JP2023539136A5 - - Google Patents

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Publication number
JP2023539136A5
JP2023539136A5 JP2023512161A JP2023512161A JP2023539136A5 JP 2023539136 A5 JP2023539136 A5 JP 2023539136A5 JP 2023512161 A JP2023512161 A JP 2023512161A JP 2023512161 A JP2023512161 A JP 2023512161A JP 2023539136 A5 JP2023539136 A5 JP 2023539136A5
Authority
JP
Japan
Application number
JP2023512161A
Other languages
Japanese (ja)
Other versions
JP2023539136A (ja
JPWO2022040293A5 (https=
Filing date
Publication date
Application filed filed Critical
Priority claimed from PCT/US2021/046475 external-priority patent/WO2022040293A1/en
Publication of JP2023539136A publication Critical patent/JP2023539136A/ja
Publication of JP2023539136A5 publication Critical patent/JP2023539136A5/ja
Publication of JPWO2022040293A5 publication Critical patent/JPWO2022040293A5/ja
Pending legal-status Critical Current

Links

JP2023512161A 2020-08-19 2021-08-18 Tlr9阻害剤として有用な置換ヘテロアリール化合物 Pending JP2023539136A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US202063067389P 2020-08-19 2020-08-19
US63/067,389 2020-08-19
PCT/US2021/046475 WO2022040293A1 (en) 2020-08-19 2021-08-18 Substituted heteroaryl compounds useful as inhibitors of tlr9

Publications (3)

Publication Number Publication Date
JP2023539136A JP2023539136A (ja) 2023-09-13
JP2023539136A5 true JP2023539136A5 (https=) 2024-08-26
JPWO2022040293A5 JPWO2022040293A5 (https=) 2024-08-26

Family

ID=77726550

Family Applications (1)

Application Number Title Priority Date Filing Date
JP2023512161A Pending JP2023539136A (ja) 2020-08-19 2021-08-18 Tlr9阻害剤として有用な置換ヘテロアリール化合物

Country Status (16)

Country Link
US (1) US20230322770A1 (https=)
EP (1) EP4200015B1 (https=)
JP (1) JP2023539136A (https=)
KR (1) KR20230052930A (https=)
CN (1) CN115956077A (https=)
AR (1) AR123284A1 (https=)
AU (1) AU2021328362A1 (https=)
BR (1) BR112023002662A2 (https=)
CA (1) CA3189816A1 (https=)
CL (1) CL2023000428A1 (https=)
CO (1) CO2023001670A2 (https=)
IL (1) IL300696A (https=)
MX (1) MX2023001883A (https=)
PE (1) PE20231318A1 (https=)
TW (1) TW202227431A (https=)
WO (1) WO2022040293A1 (https=)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2022140325A1 (en) * 2020-12-22 2022-06-30 Gilead Sciences, Inc. 6-substituted indole compounds
TWI838670B (zh) * 2020-12-22 2024-04-11 美商基利科學股份有限公司 經取代之吲哚化合物
CR20230478A (es) 2021-04-16 2023-11-30 Gilead Sciences Inc Compuestos de tienopirrol.
KR20240056747A (ko) 2021-09-10 2024-04-30 길리애드 사이언시즈, 인코포레이티드 티에노피롤 화합물
MX2024009441A (es) * 2022-02-18 2024-08-14 Bristol Myers Squibb Co Compuestos de imidazopiridinilo sustituidos utiles como inhibidores del receptor tipo toll 9 (tlr9).
WO2024102886A1 (en) * 2022-11-10 2024-05-16 Bristol-Myers Squibb Company Substituted benzimidazole compounds useful as inhibitors of tlr9
KR20250094727A (ko) * 2022-11-10 2025-06-25 브리스톨-마이어스 스큅 컴퍼니 Tlr9의 억제제로서 유용한 치환된 퀴놀론 화합물

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2013092467A1 (en) * 2011-12-20 2013-06-27 F. Hoffmann-La Roche Ag 7-azaindole inhibitors of crac
CN105992766A (zh) * 2013-12-13 2016-10-05 武田药品工业株式会社 作为tlr抑制剂的吡咯并[3,2-c]吡啶衍生物
TW201630907A (zh) * 2014-12-22 2016-09-01 必治妥美雅史谷比公司 TGFβR拮抗劑
EA202091484A1 (ru) * 2017-12-18 2021-03-25 Бристол-Маерс Сквибб Компани 4-азаиндольные соединения
JP7304352B2 (ja) * 2017-12-19 2023-07-06 ブリストル-マイヤーズ スクイブ カンパニー 6-アザインドール化合物
KR102730859B1 (ko) * 2017-12-20 2024-11-15 브리스톨-마이어스 스큅 컴퍼니 아릴 및 헤테로아릴 치환된 인돌 화합물

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