JP2023539136A5 - - Google Patents

Info

Publication number
JP2023539136A5
JP2023539136A5 JP2023512161A JP2023512161A JP2023539136A5 JP 2023539136 A5 JP2023539136 A5 JP 2023539136A5 JP 2023512161 A JP2023512161 A JP 2023512161A JP 2023512161 A JP2023512161 A JP 2023512161A JP 2023539136 A5 JP2023539136 A5 JP 2023539136A5
Authority
JP
Japan
Prior art keywords
phenyl
methyl
pyridine
pyrrolo
methylsulfonyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2023512161A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023539136A (ja
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/046475 external-priority patent/WO2022040293A1/en
Publication of JP2023539136A publication Critical patent/JP2023539136A/ja
Publication of JP2023539136A5 publication Critical patent/JP2023539136A5/ja
Pending legal-status Critical Current

Links

JP2023512161A 2020-08-19 2021-08-18 Tlr9阻害剤として有用な置換ヘテロアリール化合物 Pending JP2023539136A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063067389P 2020-08-19 2020-08-19
US63/067,389 2020-08-19
PCT/US2021/046475 WO2022040293A1 (en) 2020-08-19 2021-08-18 Substituted heteroaryl compounds useful as inhibitors of tlr9

Publications (2)

Publication Number Publication Date
JP2023539136A JP2023539136A (ja) 2023-09-13
JP2023539136A5 true JP2023539136A5 (https=) 2024-08-26

Family

ID=77726550

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023512161A Pending JP2023539136A (ja) 2020-08-19 2021-08-18 Tlr9阻害剤として有用な置換ヘテロアリール化合物

Country Status (16)

Country Link
US (1) US20230322770A1 (https=)
EP (1) EP4200015B1 (https=)
JP (1) JP2023539136A (https=)
KR (1) KR20230052930A (https=)
CN (1) CN115956077A (https=)
AR (1) AR123284A1 (https=)
AU (1) AU2021328362A1 (https=)
BR (1) BR112023002662A2 (https=)
CA (1) CA3189816A1 (https=)
CL (1) CL2023000428A1 (https=)
CO (1) CO2023001670A2 (https=)
IL (1) IL300696A (https=)
MX (1) MX2023001883A (https=)
PE (1) PE20231318A1 (https=)
TW (1) TW202227431A (https=)
WO (1) WO2022040293A1 (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI838670B (zh) * 2020-12-22 2024-04-11 美商基利科學股份有限公司 經取代之吲哚化合物
TWI887510B (zh) * 2020-12-22 2025-06-21 美商基利科學股份有限公司 6-取代之吲哚化合物
KR20230171469A (ko) 2021-04-16 2023-12-20 길리애드 사이언시즈, 인코포레이티드 티에노피롤 화합물
EP4398989A1 (en) 2021-09-10 2024-07-17 Gilead Sciences, Inc. Thienopyrrole compounds
KR20240148414A (ko) * 2022-02-18 2024-10-11 브리스톨-마이어스 스큅 컴퍼니 Tlr9의 억제제로서 유용한 치환된 이미다조피리디닐 화합물
WO2024102886A1 (en) * 2022-11-10 2024-05-16 Bristol-Myers Squibb Company Substituted benzimidazole compounds useful as inhibitors of tlr9
CN120152957A (zh) * 2022-11-10 2025-06-13 百时美施贵宝公司 用作tlr9抑制剂的经取代的喹诺酮

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20130158049A1 (en) * 2011-12-20 2013-06-20 Hoffmann-La Roche Inc. 7-azaindole inhibitors of crac
EP3080124A1 (en) * 2013-12-13 2016-10-19 Takeda Pharmaceutical Company Limited Pyrrolo[3,2-c]pyridine derivatives as tlr inhibitors
AR103232A1 (es) * 2014-12-22 2017-04-26 Bristol Myers Squibb Co ANTAGONISTAS DE TGFbR
FI3728252T3 (fi) * 2017-12-18 2023-10-18 Bristol Myers Squibb Co 4-atsaindoliyhdisteitä
WO2019126082A1 (en) * 2017-12-19 2019-06-27 Bristol-Myers Squibb Company 6-azaindole compounds
CA3085942A1 (en) * 2017-12-20 2019-06-27 Bristol-Myers Squibb Company Aryl and heteroaryl substituted indole compounds

Similar Documents

Publication Publication Date Title
JP2023539136A5 (https=)
JP2023538608A5 (https=)
RU2610262C2 (ru) ХИНОЛИНКАРБОКСАМИДНЫЕ И ХИНОЛИНКАРБОНИТРИЛЬНЫЕ ПРОИЗВОДНЫЕ В КАЧЕСТВЕ mGLuR2-НЕГАТИВНЫХ АЛЛОСТЕРИЧЕСКИХ МОДУЛЯТОРОВ, КОМПОЗИЦИИ И ИХ ПРИМЕНЕНИЕ
CN110003200B (zh) P2x7调节剂
JP2022531801A5 (https=)
US8536194B2 (en) Pyrazolopyridine derivates
JP2012525395A5 (https=)
RU2018112237A (ru) Новые бициклические соединения в качестве дуальных ингибиторов atx/ca
EA032609B1 (ru) Соединения аминопиримидинила в качестве ингибиторов jak
CN104725356B (zh) 氮杂环衍生物及其在药物中的应用
JP2013539777A5 (https=)
RU2016102137A (ru) Первичные карбоксамиды в качестве ингибиторов bik
HRP20192323T1 (hr) Novi derivati dihidrokinolin-2-ona
JP2013523884A5 (https=)
JP2005539000A5 (https=)
JP2023021316A (ja) ピリジンアミン-ピリドンおよびピリミジンアミン-ピリドン化合物
JP2020503302A5 (https=)
JP2019529443A5 (https=)
JP2014530237A5 (https=)
IL300696A (en) ALTERNATIVE HETEROARYL COMPOUNDS ARE USEFUL AS TLR9 INHIBITORS
JP2011519891A5 (https=)
TW202214233A (zh) 可做為tlr9抑制劑之經取代雜芳基化合物
JP2020529419A5 (https=)
JP2022505707A5 (https=)
JP2021501183A5 (https=)