201504763D0 (en) | 2015-03-20 | 2015-05-06 | Mironid Ltd | Compounds and uses |
| GB201616439D0 (en) | 2016-09-28 | 2016-11-09 | Mironid Limited | Compounds and uses |
| GB201805527D0 (en) | 2018-04-04 | 2018-05-16 | Mironid Ltd | Compounds and their use as pde4 activators |
| JP6815566B2 (ja) * | 2018-06-27 | 2021-01-20 | Ｍｅｉｊｉ Ｓｅｉｋａファルマ株式会社 | 炎症性疾患、自己免疫疾患、線維化疾患、及びがん疾患の治療剤 |
-
2021
- 2021-02-15 GB GBGB2102088.8A patent/GB202102088D0/en not_active Ceased
-
2022
- 2022-02-15 EP EP22706880.6A patent/EP4291557A1/en active Pending
- 2022-02-15 US US18/276,309 patent/US20240150339A1/en active Pending
- 2022-02-15 JP JP2023547798A patent/JP2024506047A/ja active Pending
- 2022-02-15 CN CN202280015113.1A patent/CN116848107A/zh active Pending
- 2022-02-15 CA CA3206667A patent/CA3206667A1/en active Pending
- 2022-02-15 WO PCT/GB2022/050402 patent/WO2022172037A1/en not_active Ceased
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