JP2023552864A5 - - Google Patents

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Publication number
JP2023552864A5
JP2023552864A5 JP2023535832A JP2023535832A JP2023552864A5 JP 2023552864 A5 JP2023552864 A5 JP 2023552864A5 JP 2023535832 A JP2023535832 A JP 2023535832A JP 2023535832 A JP2023535832 A JP 2023535832A JP 2023552864 A5 JP2023552864 A5 JP 2023552864A5
Authority
JP
Japan
Prior art keywords
methyl
formula
pyridazin
imidazo
carboxamide
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
JP2023535832A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023552864A (ja
JP7827725B2 (ja
Filing date
Publication date
Priority claimed from GBGB2019702.6A external-priority patent/GB202019702D0/en
Priority claimed from GBGB2109583.1A external-priority patent/GB202109583D0/en
Application filed filed Critical
Priority claimed from PCT/EP2021/084448 external-priority patent/WO2022128584A1/en
Publication of JP2023552864A publication Critical patent/JP2023552864A/ja
Publication of JP2023552864A5 publication Critical patent/JP2023552864A5/ja
Application granted granted Critical
Publication of JP7827725B2 publication Critical patent/JP7827725B2/ja
Active legal-status Critical Current
Anticipated expiration legal-status Critical

Links

JP2023535832A 2020-12-14 2021-12-06 Il-17モジュレータとしてのイミダゾピリダジン誘導体 Active JP7827725B2 (ja)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GBGB2019702.6A GB202019702D0 (en) 2020-12-14 2020-12-14 Therapeutic agents
GB2019702.6 2020-12-14
GB2109583.1 2021-07-02
GBGB2109583.1A GB202109583D0 (en) 2021-07-02 2021-07-02 Therapeutic agents
PCT/EP2021/084448 WO2022128584A1 (en) 2020-12-14 2021-12-06 Imidazopyridazine derivatives as il-17 modulators

Publications (3)

Publication Number Publication Date
JP2023552864A JP2023552864A (ja) 2023-12-19
JP2023552864A5 true JP2023552864A5 (enExample) 2024-11-15
JP7827725B2 JP7827725B2 (ja) 2026-03-10

Family

ID=79164779

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023535832A Active JP7827725B2 (ja) 2020-12-14 2021-12-06 Il-17モジュレータとしてのイミダゾピリダジン誘導体

Country Status (5)

Country Link
US (1) US20240140951A1 (enExample)
EP (1) EP4259631A1 (enExample)
JP (1) JP7827725B2 (enExample)
CA (1) CA3200594A1 (enExample)
WO (1) WO2022128584A1 (enExample)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB201909190D0 (en) * 2019-06-26 2019-08-07 Ucb Biopharma Sprl Therapeutic agents
EP4259631A1 (en) * 2020-12-14 2023-10-18 UCB Biopharma SRL Imidazopyridazine derivatives as il-17 modulators
AR126255A1 (es) 2021-07-01 2023-10-04 UCB Biopharma SRL Derivados de imidazotriazina como moduladores de il-17
WO2023025783A1 (en) 2021-08-23 2023-03-02 Leo Pharma A/S Small molecule modulators of il-17
WO2023111181A1 (en) 2021-12-16 2023-06-22 Leo Pharma A/S Small molecule modulators of il-17
WO2023166172A1 (en) 2022-03-04 2023-09-07 Leo Pharma A/S Small molecule modulators of il-17
GB202210731D0 (en) 2022-07-22 2022-09-07 UCB Biopharma SRL Therapeutic agents
WO2024115662A1 (en) 2022-12-02 2024-06-06 Leo Pharma A/S Small molecule modulators of il-17
WO2024138286A1 (en) * 2022-12-26 2024-07-04 Usynova Pharmaceuticals, Ltd. Il-17a modulators
WO2024188288A2 (en) * 2023-03-14 2024-09-19 Ascletis BioScience Co., Ltd Small molecule modulators of il-17a, methods of making and methods of using thereof
CN121311483A (zh) * 2023-03-28 2026-01-09 詹森药业有限公司 含内酰胺的咪唑并哒嗪il-17抑制剂化合物

Family Cites Families (18)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2009204441B2 (en) 2008-01-09 2015-03-05 The Schepens Eye Research Institute, Inc. Therapeutic compositions for treatment of ocular inflammatory disorders
WO2013116682A1 (en) 2012-02-02 2013-08-08 Ensemble Therapeutics Corporation Macrocyclic compounds for modulating il-17
WO2014066726A2 (en) 2012-10-26 2014-05-01 Ensemble Therapeutics Corporation Compounds for modulating il-17
GB201709456D0 (en) 2017-06-14 2017-07-26 Ucb Biopharma Sprl Therapeutic agents
EP3740478B1 (en) 2018-01-15 2023-11-01 UCB Biopharma SRL Fused imidazole derivatives as il-17 modulators
WO2019223718A1 (zh) 2018-05-22 2019-11-28 成都先导药物开发股份有限公司 一种免疫调节剂
CA3103711A1 (en) 2018-07-12 2020-01-16 UCB Biopharma SRL Spirocyclic indane analogues as il-17 modulators
GB201820166D0 (en) 2018-12-11 2019-01-23 Ucb Biopharma Sprl Therapeutic agents
GB201820165D0 (en) 2018-12-11 2019-01-23 Ucb Biopharma Sprl Therapeutic agents
CN113164448A (zh) 2018-12-19 2021-07-23 利奥制药有限公司 作为il-17的小分子调节剂的氨基酸苯胺类化合物
TW202214648A (zh) 2019-01-07 2022-04-16 美商美國禮來大藥廠 Il-17a抑制劑
US20220162191A1 (en) 2019-03-08 2022-05-26 Leo Pharma A/S Small molecule modulators of il-17
GB201909190D0 (en) 2019-06-26 2019-08-07 Ucb Biopharma Sprl Therapeutic agents
GB201909194D0 (en) 2019-06-26 2019-08-07 Ucb Biopharma Sprl Therapeutic agents
GB201909191D0 (en) 2019-06-26 2019-08-07 Ucb Biopharma Sprl Therapeutic agents
CA3181418A1 (en) 2020-04-30 2021-11-04 Janssen Pharmaceutica Nv Methods of identifying modulators of the il-17 pathway
KR20230019507A (ko) 2020-04-30 2023-02-08 얀센 파마슈티카 엔.브이. Il-17의 조절제로서의 이미다조피리다진
EP4259631A1 (en) * 2020-12-14 2023-10-18 UCB Biopharma SRL Imidazopyridazine derivatives as il-17 modulators

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