|
WO1990005723A1
(fr)
|
1988-11-24 |
1990-05-31 |
Yoshitomi Pharmaceutical Industries, Ltd. |
Composes de trans-4-amino(alkyl)-1-pyridylcarbamoylcyclohexane et leur utilisation en medecine
|
|
PT868186E
(pt)
|
1995-12-21 |
2005-05-31 |
Alcon Lab Inc |
Utilizacao de certos compostos de isoquinolinossulfonilo para tratamento de glaucoma e isquemia ocular
|
|
NZ513800A
(en)
|
1996-08-12 |
2001-09-28 |
Welfide Corp |
Treatment of diseases using Rho kinase inhibitors
|
|
DE69922494T2
(de)
|
1998-02-04 |
2005-05-25 |
Banyu Pharmaceutical Co., Ltd. |
Zyklische n-acylamin-derivate
|
|
JP4212149B2
(ja)
|
1998-06-11 |
2009-01-21 |
株式会社デ・ウエスタン・セラピテクス研究所 |
医薬
|
|
AU5198199A
(en)
|
1998-08-17 |
2000-03-06 |
Senju Pharmaceutical Co., Ltd. |
Preventives/remedies for glaucoma
|
|
US7217722B2
(en)
|
2000-02-01 |
2007-05-15 |
Kirin Beer Kabushiki Kaisha |
Nitrogen-containing compounds having kinase inhibitory activity and drugs containing the same
|
|
ATE273695T1
(de)
|
2000-06-28 |
2004-09-15 |
Smithkline Beecham Plc |
Nassvermahlung
|
|
US20030125344A1
(en)
|
2001-03-23 |
2003-07-03 |
Bayer Corporation |
Rho-kinase inhibitors
|
|
MXPA03008659A
(es)
|
2001-03-23 |
2005-04-08 |
Bayer Ag |
Inhibidores de rho-cinasa.
|
|
JPWO2002100833A1
(ja)
|
2001-06-12 |
2004-09-24 |
住友製薬株式会社 |
Rhoキナーゼ阻害剤
|
|
WO2005080394A1
(en)
|
2004-02-24 |
2005-09-01 |
Bioaxone Therapeutique Inc. |
4-substituted piperidine derivatives
|
|
TWI367098B
(en)
|
2004-12-23 |
2012-07-01 |
Kowa Co |
Treating agent for glaucoma
|
|
EP2455382B1
(en)
|
2005-12-13 |
2016-10-26 |
Incyte Holdings Corporation |
Heteroaryl substituted pyrrolo[2,3-b]pyridines and pyrrolo[2,3-b]pyrimidines as Janus kinase inhibitors
|
|
EP3070090B1
(en)
|
2007-06-13 |
2018-12-12 |
Incyte Holdings Corporation |
Use of salts of the janus kinase inhibitor (r)-3-(4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h- pyrazol-1-yl)-3- cyclopentylpropanenitrile
|
|
EP3053913B1
(en)
|
2009-05-01 |
2018-03-07 |
Aerie Pharmaceuticals, Inc. |
Dual mechanism inhibitors for the treatment of disease
|
|
JP5775070B2
(ja)
|
2009-05-22 |
2015-09-09 |
インサイト・コーポレイションIncyte Corporation |
ヤヌスキナーゼ阻害剤としてのピラゾール−4−イル−ピロロ[2,3−d]ピリミジンおよびピロール−3−イル−ピロロ[2,3−d]ピリミジンのN−(ヘテロ)アリール−ピロリジン誘導体
|
|
AR078012A1
(es)
|
2009-09-01 |
2011-10-05 |
Incyte Corp |
Derivados heterociclicos de las pirazol-4-il- pirrolo (2,3-d) pirimidinas como inhibidores de la quinasa janus
|
|
PT3354652T
(pt)
|
2010-03-10 |
2020-07-20 |
Incyte Holdings Corp |
Derivados de piperidin-4-ilazetidina como inibidores de jak1
|
|
CA2818542A1
(en)
|
2010-11-19 |
2012-05-24 |
Incyte Corporation |
Cyclobutyl substituted pyrrolopyridine and pyrrolopyrimidine derivatives as jak inhibitors
|
|
WO2012068440A1
(en)
|
2010-11-19 |
2012-05-24 |
Incyte Corporation |
Heterocyclic-substituted pyrrolopyridines and pyrrolopyrimidines as jak inhibitors
|
|
MY165963A
(en)
|
2011-06-20 |
2018-05-18 |
Incyte Holdings Corp |
Azetidinyl phenyl, pyridyl or pyrazinyl carboxamide derivatives as jak inhibitors
|
|
TW201313721A
(zh)
|
2011-08-18 |
2013-04-01 |
Incyte Corp |
作為jak抑制劑之環己基氮雜環丁烷衍生物
|
|
UA111854C2
(uk)
|
2011-09-07 |
2016-06-24 |
Інсайт Холдінгс Корпорейшн |
Способи і проміжні сполуки для отримання інгібіторів jak
|
|
TW201406761A
(zh)
|
2012-05-18 |
2014-02-16 |
Incyte Corp |
做爲jak抑制劑之哌啶基環丁基取代之吡咯并吡啶及吡咯并嘧啶衍生物
|
|
AU2013274030B2
(en)
|
2012-06-15 |
2016-07-07 |
Sun Pharmaceutical Industries, Inc. |
Deuterated derivatives of ruxolitinib
|
|
CA2880083A1
(en)
|
2012-08-17 |
2014-02-20 |
Concert Pharmaceuticals, Inc. |
Deuterated baricitinib
|
|
CN113620933A
(zh)
|
2012-10-05 |
2021-11-09 |
卡德门企业有限公司 |
Rho激酶抑制剂
|
|
CN104918945B
(zh)
|
2012-11-01 |
2018-01-05 |
因赛特公司 |
作为jak抑制剂的三环稠合噻吩衍生物
|
|
WO2014138168A1
(en)
|
2013-03-06 |
2014-09-12 |
Incyte Corporation |
Processes and intermediates for making a jak inhibitor
|
|
SMT201900223T1
(it)
|
2013-05-17 |
2019-07-11 |
Incyte Corp |
Sale di bipirazolo come inibitore di jak
|
|
SG10201801069QA
(en)
|
2013-08-07 |
2018-03-28 |
Incyte Corp |
Sustained release dosage forms for a jak1 inhibitor
|
|
CN106687462A
(zh)
|
2014-04-30 |
2017-05-17 |
因赛特公司 |
Jak1抑制剂的制备方法以及其新形式
|
|
MA55201A
(fr)
*
|
2019-03-05 |
2022-01-12 |
Incyte Corp |
Inhibiteurs de la voie jak1 pour le traitement d'un dysfonctionnement chronique de l'allogreffe pulmonaire
|