JP2023524519A5 - - Google Patents

Info

Publication number
JP2023524519A5
JP2023524519A5 JP2022566661A JP2022566661A JP2023524519A5 JP 2023524519 A5 JP2023524519 A5 JP 2023524519A5 JP 2022566661 A JP2022566661 A JP 2022566661A JP 2022566661 A JP2022566661 A JP 2022566661A JP 2023524519 A5 JP2023524519 A5 JP 2023524519A5
Authority
JP
Japan
Prior art keywords
compound
pharmaceutical composition
formula
hydrogen
alkyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
JP2022566661A
Other languages
English (en)
Japanese (ja)
Other versions
JP2023524519A (ja
Filing date
Publication date
Priority claimed from GBGB2006390.5A external-priority patent/GB202006390D0/en
Application filed filed Critical
Publication of JP2023524519A publication Critical patent/JP2023524519A/ja
Publication of JP2023524519A5 publication Critical patent/JP2023524519A5/ja
Pending legal-status Critical Current

Links

JP2022566661A 2020-04-30 2021-04-30 炎症性腸疾患の治療 Pending JP2023524519A (ja)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB2006390.5 2020-04-30
GBGB2006390.5A GB202006390D0 (en) 2020-04-30 2020-04-30 Novel treatments
PCT/EP2021/061462 WO2021219879A1 (en) 2020-04-30 2021-04-30 Treatments of inflammatory bowel disease

Publications (2)

Publication Number Publication Date
JP2023524519A JP2023524519A (ja) 2023-06-12
JP2023524519A5 true JP2023524519A5 (https=) 2024-05-10

Family

ID=71080611

Family Applications (2)

Application Number Title Priority Date Filing Date
JP2022566660A Active JP7702427B2 (ja) 2020-04-30 2021-04-30 炎症性腸疾患を治療するための5-クロロ-4-ヒドロキシ-1-メチル-2-オキソ-n-フェニル-キノリン-3-カルボキサミドカリウム塩
JP2022566661A Pending JP2023524519A (ja) 2020-04-30 2021-04-30 炎症性腸疾患の治療

Family Applications Before (1)

Application Number Title Priority Date Filing Date
JP2022566660A Active JP7702427B2 (ja) 2020-04-30 2021-04-30 炎症性腸疾患を治療するための5-クロロ-4-ヒドロキシ-1-メチル-2-オキソ-n-フェニル-キノリン-3-カルボキサミドカリウム塩

Country Status (9)

Country Link
US (2) US20230167064A1 (https=)
EP (2) EP4142725A1 (https=)
JP (2) JP7702427B2 (https=)
KR (2) KR20230018386A (https=)
CN (2) CN115768429B (https=)
AU (2) AU2021262514A1 (https=)
CA (2) CA3177000A1 (https=)
GB (2) GB202006390D0 (https=)
WO (2) WO2021219881A1 (https=)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB202006390D0 (en) * 2020-04-30 2020-06-17 Aqilion Ab Novel treatments
CN115836056A (zh) * 2020-05-21 2023-03-21 Stemsynergy疗法有限责任公司 Notch抑制剂及其用途
CN115120727B (zh) * 2022-06-16 2024-02-23 甘肃农业大学 S100a9抑制剂在制备防治c型产气荚膜梭菌感染性腹泻药物中的应用

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE52670B1 (en) * 1981-03-03 1988-01-20 Leo Ab Heterocyclic carboxamides,compositions containing such compounds,and processes for their preparation
SE9400809D0 (sv) * 1994-03-10 1994-03-10 Pharmacia Ab New use of quinoline-3-carboxamide compounds
ES2393814T3 (es) * 2007-04-04 2012-12-28 Sigmoid Pharma Limited Una composición farmacéutica oral
PL2458992T3 (pl) * 2009-07-30 2016-07-29 Teva Pharma Leczenie choroby Leśniowskiego-Crohna z użyciem lakwinimodu
WO2012006538A1 (en) * 2010-07-09 2012-01-12 Teva Pharmaceutical Industries Ltd. Deuterated n-ethyl-n-phenyl-1,2-dihydro-4-hydroxy-5-chloro-1-methyl-2-oxoquinoline-3-carboxamide, salts and uses thereof
EP2590653A4 (en) * 2010-07-09 2014-01-01 Teva Pharma 5-CHLORO-4-HYDROXY-1-METHYL-2-OXO-N-PHENYL-1,2-DIHYDROCHINOLINE-3-CARBOXAMIDE, SALT THEREOF AND APPLICATIONS THEREOF
WO2012050500A1 (en) 2010-10-14 2012-04-19 Lars Pettersson 1,2-dihydro-4-hydroxy-2-oxo-quinoline-3-carboxanilides as ahr activators.
US9200046B2 (en) * 2011-06-29 2015-12-01 Cornell University Reporter system for high throughput screening of compounds and uses thereof
GB202006390D0 (en) * 2020-04-30 2020-06-17 Aqilion Ab Novel treatments

Similar Documents

Publication Publication Date Title
JP2023524519A5 (https=)
CN106573902B (zh) 氨基烷基苯并硫氮杂*衍生物及其用途
CN103492361B (zh) 取代的1-苄基环烷基羧酸及其用途
JP2024504932A5 (https=)
CN1040323C (zh) 噻唑烷衍生物
ES2670571T3 (es) Derivados de pirrolamida sustituidos con glioxamida y su uso como medicamentos para el tratamiento de la hepatitis B
JP2022534426A5 (https=)
RU2008127312A (ru) Мезилатное пролекарство леводопы, его композиции и применение
AR051248A1 (es) Derivados de 3-arilamino piridina
JP2005526011A5 (https=)
JP2008509953A5 (https=)
JP2013500304A5 (https=)
JP2020507589A5 (https=)
RU2008119651A (ru) Производные дикарбоновых кислот и их применение
KR20120055571A (ko) 종양성 또는 자가면역 질환 치료용 전구약물로서의 푸라자노벤즈이미다졸
RU2013120556A (ru) 1,2-гидрокси-2-оксо-хинолин-3-карбоксанилиды в качестве активаторов ahr
TW201538155A (zh) 活性成份輔助組成物及將活性成份化合物遞送給對象之方法
FR2762315A1 (fr) Derives d'amino-acides inhibiteurs des metalloproteases de la matrice extracellulaire et de la liberation du tnf alpha
JP2011520931A (ja) {f−19}標識l−グルタミン酸及びl−グルタミン誘導体(iii)、それらの使用並びにそれらを得る方法
JP7728260B6 (ja) 発毛を促進する化合物の合成
JP2024507140A (ja) 抗菌性化合物
JP2024502178A5 (https=)
WO2006043655A1 (ja) 吸入用医薬組成物
JP7835403B2 (ja) イタコネートおよびメチルイタコネートの新規プロドラッグ
WO2006103274A8 (fr) Inhibiteurs d'age