JP2024500605A5 - - Google Patents

Info

Publication number
JP2024500605A5
JP2024500605A5 JP2023526518A JP2023526518A JP2024500605A5 JP 2024500605 A5 JP2024500605 A5 JP 2024500605A5 JP 2023526518 A JP2023526518 A JP 2023526518A JP 2023526518 A JP2023526518 A JP 2023526518A JP 2024500605 A5 JP2024500605 A5 JP 2024500605A5
Authority
JP
Japan
Prior art keywords
peptide
receptor
activity
glucagon
gip
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023526518A
Other languages
English (en)
Japanese (ja)
Other versions
JP2024500605A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/KR2021/019791 external-priority patent/WO2022139538A1/ko
Publication of JP2024500605A publication Critical patent/JP2024500605A/ja
Publication of JP2024500605A5 publication Critical patent/JP2024500605A5/ja
Pending legal-status Critical Current

Links

JP2023526518A 2020-12-24 2021-12-24 新規なグルカゴン、glp-1及びgip受容体の全てに対して活性を有する三重活性体及びその用途 Pending JP2024500605A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
KR10-2020-0183576 2020-12-24
KR20200183576 2020-12-24
PCT/KR2021/019791 WO2022139538A1 (ko) 2020-12-24 2021-12-24 신규한 글루카곤, glp-1 및 gip 수용체 모두에 활성을 갖는 삼중활성체 및 이의 용도

Publications (2)

Publication Number Publication Date
JP2024500605A JP2024500605A (ja) 2024-01-10
JP2024500605A5 true JP2024500605A5 (https=) 2025-01-08

Family

ID=82159979

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023526518A Pending JP2024500605A (ja) 2020-12-24 2021-12-24 新規なグルカゴン、glp-1及びgip受容体の全てに対して活性を有する三重活性体及びその用途

Country Status (6)

Country Link
US (1) US20230382974A1 (https=)
EP (1) EP4269425A4 (https=)
JP (1) JP2024500605A (https=)
KR (1) KR20220092442A (https=)
CN (1) CN116635050A (https=)
WO (1) WO2022139538A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US12281149B2 (en) 2021-05-13 2025-04-22 Carmot Therapeutics, Inc. Modulators of G-protein coupled receptors
KR20250177377A (ko) * 2024-06-13 2025-12-23 한미약품 주식회사 Glp-1, gip, 및 글루카곤 수용체 모두에 활성을 갖는 삼중 활성체 및 이를 포함하는 당뇨 예방 또는 치료용 약학적 조성물
KR20250177375A (ko) * 2024-06-13 2025-12-23 한미약품 주식회사 Glp-1, gip, 및 글루카곤 수용체 모두에 활성을 갖는 삼중 활성체 및 이를 포함하는 지질 대사 질환 예방 또는 치료용 약학적 조성물

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6096871A (en) 1995-04-14 2000-08-01 Genentech, Inc. Polypeptides altered to contain an epitope from the Fc region of an IgG molecule for increased half-life
JP4046354B2 (ja) 1996-03-18 2008-02-13 ボード オブ リージェンツ,ザ ユニバーシティ オブ テキサス システム 増大した半減期を有する免疫グロブリン様ドメイン
AR092873A1 (es) * 2012-09-26 2015-05-06 Cadila Healthcare Ltd Peptidos como agonistas triples de los receptores de gip, glp-1 y glugagon
CN105829339B (zh) * 2013-11-06 2021-03-12 西兰制药公司 胰高血糖素-glp-1-gip三重激动剂化合物
SG11201805586SA (en) 2015-12-31 2018-07-30 Hanmi Pharmaceutical Co Ltd Triple glucagon/glp-1/gip receptor agonist
CN113453703A (zh) * 2018-12-21 2021-09-28 韩美药品株式会社 包括胰岛素和对胰高血糖素和glp-1和gip受体均具有活性的三重激动剂的药物组合物
WO2020214013A1 (ko) * 2019-04-19 2020-10-22 한미약품 주식회사 글루카곤, glp-1 및 gip 수용체 모두에 활성을 갖는 삼중 활성체 또는 이의 결합체의 고지혈증에 대한 치료적 용도

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